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Solute carrier family 40 member 1 Inhibitors (IC50, Ki)

Structure
Compound Name
Standard Type
Standard Values (in nM)
Benzenesulfonamide, 4-methyl-N-8-quinolinyl-IC5049900.0 [1]
8-(4-Benzenesulfonylamino)quinolineIC504590.0 [1]
5H-Quinolino[8,7-c][1,2]benzothiazine 6,6-dioxideIC502900.0 [1]
2-Nitro-N-quinolin-8-ylbenzenesulfonamideIC502900.0 [1]
2-Amino-N-quinolin-8-yl-benzenesulfonamideIC5020800.0 [1]
2-Amino-N-(2-methylquinolin-8-yl)benzenesulfonamideIC50100000.0 [1]
9-Trifluoromethyl-5H-6-thia-4,5-diaza-chrysene 6,6-dioxideIC50130.0 [1]
2-Amino-N-(6-methoxyquinolin-8-yl)-4-methylbenzenesulfonamideIC50585.0 [1]
2-Nitro-N-quinolin-8-yl-4-(trifluoromethyl)benzenesulfonamideIC50100000.0 [1]
9-Fluoro-5H-6-thia-4,5-diaza-chrysene 6,6-dioxideIC501560.0 [1]
9-Methyl-5H-quinolino[8,7-c][1,2]benzothiazine 6,6-dioxideIC503200.0 [1]
9-Chloro-5H-6-thia-4,5-diaza-chrysene 6,6-dioxideIC50770.0 [1]
9-Methoxy-5H-6-thia-4,5-diaza-chrysene 6,6-dioxideIC501580.0 [1]
5-Bromo-N-quinolin-8-ylthiophene-2-sulfonamideIC506800.0 [1]
N-(2-Methylquinolin-8-yl)benzenesulfonamideIC50100000.0 [1]
2,4-Dichloro-N-quinolin-8-yl-benzenesulfonamideIC50989.0 [1]
4-Methoxy-N-quinolin-8-ylbenzenesulfonamideIC50100000.0 [1]
N-(6-Methoxyquinolin-8-yl)benzenesulfonamideIC506400.0 [1]
4-Chloro-N-(8-quinolinyl)benzenesulfonamideIC503200.0 [1]
N-(5,7-Dichloroquinolin-8-yl)-4-methylbenzenesulfonamideIC5079000.0 [1]
N-(6-Fluoroquinolin-8-yl)-4-(trifluoromethyl)benzenesulfonamideIC5025000.0 [1]
1-[2-Fluoro-5-(3-methyl-2,2-dioxo-1,4-dihydropyrido[3,2-h][2,1,3]benzothiadiazin-4-yl)phenyl]ethanoneIC505430.0 [1]
N-(7-Hydroxyquinolin-8-yl)benzenesulfonamideIC50100000.0 [1]
N-(5,7-Dichloroquinolin-8-yl)-2,4,6-trimethylbenzenesulfonamideIC50100000.0 [1]
2-Amino-4-methoxy-N-quinolin-8-ylbenzenesulfonamideIC50100000.0 [1]
3-Methyl-5H-6-thia-4,5-diaza-chrysene 6,6-dioxideIC50100000.0 [1]
4-Methoxy-2-nitro-N-(quinolin-8-yl)benzene-1-sulfonamideIC501810.0 [1]
2-Amino-N-quinolin-8-yl-4-(trifluoromethyl)benzenesulfonamideIC50760.0 [1]
2-Amino-4-methyl-N-quinolin-8-ylbenzenesulfonamideIC50300.0 [1]
4-Fluoro-2-nitro-N-quinolin-8-ylbenzenesulfonamideIC50920.0 [1]
2-Amino-4-fluoro-N-quinolin-8-ylbenzenesulfonamideIC503940.0 [1]
12-Chloro-5H-6-thia-4,5-diaza-chrysene 6,6-dioxideIC50320.0 [1]
12-Bromo-5H-6-thia-4,5-diaza-chrysene 6,6-dioxideIC5012600.0 [1]
2-Amino-4-methoxy-N-(2-methylquinolin-8-yl)benzenesulfonamideIC50100000.0 [1]
N-(Quinolin-8-yl)-2-(trifluoromethoxy)benzene-1-sulfonamideIC502500.0 [1]
N-Quinolin-8-ylpyridine-2-sulfonamideIC501890.0 [1]
8-Methoxy-5H-6-thia-4,5-diaza-chrysene 6,6-dioxideIC502110.0 [1]
8-Trifluoromethyl-5H-6-thia-4,5-diaza-chrysene 6,6-dioxideIC502340.0 [1]
8-Methyl-5H-6-thia-4,5-diaza-chrysene 6,6-dioxideIC50360.0 [1]
8-Fluoro-5H-6-thia-4,5-diaza-chrysene 6,6-dioxideIC501620.0 [1]
N-Quinolin-8-ylpyridine-3-sulfonamideIC503640.0 [1]
2,6-Dichloro-N-quinolin-8-ylbenzenesulfonamideIC50100000.0 [1]
2-Cyano-N-quinolin-8-ylbenzenesulfonamideIC50815.0 [1]
Methyl 3-[(quinolin-8-yl)sulfamoyl]benzoateIC501420.0 [1]
N-Quinolin-8-yl-3-(trifluoromethoxy)benzenesulfonamideIC501200.0 [1]
N-(5-Chloroquinolin-8-yl)benzenesulfonamideIC501670.0 [1]
2-Chloro-N-(quinolin-8-yl)benzene-1-sulfonamideIC508000.0 [1]
2,6-Difluoro-N-quinolin-8-ylbenzenesulfonamideIC501140.0 [1]
N-(8-Quinolinyl)-3-(trifluoromethyl)benzenesulfonamideIC50720.0 [1]
2-Methyl-N-(8-quinolinyl)benzenesulfonamideIC50100000.0 [1]
N-(5-Bromoquinolin-8-yl)benzenesulfonamideIC50100000.0 [1]
3-Methyl-N-(8-quinolinyl)benzenesulfonamideIC502090.0 [1]
2-Methoxy-N-quinolin-8-ylbenzenesulfonamideIC50100000.0 [1]
1-[4-(4-Fluorophenyl)-3-methyl-2,2-dioxo-1,4-dihydropyrido[3,2-h][2,1,3]benzothiadiazin-6-yl]ethanoneIC50250.0 [1]
1-(3,4-Difluoro-phenyl)-2-methyl-1,4-dihydro-2H-3-thia-2,4,5-triaza-phenanthrene 3,3-dioxideIC50250.0 [1]
N-(7-Methylquinolin-8-yl)benzenesulfonamideIC50100000.0 [1]
N-(6-Chloroquinolin-8-yl)benzenesulfonamideIC50100000.0 [1]
N-(3-Methylquinolin-8-yl)benzenesulfonamideIC50610.0 [1]
2,4,6-Trichloro-N-quinolin-8-ylbenzenesulfonamideIC50857.0 [1]
2-Methyl-N-[2-(quinolin-8-ylsulfamoyl)phenyl]propanamideIC5024600.0 [1]
2,2,2-Trifluoro-N-[2-(quinolin-8-ylsulfamoyl)phenyl]acetamideIC50307.0 [1]
4-Chloro-N-(5-chloroquinolin-8-yl)-2-fluorobenzenesulfonamideIC501380.0 [1]
CID 60163923IC501750.0 [1]
N-(6-Methoxyquinolin-8-yl)pyridine-3-sulfonamideIC502800.0 [1]
N-(5-Chloroquinolin-8-yl)pyridine-3-sulfonamideIC501780.0 [1]
2-Amino-N-(6-methoxyquinolin-8-yl)-4-(trifluoromethyl)benzenesulfonamideIC501000.0 [1]
2,4-Dichloro-N-(3-methylquinolin-8-yl)benzenesulfonamideIC50100000.0 [1]
N-(3-Methylquinolin-8-yl)pyridine-3-sulfonamideIC501390.0 [1]
N-(5-Chloro-6-methylquinolin-8-yl)benzenesulfonamideIC50100000.0 [1]
N-(7-Chloroquinolin-8-yl)benzenesulfonamideIC50100000.0 [1]
N-(7-Methoxyquinolin-8-yl)benzenesulfonamideIC50100000.0 [1]
8,9-Dimethyl-5H-6-thia-4,5-diaza-chrysene 6,6-dioxideIC504020.0 [1]
12-Methyl-5H-6-thia-4,5-diaza-chrysene 6,6-dioxideIC50599.0 [1]
11-Methoxy-5H-6-thia-4,5-diaza-chrysene 6,6-dioxideIC50100000.0 [1]
1-Methoxy-9-trifluoromethyl-5H-6-thia-4,5-diaza-chrysene 6,6-dioxideIC50979.0 [1]
2-Phenyl-1,4-dihydro-2H-3-thia-2,4,5-triaza-phenanthrene 3,3-dioxideIC50460.0 [1]
1,4-Dihydro-2H-3-thia-2,4,5-triaza-phenanthrene 3,3-dioxideIC5039500.0 [1]
2-Methyl-1-phenyl-1,4-dihydro-2H-3-thia-2,4,5-triaza-phenanthrene 3,3-dioxideIC50870.0 [1]
N-Quinolin-8-yl-1,3-thiazole-2-sulfonamideIC504580.0 [1]
N-Quinolin-8-ylpyrazine-2-sulfonamideIC501910.0 [1]
N-[6-(Trifluoromethoxy)quinolin-8-yl]-6-(trifluoromethyl)pyridine-3-sulfonamideIC5012500.0 [1]
6-(Trifluoromethyl)-N-[5-(trifluoromethyl)quinolin-8-yl]pyridine-3-sulfonamideIC5025000.0 [1]
N-[5-(Trifluoromethyl)quinolin-8-yl]pyridine-2-sulfonamideIC50460.0 [1]
N-[6-(Trifluoromethoxy)quinolin-8-yl]pyridine-2-sulfonamideIC501090.0 [1]
N-(6-Fluoroquinolin-8-yl)pyridine-2-sulfonamideIC502370.0 [1]
6-Cyano-N-[6-(trifluoromethoxy)quinolin-8-yl]pyridine-3-sulfonamideIC502110.0 [1]
6-Cyano-N-(6-fluoroquinolin-8-yl)pyridine-3-sulfonamideIC503750.0 [1]
Methyl 6,6-dioxo-5H-quinolino[8,7-c][1,2]benzothiazine-9-carboxylateIC504180.0 [1]
6,6-Dioxo-5H-quinolino[8,7-c][1,2]benzothiazine-9-carbonitrileIC502830.0 [1]
1-Trifluoromethyl-5H-6-thia-4,5-diaza-chrysene 6,6-dioxideIC5025000.0 [1]
9-Chloro-1-trifluoromethyl-5H-6-thia-4,5-diaza-chrysene 6,6-dioxideIC5025000.0 [1]
12-Trifluoromethyl-5H-6-thia-4,5-diaza-chrysene 6,6-dioxideIC5014100.0 [1]
9-Chloro-12-trifluoromethyl-5H-6-thia-4,5-diaza-chrysene 6,6-dioxideIC508510.0 [1]
3-Chloro-5H-6-thia-4,5-diaza-chrysene 6,6-dioxideIC5025000.0 [1]
8,12-Dichloro-9-fluoro-5H-6-thia-4,5-diaza-chrysene 6,6-dioxideIC5025000.0 [1]
12-Chloro-8,9-difluoro-5H-quinolino[8,7-c][1,2]benzothiazine 6,6-dioxideIC5025000.0 [1]
9-Chloro-6,6-dioxo-5H-quinolino[8,7-c][1,2]benzothiazine-12-carbonitrileIC5025000.0 [1]
3,9-Dichloro-5H-6-thia-4,5-diaza-chrysene 6,6-dioxideIC5025000.0 [1]
12-Chloro-9-methanesulfonyl-5H-6-thia-4,5-diaza-chrysene 6,6-dioxideIC5025000.0 [1]
Methyl 6,6-dioxo-5H-quinolino[8,7-c][1,2]benzothiazine-1-carboxylateIC502940.0 [1]



References

This online tool may be cited as follows

MLA

"Quest Database™ Solute carrier family 40 member 1 Inhibitors (IC50, Ki)." AAT Bioquest, Inc.9 May2024https://www.aatbio.com/data-sets/solute-carrier-family-40-member-1-inhibitors-ic50-ki.

APA

AAT Bioquest, Inc. (2024May 9). Quest Database™ Solute carrier family 40 member 1 Inhibitors (IC50, Ki). AAT Bioquest. https://www.aatbio.com/data-sets/solute-carrier-family-40-member-1-inhibitors-ic50-ki.
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