Solute carrier family 2, facilitated glucose transporter member 3 Inhibitors (IC50, Ki)

Structure ▲ ▼	Compound Name ▲ ▼	Standard Type ▲ ▼	Standard Values (in nM) ▲ ▼
	4-[4-(2-Methoxyphenyl)piperazin-1-yl]-1-(4-methylphenyl)-1H-pyrazolo[3,4-d]pyrimidine	IC50	3000.0 [1]
	1-Cyclopentyl-4-[4-(2-methoxyphenyl)piperazin-1-yl]pyrazolo[3,4-d]pyrimidine	IC50	120.0 [1]
	1-(5-Fluoro-2-methoxyphenyl)-4-[4-(2-methoxyphenyl)piperazin-1-yl]pyrazolo[3,4-d]pyrimidine	IC50	320.0 [1]
	1-(3,5-Difluorophenyl)-4-[4-(2-methoxyphenyl)piperazin-1-yl]pyrazolo[3,4-d]pyrimidine	IC50	90.0 [1]
	6-[4-(2-Methoxyphenyl)piperazin-1-yl]-9-phenylpurine	IC50	64.0 [1]
	1-(2-Methoxyphenyl)-4-[4-(2-methoxyphenyl)piperazin-1-yl]pyrazolo[3,4-d]pyrimidine	IC50	110.0 [1]
	4-[4-(2-Methoxyphenyl)piperazin-1-yl]-1-phenylpyrazolo[3,4-b]pyridine	IC50	4000.0 [1]
	4-Methoxy-3-[4-(1-phenylpyrazolo[3,4-d]pyrimidin-4-yl)piperazin-1-yl]benzonitrile	IC50	50.0 [1]
	6-[4-(2-Methoxyphenyl)piperazin-1-yl]-9-phenyl-7H-purin-8-one	IC50	630.0 [1]
	3-[4-[4-(2-Methoxyphenyl)piperazin-1-yl]pyrazolo[3,4-d]pyrimidin-1-yl]benzonitrile	IC50	350.0 [1]
	4-[4-(2-Methoxyphenyl)piperazin-1-yl]-1-(6-methoxypyridin-3-yl)pyrazolo[3,4-d]pyrimidine	IC50	340.0 [1]
	4-[6-(2-Methoxyphenyl)-2,6-diazaspiro[3.3]heptan-2-yl]-1-phenylpyrazolo[3,4-d]pyrimidine	IC50	2200.0 [1]
	1-(3-Methoxyphenyl)-4-[4-(2-methoxyphenyl)piperazin-1-yl]pyrazolo[3,4-d]pyrimidine	IC50	170.0 [1]
	4-[4-[4-(2-Methoxyphenyl)piperazin-1-yl]pyrazolo[3,4-d]pyrimidin-1-yl]benzonitrile	IC50	200.0 [1]
	4-[4-(2-Methoxyphenyl)piperazin-1-yl]-1-phenylpyrazolo[4,3-c]pyridine	IC50	2000.0 [1]
	4-[4-(2-Methoxyphenyl)piperazin-1-yl]-1-(1-phenylethyl)pyrazolo[3,4-d]pyrimidine	IC50	950.0 [1]
	4-[4-(2-Methoxyphenyl)piperazin-1-yl]-1-pyridin-3-ylpyrazolo[3,4-d]pyrimidine	IC50	1500.0 [1]
	4-[4-(2-Methoxyphenyl)piperazin-1-yl]-1-pyridin-4-ylpyrazolo[3,4-d]pyrimidine	IC50	1600.0 [1]
	2-[4-(1-Phenylpyrazolo[3,4-d]pyrimidin-4-yl)piperazin-1-yl]benzonitrile	IC50	2050.0 [1]
	4-[4-(2-Methoxyphenyl)piperazin-1-yl]-7-phenylpyrazolo[3,4-d]triazine	IC50	10000.0 [1]
	1-Phenyl-4-[4-[2-(trifluoromethyl)phenyl]piperazin-1-yl]pyrazolo[3,4-d]pyrimidine	IC50	10000.0 [1]
	4-[4-(3-Fluorophenyl)piperazin-1-yl]-1-phenylpyrazolo[3,4-d]pyrimidine	IC50	540.0 [1]
	3-[4-(1-Phenylpyrazolo[3,4-d]pyrimidin-4-yl)piperazin-1-yl]benzonitrile	IC50	69.0 [1]
	4-[4-(2-Fluoro-6-methoxyphenyl)piperazin-1-yl]-1-phenylpyrazolo[3,4-d]pyrimidine	IC50	1600.0 [1]
	4-[4-(2-Methoxypyridin-3-yl)piperazin-1-yl]-1-phenylpyrazolo[3,4-d]pyrimidine	IC50	680.0 [1]
	4-[4-(3-Methoxypyridin-4-yl)piperazin-1-yl]-1-phenylpyrazolo[3,4-d]pyrimidine	IC50	1510.0 [1]
	1-Phenyl-4-[4-[2-(trifluoromethoxy)phenyl]piperazin-1-yl]pyrazolo[3,4-d]pyrimidine	IC50	10000.0 [1]
	4-[4-(3-Fluoro-2-methoxyphenyl)piperazin-1-yl]-1-phenylpyrazolo[3,4-d]pyrimidine	IC50	10000.0 [1]
	2-Methoxy-3-[4-(1-phenylpyrazolo[3,4-d]pyrimidin-4-yl)piperazin-1-yl]benzonitrile	IC50	540.0 [1]
	4-[4-(4-Methoxypyridin-3-yl)piperazin-1-yl]-1-phenylpyrazolo[3,4-d]pyrimidine	IC50	60.0 [1]
	4-[4-(3-Methoxypyridin-2-yl)piperazin-1-yl]-1-phenylpyrazolo[3,4-d]pyrimidine	IC50	70.0 [1]
	2-[4-(1-Phenylpyrazolo[3,4-d]pyrimidin-4-yl)piperazin-1-yl]cyclohexan-1-ol	IC50	10000.0 [1]
	4-[4-(2-Methoxyphenyl)piperidin-1-yl]-1-phenylpyrazolo[3,4-d]pyrimidine	IC50	10000.0 [1]
	4-[1-(2-Methoxyphenyl)piperidin-4-yl]-1-phenylpyrazolo[3,4-d]pyrimidine	IC50	1200.0 [1]
	4-[4-(2-Methoxyphenyl)-3-methylpiperazin-1-yl]-1-phenylpyrazolo[3,4-d]pyrimidine	IC50	120.0 [1]
	4-[4-(2-Methoxyphenyl)-2-methylpiperazin-1-yl]-1-phenylpyrazolo[3,4-d]pyrimidine	IC50	480.0 [1]
	4-[(1S,4S)-5-(2-Methoxyphenyl)-2,5-diazabicyclo[2.2.1]heptan-2-yl]-1-phenylpyrazolo[3,4-d]pyrimidine	IC50	4100.0 [1]
	4-[(1R,4R)-5-(2-Methoxyphenyl)-2,5-diazabicyclo[2.2.1]heptan-2-yl]-1-phenylpyrazolo[3,4-d]pyrimidine	IC50	10000.0 [1]
	4-[4-(3-Methoxyphenyl)piperazin-1-yl]-1-phenyl-1H-pyrazolo[3,4-d]pyrimidine	IC50	320.0 [1]
	1-(4-Methoxyphenyl)-4-[4-(2-methoxyphenyl)piperazin-1-yl]-1H-pyrazolo[3,4-d]pyrimidine	IC50	170.0 [1]
	4-[4-(2-Methoxyphenyl)piperazino]-1-(3-methylphenyl)-1H-pyrazolo[3,4-d]pyrimidine	IC50	96.0 [1]
	4-[4-(2-Fluorophenyl)piperazin-1-yl]-1-phenyl-1H-pyrazolo[3,4-d]pyrimidine	IC50	680.0 [1]
	4-(4-(2-Methoxyphenyl)piperazin-1-yl)-1-(o-tolyl)-1H-pyrazolo[3,4-d]pyrimidine	IC50	250.0 [1]
	4-(4-(4-Methoxyphenyl)piperazin-1-yl)-1-phenyl-1H-pyrazolo[3,4-d]pyrimidine	IC50	1770.0 [1]
	4-[4-(2-Methoxyphenyl)piperazin-1-yl]-1-phenyl-1H-pyrazolo[3,4-d]pyrimidine	IC50	250.0 [1]
	1-(4-Fluorophenyl)-4-[4-(2-methoxyphenyl)piperazin-1-yl]-1H-pyrazolo[3,4-d]pyrimidine	IC50	46.0 [1]
	4-[4-(2-Methoxyphenyl)piperazin-1-yl]-1-pyridin-2-ylpyrazolo[3,4-d]pyrimidine	IC50	940.0 [1]
	4-[4-(5-Fluoro-2-methoxyphenyl)piperazin-1-yl]-1-phenylpyrazolo[3,4-d]pyrimidine	IC50	10.0 [1]
	7-[4-(2-Methoxyphenyl)piperazin-1-yl]-3-phenyltriazolo[4,5-d]pyrimidine	IC50	430.0 [1]
	2-[4-(1-Phenylpyrazolo[3,4-d]pyrimidin-4-yl)piperazin-1-yl]phenol	IC50	60.0 [1]
	1-(3-Fluorophenyl)-4-[4-(2-methoxyphenyl)piperazin-1-yl]pyrazolo[3,4-d]pyrimidine	IC50	120.0 [1]
	4-[4-(2-Methoxyphenyl)-1,4-diazepan-1-yl]-1-phenylpyrazolo[3,4-d]pyrimidine	IC50	8.0 [1]
	1-(2-Fluorophenyl)-4-[4-(2-methoxyphenyl)piperazin-1-yl]pyrazolo[3,4-d]pyrimidine	IC50	40.0 [1]
	4-Methoxy-3-[4-(1-phenylpyrazolo[3,4-d]pyrimidin-4-yl)piperazin-1-yl]benzamide	IC50	37.0 [1]
	3-Methoxy-4-[4-(1-phenylpyrazolo[3,4-d]pyrimidin-4-yl)piperazin-1-yl]benzonitrile	IC50	170.0 [1]
	4-[4-(4-Fluoro-2-methoxyphenyl)piperazin-1-yl]-1-phenylpyrazolo[3,4-d]pyrimidine	IC50	40.0 [1]

Entire TableStructureCompound NameStandard TypeStandard Values (in nM)

Items per page: 510All1 - 10 of 56 ⟨⟩

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References

This online tool may be cited as follows

MLA	"Quest Database™ Solute carrier family 2, facilitated glucose transporter member 3 Inhibitors (IC50, Ki)." AAT Bioquest, Inc., 9 May. 2024, https://www.aatbio.com/data-sets/solute-carrier-family-2-facilitated-glucose-transporter-member-3-inhibitors-ic50-ki.
APA	AAT Bioquest, Inc. (2024, May 9). Quest Database™ Solute carrier family 2, facilitated glucose transporter member 3 Inhibitors (IC50, Ki). AAT Bioquest. https://www.aatbio.com/data-sets/solute-carrier-family-2-facilitated-glucose-transporter-member-3-inhibitors-ic50-ki.
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