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Solute carrier family 22 member 8 Inhibitors (IC50, Ki)

Structure
Compound Name
Standard Type
Standard Values (in nM)
ProbenecidIC504930.0 [1]
ProbenecidKi4410.0 [1], 9000.0 [2], 29800.0 [3]
CimetidineIC5092400.0 [1]
CimetidineKi53000.0 [1]
PiroxicamKi4880.0 [1], 1200000.0 [2]
CilastatinIC50249000.0 [1]
CilastatinKi231000.0 [1]
Indoxyl sulfateKi168700.0 [1], 169000.0 [2]
CefadroxilKi8620.0 [1]
BetamipronIC509920.0 [1]
BetamipronKi48300.0 [1]
IndomethacinKi5950.0 [1]
Uric acidKi275000.0 [1]
IbuprofenKi1170000.0 [1]
Salicylic acidKi1020000.0 [1]
Penicillin gKi97600.0 [1]
PravastatinIC5013700.0 [1]
CeftriaxoneKi4390.0 [1]
PhenylbutazoneKi34700.0 [1]
CefotaximeKi290.0 [1]
KetoprofenKi1160000.0 [1]
CefazolinKi550.0 [1]
Aminohippuric acidKi19600.0 [1]
CephalothinKi40.0 [1]
Octanoic acidKi8600.0 [1]
PepcidKi300000.0 [1]
CefoperazoneKi1890.0 [1]
Hippuric acidKi31000.0 [1]
CefaclorIC50120000.0 [1]
CefamandoleKi46.0 [1]
LinagliptinIC50100000.0 [1]
CitrininKi15400.0 [1]
3-AcetoxyindoleKi491000.0 [1]
RolofyllineKi3700.0 [1]
ZonampanelIC506600.0 [1]
(6R,7R)-8-Oxo-3-(pyridin-1-ium-1-ylmethyl)-7-[(2-thiophen-2-ylacetyl)amino]-5-thia-1-azabicyclo[4.2.0]oct-2-ene-2-carboxylic acidKi2460.0 [1]
4-{[1-Methyl-2,4-Dioxo-6-(3-Phenylprop-1-Yn-1-Yl)-1,4-Dihydroquinazolin-3(2h)-Yl]methyl}benzoic AcidIC5018000.0 [1]
4-((6-(4-Methoxybenzylcarbamoyl)-4-oxopyrido[3,4-d]pyrimidin-3(4H)-yl)methyl)benzoic acidIC5059000.0 [1]
4-[[5-[2-[(4-Fluorophenyl)methylcarbamoyl]-6-methylpyridin-4-yl]tetrazol-2-yl]methyl]cyclohexane-1-carboxylic acidIC506000.0 [1]
2-(Trifluoromethyl)-N-[6-(trifluoromethyl)pyridin-3-yl]benzenesulfonamideIC503300.0 [1]
2-(Trifluoromethyl)-N-[5-(trifluoromethyl)pyridin-3-yl]benzenesulfonamideIC503400.0 [1]
CID 86271138IC50500.0 [1]
CID 86294663IC50720.0 [1]



References

This online tool may be cited as follows

MLA

"Quest Database™ Solute carrier family 22 member 8 Inhibitors (IC50, Ki)." AAT Bioquest, Inc.8 May2024https://www.aatbio.com/data-sets/solute-carrier-family-22-member-8-inhibitors-ic50-ki.

APA

AAT Bioquest, Inc. (2024May 8). Quest Database™ Solute carrier family 22 member 8 Inhibitors (IC50, Ki). AAT Bioquest. https://www.aatbio.com/data-sets/solute-carrier-family-22-member-8-inhibitors-ic50-ki.
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