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Solute carrier family 22 member 1 Inhibitors (IC50, Ki)

Structure
Compound Name
Standard Type
Standard Values (in nM)
ClonidineIC5018980.0 [1], 22600.0 [2]
ClonidineKi550.0 [1]
ImipramineIC507950.0 [1], 17100.0 [2], 37000.0 [3]
CimetidineIC50100000.0 [1], 149000.0 [2]
CimetidineKi166000.0 [1]
QuinidineIC5023400.0 [1], 113800.0 [2]
QuinidineKi17500.0 [1]
TetraethylammoniumKi158000.0 [1], 161000.0 [2], 163000.0 [3]
DesipramineIC509180.0 [1], 56800.0 [2]
DesipramineKi5360.0 [1]
OndansetronIC5020400.0 [1], 100000.0 [2], 300000.0 [3]
PseudoisocyanineIC50980.0 [1]
PseudoisocyanineKi2730.0 [1], 4400.0 [2]
CorticosteroneIC5021700.0 [1]
CorticosteroneKi7020.0 [1]
VerapamilIC506800.0 [1]
VerapamilKi2900.0 [1]
MetforminIC501230000.0 [1], 2010000.0 [2]
ChlorpromazineIC504300.0 [1], 27000.0 [2]
PrazosinIC501840.0 [1], 9900.0 [2]
QuinineIC5051600.0 [1]
QuinineKi22900.0 [1]
TrimethoprimIC5050680.0 [1], 56800.0 [2]
PhenoxybenzamineIC502720.0 [1], 15100.0 [2]
VecuroniumKi120000.0 [1], 232000.0 [2]
TacrineIC5021720.0 [1], 83000.0 [2]
DisopyramideIC5081700.0 [1], 100000.0 [2]
PropafenoneIC5011100.0 [1], 15540.0 [2]
TetrabutylammoniumIC5052000.0 [1]
TetrabutylammoniumKi29600.0 [1]
OrphenadrineIC5012600.0 [1], 100000.0 [2]
BithionolIC502230.0 [1], 3900.0 [2]
TetrapropylammoniumIC5090000.0 [1]
TetrapropylammoniumKi102000.0 [1]
EstradiolIC505730.0 [1]
ProgesteroneIC503050.0 [1]
MorphineIC5028000.0 [1]
PropranololIC5063200.0 [1]
AtropineIC5012200.0 [1]
ImatinibIC50107000.0 [1]
HaloperidolIC50141900.0 [1]
MidazolamKi3700.0 [1]
ThiamineIC504354000.0 [1]
IrinotecanIC5020800.0 [1]
ApomorphineIC5020800.0 [1]
DipyridamoleIC5081000.0 [1]
AmilorideIC5057000.0 [1]
AmitriptylineIC5016900.0 [1]
KetoconazoleIC502600.0 [1]
CitalopramIC5018800.0 [1]
DiltiazemIC5012400.0 [1]
ChlorhexidineIC50210.0 [1]
RitonavirIC5033900.0 [1]
ErlotinibIC5016200.0 [1]
MitoxantroneIC5043900.0 [1]
MetoclopramideIC5094800.0 [1]
DobutamineIC504170.0 [1]
PyrimethamineIC5013570.0 [1]
CarvedilolIC503400.0 [1]
ProcainamideKi73900.0 [1]
ClomipramineIC5019300.0 [1]
PromethazineIC5035100.0 [1]
SunitinibIC506100.0 [1]
IndinavirIC50208000.0 [1]
NandroloneIC5035100.0 [1]
GriseofulvinIC507300.0 [1]
UltramIC5052500.0 [1]
ClotrimazoleIC5011970.0 [1]
CyperquatKi12300.0 [1]
FluphenazineIC50110000.0 [1]
PantoprazoleIC50500000.0 [1]
PentamidineIC5022100.0 [1]
MemantineIC5027200.0 [1]
DextromethorphanIC5010450.0 [1]
LoperamideIC5023700.0 [1]
PepcidIC50300000.0 [1]
PhenforminIC5010000.0 [1]
AgmatineKi24000000.0 [1]
AmsacrineIC505000.0 [1]
ProchlorperazineIC5049600.0 [1]
PromazineIC5017200.0 [1]
DoxepinIC5011190.0 [1]
TetramethylammoniumKi12400000.0 [1]
RepaglinideIC509200.0 [1]
OxprenololIC5028600.0 [1]
TerazosinIC5023700.0 [1]
AcebutololKi95800.0 [1]
FlupentixolIC5089500.0 [1]
AlfuzosinIC5014870.0 [1]
EltrombopagKi103000.0 [1]
ChlorprothixeneIC5077800.0 [1]
TrimipramineIC5027700.0 [1]
ClemastineIC504900.0 [1]
N-(2,6-Dichlorobenzylidene)-N'-amidinohydrazineIC504850.0 [1]
N-MethylnicotinamideKi7700000.0 [1]
ClosantelIC503000.0 [1]
NifekalantIC50300000.0 [1]
DichlorophenIC508410.0 [1]
BucindololIC5027200.0 [1]
DenopamineIC5046900.0 [1]



References

This online tool may be cited as follows

MLA

"Quest Database™ Solute carrier family 22 member 1 Inhibitors (IC50, Ki)." AAT Bioquest, Inc.9 May2024https://www.aatbio.com/data-sets/solute-carrier-family-22-member-1-inhibitors-ic50-ki.

APA

AAT Bioquest, Inc. (2024May 9). Quest Database™ Solute carrier family 22 member 1 Inhibitors (IC50, Ki). AAT Bioquest. https://www.aatbio.com/data-sets/solute-carrier-family-22-member-1-inhibitors-ic50-ki.
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