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Solute carrier family 22 member 2 Inhibitors (IC50, Ki)

Structure
Compound Name
Standard Type
Standard Values (in nM)
PrazosinIC5013600.0 [1], 100000.0 [2]
CimetidineIC5023000.0 [1]
CimetidineKi57000.0 [1]
OndansetronIC50890.0 [1], 1700.0 [2]
PepcidIC5036100.0 [1]
PepcidKi1800000.0 [1]
TetramethylammoniumIC50150000.0 [1]
TetramethylammoniumKi180000.0 [1]
PseudoisocyanineIC501130.0 [1]
PseudoisocyanineKi100.0 [1]
MetiprenalineIC50100000.0 [1]
MetiprenalineKi570000.0 [1]
EstradiolIC5030000.0 [1]
ProgesteroneIC5026700.0 [1]
CorticosteroneIC5034200.0 [1]
MetforminIC501700000.0 [1]
ImatinibIC504200.0 [1]
IrinotecanIC502700.0 [1]
RisperidoneIC5011000.0 [1]
Ethinyl estradiolIC502200.0 [1]
ImipramineIC50600.0 [1]
DipyridamoleIC502600.0 [1]
QuinineKi3400.0 [1]
ChlorhexidineIC50400.0 [1]
RitonavirIC5024800.0 [1]
MitoxantroneIC5073300.0 [1]
TetraethylammoniumIC50156000.0 [1]
DesipramineKi16000.0 [1]
PhenoxybenzamineIC504900.0 [1]
TubocurarineIC5078800.0 [1]
CarvedilolIC507500.0 [1]
AripiprazoleIC50239000.0 [1]
TopotecanIC5061000.0 [1]
ProcainamideKi50000.0 [1]
AmantadineIC5023000.0 [1]
DabigatranIC504700.0 [1]
IndinavirIC50142000.0 [1]
VecuroniumIC503500.0 [1]
BuspironeIC5012000.0 [1]
CyperquatKi2400.0 [1]
DomperidoneIC507900.0 [1]
PantoprazoleIC501500.0 [1]
PentamidineIC501200.0 [1]
PimozideIC5034200.0 [1]
TacrineIC50680.0 [1]
DihydroergotamineIC5049900.0 [1]
DisopyramideIC502900.0 [1]
TetrabutylammoniumIC50120000.0 [1]
PhenforminIC5065000.0 [1]
MaravirocIC50255000.0 [1]
GranisetronIC504300.0 [1]
ZafirlukastIC509700.0 [1]
GabexateIC50900.0 [1]
DolutegravirIC501900.0 [1]
OrphenadrineIC502500.0 [1]
RimantadineIC504400.0 [1]
NoscapineIC502600.0 [1]
CamostatIC5016500.0 [1]
EpinastineIC504300.0 [1]
N-MethylnicotinamideKi266000.0 [1]
BithionolIC501900.0 [1]
NifekalantIC5010300.0 [1]
TetrapropylammoniumIC50128000.0 [1]
TetrapentylammoniumKi1500.0 [1]
1-PhenylguanidineIC5089000.0 [1]
1-(3-Chlorophenyl)guanidineIC5060500.0 [1]
MepiperphenidolKi4800.0 [1]
1-(4-Chlorophenyl)guanidineIC5018900.0 [1]
N-p-Tolyl-guanidineIC509300.0 [1]
1-(4-Fluorophenyl)guanidineIC5048300.0 [1]
N-(2-Chloroethyl)-N-methyl-9H-fluoren-9-amineIC50100.0 [1]
1-(4-Bromophenyl)guanidineIC5011300.0 [1]
N-(4-Benzylphenyl)guanidineIC5096200.0 [1]
N-(4-Iodo-phenyl)-guanidineIC504400.0 [1]
1-(4-Tert-Butylphenyl)guanidineIC508300.0 [1]
2-[(3,6-Dimethyl-2-phenyl-4H-pyrimidin-4-yl)methyl]-1-ethylquinolin-1-iumKi210.0 [1]



References

This online tool may be cited as follows

MLA

"Quest Database™ Solute carrier family 22 member 2 Inhibitors (IC50, Ki)." AAT Bioquest, Inc.8 May2024https://www.aatbio.com/data-sets/solute-carrier-family-22-member-2-inhibitors-ic50-ki.

APA

AAT Bioquest, Inc. (2024May 8). Quest Database™ Solute carrier family 22 member 2 Inhibitors (IC50, Ki). AAT Bioquest. https://www.aatbio.com/data-sets/solute-carrier-family-22-member-2-inhibitors-ic50-ki.
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