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Solute carrier family 15 member 2 Inhibitors (IC50, Ki)

Structure
Compound Name
Standard Type
Standard Values (in nM)
CefadroxilIC5066000.0 [1]
CefadroxilKi2500.0 [1], 2800.0 [2], 3019.95 [3]
CyclacillinIC50610000.0 [1]
CyclacillinKi36800.0 [1], 39100.0 [2], 43651.58 [3]
CephalexinKi68200.0 [1], 75857.76 [2]
L-Alanyl-L-alanineKi6000.0 [1], 6025.6 [2]
L-Lysyl-L-alanineKi23000.0 [1], 40738.03 [2]
Ala-LysKi11000.0 [1], 22908.68 [2]
AmpicillinKi1288249.55 [1]
AmoxicillinKi426579.52 [1]
Penicillin gKi10964781.96 [1]
CefotaximeKi19952623.15 [1]
OxacillinKi3311311.21 [1]
CephalothinKi8317637.71 [1]
CefuroximeKi12589254.12 [1]
CloxacillinKi954992.59 [1]
CefaclorKi28840.32 [1]
CefamandoleKi2818382.93 [1]
DicloxacillinKi416869.38 [1]
CefiximeKi2570395.78 [1]
GlycylglycineKi53703.18 [1]
Levulinic acidKi229086.77 [1]
CysteinylglycineKi28840.32 [1]
CefmetazoleKi4265795.19 [1]
GlycylsarcosineKi64000.0 [1]
Cephapirin sodiumKi11220184.54 [1]
CefodizimeKi8912509.38 [1]
d-Alanyl-l-alanineKi128824.96 [1]
CeftibutenKi90000.0 [1]
Alanyl-D-alanineKi269153.48 [1]
CefpodoximeKi30902954.33 [1]
Val-pro-proKi22908.68 [1]
Glycyl-l-histidyl-l-lysineKi3090295.43 [1]
Glycyl-L-alanineKi3467.37 [1]
Ala-Ala-AlaKi18197.01 [1]
Ala-GlyKi7079.46 [1]
H-Phe-phe-OHKi37153.52 [1]
L-Alanyl-L-prolineKi12022.64 [1]
Val-TyrKi2511.89 [1]
Phe-alaKi15848.93 [1]
Phe-glyKi14125.38 [1]
Glycyl-L-histidineKi38904.51 [1]
Asp-AspKi151356.12 [1]
LeucylprolineKi10000.0 [1]
Val-proKi38904.51 [1]
MetampicillinKi724435.96 [1]
Ala-aspKi18000.0 [1]
GlutamylalanineKi30199.52 [1]
H-Met-met-OHKi3019.95 [1]
Trp-TrpKi794.33 [1]
AspartyllysineKi8000.0 [1]
Leucyl-glycyl-glycineKi18197.01 [1]
Isoleucyl-TyrosineKi7943.28 [1]
H-Pro-gly-gly-OHKi10964781.96 [1]
Pro-gluKi2570395.78 [1]
(6R,7R)-8-Oxo-3-(pyridin-1-ium-1-ylmethyl)-7-[(2-thiophen-2-ylacetyl)amino]-5-thia-1-azabicyclo[4.2.0]oct-2-ene-2-carboxylic acidKi8511380.38 [1]
(2S)-2-[[(2S)-2-[[(2S,3S)-2-Amino-3-methylpentanoyl]amino]-3-methylbutanoyl]amino]-3-(4-hydroxyphenyl)propanoic acidKi14125.38 [1]
TrimethionineKi1995.26 [1]
Tyr-AlaKi4365.16 [1]
Val-pheKi3801.89 [1]
Trp-AlaKi3981.07 [1]
TyrosylphenylalanineKi8912.51 [1]
Ala-SerKi6025.6 [1]
Ser-AlaKi7079.46 [1]
Pro-AspKi2089296.13 [1]
H-Trp-Gly-Tyr-OHKi1698.24 [1]
L-Alanyl-L-norleucineKi30902.95 [1]
(S)-2-[(S)-2-((S)-2-Amino-3-methyl-butyrylamino)-propionylamino]-4-methyl-pentanoic acidKi8912.51 [1]
H-Trp-Trp-Trp-OHKi302.0 [1]
H-Pro-Phe-Lys-OHKi891250.94 [1]
(2S)-2-[[(2S)-2-Acetamido-6-aminohexanoyl]amino]propanoic acidKi15848.93 [1]
(2S)-2-[[(2S)-2-[[(2R)-2-Amino-4-methylsulfanylbutanoyl]amino]-4-methylsulfanylbutanoyl]amino]-4-methylsulfanylbutanoic acidKi6025.6 [1]
(2S)-2-[[(2S)-2-[[(2S,3R)-2-[[(2S)-2-Aminopropanoyl]amino]-3-hydroxybutanoyl]amino]propanoyl]amino]propanoic acidKi549540.87 [1]
(2S)-2-[[(2S)-2-[[(2S,3R)-2-[[(2S)-2-[[(2S)-2-Amino-3-phenylpropanoyl]amino]propanoyl]amino]-3-hydroxybutanoyl]amino]propanoyl]amino]propanoic acidKi239883.29 [1]
(2S)-2-[[(2S)-2-[[(2S,3R)-2-[[(2S)-2-[[(2S)-2-Aminopropanoyl]amino]propanoyl]amino]-3-hydroxybutanoyl]amino]propanoyl]amino]propanoic acidKi190546.07 [1]
(2S)-2-[[(2S)-6-Amino-2-(benzylamino)hexanoyl]amino]propanoic acidKi6025.6 [1]
(2S)-2-[[(2S)-2-[[(2S,3R)-2-[[(2S)-2-[[(2S)-2-Amino-3-methylbutanoyl]amino]propanoyl]amino]-3-hydroxybutanoyl]amino]propanoyl]amino]propanoic acidKi109647.82 [1]
H-Ala-Val-Leu-OHKi12022.64 [1]
Ala-Ala-AspKi158489.32 [1]
Cefepime conjugate acidKi10964781.96 [1]



References

This online tool may be cited as follows

MLA

"Quest Database™ Solute carrier family 15 member 2 Inhibitors (IC50, Ki)." AAT Bioquest, Inc.9 May2024https://www.aatbio.com/data-sets/solute-carrier-family-15-member-2-inhibitors-ic50-ki.

APA

AAT Bioquest, Inc. (2024May 9). Quest Database™ Solute carrier family 15 member 2 Inhibitors (IC50, Ki). AAT Bioquest. https://www.aatbio.com/data-sets/solute-carrier-family-15-member-2-inhibitors-ic50-ki.
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