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Somatostatin receptor 4 Inhibitors (IC50, Ki)

Structure
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Compound Name
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Standard Type
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Standard Values (in nM)
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SomatostatinIC500.08 [1], 1.6 [2], 1.7 [3]
SomatostatinKi0.59 [1], 0.63 [2], 2.0 [3]
(4R,7S,10R,13S,16R,19S,22R,25S,28R,31S,34R,37S)-37-[[2-[[(2S)-2-[[(2S)-6-Amino-2-[[(2S)-2-[[(2S)-2-[[(2S)-2-[[(2S)-1-[(2S)-2-[[(2S)-2-[[(2S)-2-[[(2S)-1-[(2S)-4-amino-2-[[(2S)-2-[[(2S)-4-amino-2-[[(2S)-2-[[(2S)-2-amino-3-hydroxypropanoyl]amino]propanoyl]amino]-4-oxobutanoyl]amino]-3-hydroxypropanoyl]amino]-4-oxobutanoyl]pyrrolidine-2-carbonyl]amino]propanoyl]amino]-4-methylsulfanylbutanoyl]amino]propanoyl]pyrrolidine-2-carbonyl]amino]-5-(diaminomethylideneamino)pentanoyl]amino]-4-carboxybutanoyl]amino]-5-(diaminomethylideneamino)pentanoyl]amino]hexanoyl]amino]propanoyl]amino]acetyl]amino]-19,34-bis(4-aminobutyl)-31-(2-amino-2-oxoethyl)-13,25,28-tribenzyl-10,16-bis[(1R)-1-hydroxyethyl]-7-(hydroxymethyl)-22-(1H-indol-3-ylmethyl)-6,9,12,15,18,21,24,27,30,33,36-undecaoxo-1,2-dithia-5,8,11,14,17,20,23,26,29,32,35-undecazacyclooctatriacontane-4-carboxylic acidIC502.6 [1]
(4R,7S,10R,13S,16R,19S,22R,25S,28R,31S,34R,37S)-37-[[2-[[(2S)-2-[[(2S)-6-Amino-2-[[(2S)-2-[[(2S)-2-[[(2S)-2-[[(2S)-1-[(2S)-2-[[(2S)-2-[[(2S)-2-[[(2S)-1-[(2S)-4-amino-2-[[(2S)-2-[[(2S)-4-amino-2-[[(2S)-2-[[(2S)-2-amino-3-hydroxypropanoyl]amino]propanoyl]amino]-4-oxobutanoyl]amino]-3-hydroxypropanoyl]amino]-4-oxobutanoyl]pyrrolidine-2-carbonyl]amino]propanoyl]amino]-4-methylsulfanylbutanoyl]amino]propanoyl]pyrrolidine-2-carbonyl]amino]-5-(diaminomethylideneamino)pentanoyl]amino]-4-carboxybutanoyl]amino]-5-(diaminomethylideneamino)pentanoyl]amino]hexanoyl]amino]propanoyl]amino]acetyl]amino]-19,34-bis(4-aminobutyl)-31-(2-amino-2-oxoethyl)-13,25,28-tribenzyl-10,16-bis[(1R)-1-hydroxyethyl]-7-(hydroxymethyl)-22-(1H-indol-3-ylmethyl)-6,9,12,15,18,21,24,27,30,33,36-undecaoxo-1,2-dithia-5,8,11,14,17,20,23,26,29,32,35-undecazacyclooctatriacontane-4-carboxylic acidKi5.4 [1]
(4R,7S,10S,13S,16R,19S,22S,25R)-25-Amino-13-(4-aminobutyl)-7,19,22-tribenzyl-10-[(1R)-1-hydroxyethyl]-16-(1H-indol-3-ylmethyl)-6,9,12,15,18,21,24-heptaoxo-1,2-dithia-5,8,11,14,17,20,23-heptazacyclohexacosane-4-carboxylic acidIC501.8 [1]
(4R,7S,10S,13R,16S,19R)-10-(4-Aminobutyl)-19-[[(2R)-2-amino-3-phenylpropanoyl]amino]-16-benzyl-N-[(2S,3R)-1,3-dihydroxybutan-2-yl]-7-[(1R)-1-hydroxyethyl]-13-(1H-indol-3-ylmethyl)-6,9,12,15,18-pentaoxo-1,2-dithia-5,8,11,14,17-pentazacycloicosane-4-carboxamideIC503.0 [1]
(4R,7S,10S,13R,16S,19R)-10-(4-Aminobutyl)-19-[[(2R)-2-amino-3-phenylpropanoyl]amino]-16-benzyl-N-[(2S,3R)-1,3-dihydroxybutan-2-yl]-7-[(1R)-1-hydroxyethyl]-13-(1H-indol-3-ylmethyl)-6,9,12,15,18-pentaoxo-1,2-dithia-5,8,11,14,17-pentazacycloicosane-4-carboxamideKi1000.0 [1], 1904.0 [2]
(4R,7S,10S,13S,16S,19S,22S,25S,28S,31S,34S,37R)-37-[[2-[[(2S)-2-[[(2S)-6-Amino-2-[[(2S)-2-[[(2S)-2-[[(2S)-2-[[(2S)-1-[(2S)-2-[[(2S)-2-[[(2S)-2-[[(2S)-1-[(2S)-4-amino-2-[[(2S)-2-[[(2S)-4-amino-2-[[(2S)-2-[[(2S)-2-amino-3-hydroxypropanoyl]amino]propanoyl]amino]-4-oxobutanoyl]amino]-3-hydroxypropanoyl]amino]-4-oxobutanoyl]pyrrolidine-2-carbonyl]amino]propanoyl]amino]-4-methylsulfanylbutanoyl]amino]propanoyl]pyrrolidine-2-carbonyl]amino]-5-(diaminomethylideneamino)pentanoyl]amino]-4-carboxybutanoyl]amino]-5-(diaminomethylideneamino)pentanoyl]amino]hexanoyl]amino]propanoyl]amino]acetyl]amino]-19,34-bis(4-aminobutyl)-31-(2-amino-2-oxoethyl)-13,25,28-tribenzyl-10,16-bis[(1S)-1-hydroxyethyl]-7-(hydroxymethyl)-22-(1H-indol-2-ylmethyl)-6,9,12,15,18,21,24,27,30,33,36-undecaoxo-1,2-dithia-5,8,11,14,17,20,23,26,29,32,35-undecazacyclooctatriacontane-4-carboxylic acidIC502.5 [1], 3.0 [2], 3.1 [3], 3.8 [4]
SeglitideIC501000.0 [1]
SeglitideKi1000.0 [1], 3200.0 [2]
CID 5311374IC504.2 [1]
1-[3-[(5-Bromopyridin-2-yl)-[(3,4-dichlorophenyl)methyl]amino]propyl]-3-[3-(1H-imidazol-5-yl)propyl]thioureaKi6.0 [1], 17.0 [2]
5-{3,4,5-Tris-benzyloxy-6-[2-(1H-indol-3-yl)-ethoxy]-tetrahydro-pyran-2-ylmethoxy}-pentylamineKi1100.0 [1], 1650.0 [2]
(4R,7S,10S,13S,16S,19S,22S,25R)-25-Amino-13-(4-aminobutyl)-7,19,22-tribenzyl-10-[(1R)-1-hydroxyethyl]-16-(1H-indol-3-ylmethyl)-6,9,12,15,18,21,24-heptaoxo-1,2-dithia-5,8,11,14,17,20,23-heptazacyclohexacosane-4-carboxylic acidIC500.7 [1]
H-DPhe-c[Cys-Phe-DTrp-Lys-Thr-Cys]-Thr-NH2IC501000.0 [1], 10000.0 [2]
5-[[(2R,3R,4S,5R,6R)-5-(1H-Imidazol-5-ylmethoxy)-6-[2-(1H-indol-3-yl)ethoxy]-4-phenylmethoxy-3-(pyridin-3-ylmethoxy)oxan-2-yl]methoxy]pentan-1-amineIC5053.0 [1]
5-[[(2R,3R,4S,5R,6R)-5-(1H-Imidazol-5-ylmethoxy)-6-[2-(1H-indol-3-yl)ethoxy]-4-phenylmethoxy-3-(pyridin-3-ylmethoxy)oxan-2-yl]methoxy]pentan-1-amineKi53.0 [1]
Cyclo(Pro-Phe-D-Trp-Lys-Thr-Phe)Ki100.0 [1], 1000.0 [2]
8-D-Tryptophan-somatostatinIC502.3 [1]
8-D-Tryptophan-somatostatinKi5.83 [1]
2-(1-(4-Amino-3,5-diethoxybenzyl)piperidin-4-ylamino)benzo[d]oxazole-5-sulfonamideKi10000.0 [1]
(4R,7S,10S,13R,16S,19S)-10-(4-Aminobutyl)-19-[[(2S)-2-amino-3-(4-chlorophenyl)propanoyl]amino]-N-[(2S)-1-amino-3-naphthalen-2-yl-1-oxopropan-2-yl]-7-[(1R)-1-hydroxyethyl]-16-[(4-hydroxyphenyl)methyl]-13-(1H-indol-3-ylmethyl)-6,9,12,15,18-pentaoxo-1,2-dithia-5,8,11,14,17-pentazacycloicosane-4-carboxamideKi1000.0 [1]
(4R,7S,10S,13S,16S,19S,22S,25R)-25-Amino-13-(4-aminobutyl)-7,22-dibenzyl-10-[(1R)-1-hydroxyethyl]-19-[(4-hydroxyphenyl)methyl]-16-[(1S)-1-naphthalen-2-ylethyl]-6,9,12,15,18,21,24-heptaoxo-1,2-dithia-5,8,11,14,17,20,23-heptazacyclohexacosane-4-carboxylic acidIC502.1 [1], 2.8 [2]
(4R,7S,10S,13S,16R,19S,22S,25R)-25-Amino-13-(4-aminobutyl)-7,22-dibenzyl-10-[(1R)-1-hydroxyethyl]-16-(1H-indol-3-ylmethyl)-19-methyl-6,9,12,15,18,21,24-heptaoxo-1,2-dithia-5,8,11,14,17,20,23-heptazacyclohexacosane-4-carboxylic acidIC500.98 [1]
(4R,7S,10S,13S,16R,19S,22S,25R)-25-Amino-13-(4-aminobutyl)-7,22-dibenzyl-10-[(1R)-1-hydroxyethyl]-19-[(4-hydroxyphenyl)methyl]-16-[(1S)-1-naphthalen-2-ylethyl]-6,9,12,15,18,21,24-heptaoxo-1,2-dithia-5,8,11,14,17,20,23-heptazacyclohexacosane-4-carboxylic acidIC502.3 [1], 3.5 [2]
Des-AA1,2,5-[IAmp9,Tyr11]-SRIFIC50384.0 [1], 10000.0 [2]
(4R,7S,10R,13S,16R,19S,22S,25S,28R,31R,34S)-31-(4-Aminobutyl)-34-[[(2S)-2-amino-3-(4-hydroxyphenyl)propanoyl]amino]-13,25,28-tribenzyl-10,16-bis[(1R)-1-hydroxyethyl]-7-(hydroxymethyl)-22-(1H-indol-3-ylmethyl)-6,9,12,15,18,21,24,27,30,33-decaoxo-19-[[4-[(propan-2-ylamino)methyl]phenyl]methyl]-1,2-dithia-5,8,11,14,17,20,23,26,29,32-decazacyclopentatriacontane-4-carboxylic acidIC501000.0 [1]
(4R,7S,10S,13S,16S,19S,22S,25R)-25-Amino-13-(4-aminobutyl)-7,22-dibenzyl-10-[(1R)-1-hydroxyethyl]-16-(1H-indol-3-ylmethyl)-19-methyl-6,9,12,15,18,21,24-heptaoxo-1,2-dithia-5,8,11,14,17,20,23-heptazacyclohexacosane-4-carboxylic acidIC500.84 [1]
5-[[(2S,3S,5R,6S)-5-(1H-Imidazol-5-ylmethoxy)-6-[2-(1H-indol-3-yl)ethoxy]-3,4-bis(phenylmethoxy)oxan-2-yl]methoxy]pentan-1-amineIC50100.0 [1]
5-[[(2S,3S,5R,6S)-5-(1H-Imidazol-5-ylmethoxy)-6-[2-(1H-indol-3-yl)ethoxy]-3,4-bis(phenylmethoxy)oxan-2-yl]methoxy]pentan-1-amineKi100.0 [1]
5-[[(2R,3R,4R,5S)-1-[2-(1H-Indol-3-yl)ethyl]-3,4,5-tris(phenylmethoxy)piperidin-2-yl]methoxy]pentan-1-amineKi4400.0 [1]
(4R,7S,10R,13S,16R,19R,22S,25R,28S,31R,34S,37R)-19,34-Bis(4-aminobutyl)-31-(2-amino-2-oxoethyl)-37-[[2-[[(2S)-2-aminopropanoyl]amino]acetyl]amino]-13,25-dibenzyl-10,16-bis[(1S)-1-hydroxyethyl]-7-(hydroxymethyl)-22-(1H-indol-3-ylmethyl)-6,9,12,15,18,21,24,27,30,33,36-undecaoxo-28-(pyrazin-2-ylmethyl)-1,2-dithia-5,8,11,14,17,20,23,26,29,32,35-undecazacyclooctatriacontane-4-carboxylic acidKi60.0 [1], 77.0 [2]
4-Fluoro-N-[(1R,2S)-2-(1H-indol-3-ylmethylamino)cyclohexyl]benzamideKi1089.0 [1], 5930.0 [2]
AstemizoleKi10000.0 [1]
LanreotideKi1000.0 [1]
PasireotideKi100.0 [1]
EdotreotideIC501000.0 [1]
VapreotideKi158.49 [1]
(4R,7S,10S,13S,16S,19S,22R,25S,28S,31S,34R)-34-Amino-31-(4-aminobutyl)-13,25,28-tribenzyl-10,16-bis[(1R)-1-hydroxyethyl]-7-(hydroxymethyl)-22-(1H-indol-3-ylmethyl)-6,9,12,15,18,21,24,27,30,33-decaoxo-19-[[4-[(propan-2-ylamino)methyl]phenyl]methyl]-1,2-dithia-5,8,11,14,17,20,23,26,29,32-decazacyclopentatriacontane-4-carboxylic acidIC501000.0 [1]
CID 15965425Ki81.0 [1]
CID 56927659IC50384.0 [1]
(1R,3R)-1-(Oxan-4-yl)-3-(5-phenyl-1H-imidazol-2-yl)-2,3,4,9-tetrahydro-1H-pyrido[3,4-b]indoleIC501000.0 [1]
(3R)-1,1-Dibutyl-3-(5-phenyl-1H-imidazol-2-yl)-2,3,4,9-tetrahydropyrido[3,4-b]indoleKi7100.0 [1]
3-[3-(1H-Imidazole-4-yl)propyl]-1-[2-[(5-bromo-2-pyridinyl)(3,4-dichlorobenzyl)amino]ethyl]thioureaKi70.0 [1]
(2R,5R)-5-(4-Aminobutyl)-2-(1H-indol-3-ylmethyl)-7-(naphthalen-1-ylmethyl)-1,4,7-thiadiazonane-3,6-dioneIC501047.0 [1]
H-c[Cys-Phe-DTrp-Lys-Thr-Cys]-OHIC501000.0 [1]
(3S)-1,1-Dibutyl-3-(5-phenyl-1H-imidazol-2-yl)-2,3,4,9-tetrahydropyrido[3,4-b]indoleKi9800.0 [1]
N-(1-(3-Ethoxy-4-methoxybenzyl)piperidin-4-yl)benzo[d]oxazol-2-amineKi10000.0 [1]
2-(1-(3-Ethoxy-4-methoxybenzyl)piperidin-4-ylamino)benzo[d]oxazole-5-sulfonamideKi10000.0 [1]
3-[(1R,3R)-3-[5-(5-Fluoropyridin-2-yl)-1H-imidazol-2-yl]-1-(1-methylpyrazol-4-yl)-2,3,4,9-tetrahydropyrido[3,4-b]indol-1-yl]-5-methyl-1,2,4-oxadiazoleIC503200.0 [1]
4-((4-(Benzo[d]oxazol-2-ylamino)piperidin-1-yl)methyl)-2-ethoxyphenolKi10000.0 [1]
N-(1-(3-(Cyclopentyloxy)-4-methoxybenzyl)piperidin-4-yl)benzo[d]oxazol-2-amineKi10000.0 [1]
Benzooxazol-2-yl-[1-(3-isobutoxy-4-methoxy-benzyl)-piperidin-4-yl]-amineKi10000.0 [1]
N-(1-(4-Methoxy-3-propoxybenzyl)piperidin-4-yl)benzo[d]oxazol-2-amineKi10000.0 [1]
N-(1-(3-Ethoxy-4-fluorobenzyl)piperidin-4-yl)benzo[d]oxazol-2-amineKi10000.0 [1]
N-(1-(4-Chloro-3-ethoxybenzyl)piperidin-4-yl)benzo[d]oxazol-2-amineKi10000.0 [1]
N-(1-(3-Ethoxy-4-methylbenzyl)piperidin-4-yl)benzo[d]oxazol-2-amineKi10000.0 [1]
(3R,6S,9R,12S,15R,18S)-9-(4-Aminobutyl)-N-[(2S,3R)-1-amino-3-hydroxy-1-oxobutan-2-yl]-18-[[(2R)-2-amino-3-phenylpropanoyl]amino]-15-benzyl-6-[(1R)-1-hydroxyethyl]-12-(1H-indol-3-ylmethyl)-5,8,11,14,17-pentaoxo-1-thia-4,7,10,13,16-pentazacyclononadecane-3-carboxamideIC501000.0 [1]
(2S,3R)-2-[[(3R,6S,9R,12S,15R,18S)-9-(4-Aminobutyl)-18-[[(2R)-2-amino-3-phenylpropanoyl]amino]-15-benzyl-6-[(1R)-1-hydroxyethyl]-12-(1H-indol-3-ylmethyl)-5,8,11,14,17-pentaoxo-1-thia-4,7,10,13,16-pentazacyclononadecane-3-carbonyl]amino]-3-hydroxybutanoic acidIC501000.0 [1]
(3R,6S,9R,12S,15R,18S)-9-(4-Aminobutyl)-18-[[(2R)-2-amino-3-phenylpropanoyl]amino]-15-benzyl-6-[(1R)-1-hydroxyethyl]-12-(1H-indol-3-ylmethyl)-5,8,11,14,17-pentaoxo-1-thia-4,7,10,13,16-pentazacyclononadecane-3-carboxylic acidIC501000.0 [1]
(4S,7R,10S,13R,16S,19R)-10-(4-Aminobutyl)-19-[[(2S)-2-amino-3-phenylpropanoyl]amino]-16-benzyl-7-[(1R)-1-hydroxyethyl]-13-(1H-indol-3-ylmethyl)-6,9,12,15,18-pentaoxo-1,2-dithia-5,8,11,14,17-pentazacycloicosane-4-carboxylic acidIC501000.0 [1]
(4R,7S,10S,13S,16S,19S,22R,25S,28S,31S,34S,37R)-19,34-Bis(4-aminobutyl)-31-(2-amino-2-oxoethyl)-37-[[2-[[(2S)-2-aminopropanoyl]amino]acetyl]amino]-13,25,28-tribenzyl-10,16-bis[(1R)-1-hydroxyethyl]-7-(hydroxymethyl)-22-[(4-hydroxyphenyl)methyl]-6,9,12,15,18,21,24,27,30,33,36-undecaoxo-1,2-dithia-5,8,11,14,17,20,23,26,29,32,35-undecazacyclooctatriacontane-4-carboxylic acidIC5016.0 [1]
5-Methyl-1,5-diazapentacyclo[10.8.1.02,7.08,21.013,18]henicosa-2(7),8(21),9,11,13,15,17-heptaeneKi10000.0 [1]
5-[[(2R,3S,5R,6R)-6-[2-(1H-Indol-3-yl)ethoxy]-3,5-bis(phenylmethoxy)oxan-2-yl]methoxy]pentan-1-amineKi1700.0 [1]
5-[[(2S,3S,4R,5R,6S)-5-(1H-Imidazol-5-ylmethoxy)-6-[2-(1H-indol-3-yl)ethoxy]-3,4-bis(phenylmethoxy)oxan-2-yl]methoxy]pentan-1-amineKi100.0 [1]
(2R,3S)-N-[(5-Amino-1,3-dioxan-2-yl)methyl]-3-(1H-indol-3-yl)-N-methyl-2-[2-oxo-3-(1-phenylpiperidin-3-yl)imidazolidin-1-yl]butanamideKi1400.0 [1]
N-[(R)-2-(1H-Indol-3-yl)-1-(4-phenyl-1H-imidazol-2-yl)-ethyl]-4-methoxy-benzamidineKi5010.0 [1]
2-[8-(3-Aminopropyl)-6-(1-benzothiophen-3-yl)imidazo[1,2-a]pyrazin-2-yl]-N-cyclohexyl-2-methylpropanamideKi10000.0 [1]
4-Chloro-N'-[(1R)-2-(1H-indol-3-yl)-1-(5-phenyl-1H-imidazol-2-yl)ethyl]benzenecarboximidamideKi3840.0 [1]
[(R)-1-(4-Phenyl-1H-imidazole-2-yl)-2-(1H-indole-3-yl)ethyl]carbamic acid tert-butyl esterKi10000.0 [1]
(3S,6S,9S,12R,15S,18R)-9-(4-Aminobutyl)-3-benzyl-15-[(4-hydroxyphenyl)methyl]-12-(1H-indol-3-ylmethyl)-1,18-dimethyl-6-propan-2-yl-1,4,7,10,13,16-hexazacyclooctadecane-2,5,8,11,14,17-hexoneIC501000.0 [1]
2,4-Difluoro-N'-[(1R)-2-(1H-indol-3-yl)-1-(5-phenyl-1H-imidazol-2-yl)ethyl]benzenecarboximidamideKi10000.0 [1]
3-[6-(3-Nitrophenyl)-2-phenylimidazo[1,2-a]pyrazin-8-yl]propan-1-amineKi10000.0 [1]
5-((2R,3R,4S,5R,6R)-3,4,5-Tris-benzyloxy-6-methoxy-tetrahydro-pyran-2-ylmethoxy)-pentylamineKi2000.0 [1]
3-[3-(1H-Imidazole-4-yl)propyl]-1-[3-[(5-bromo-2-pyridinyl)(1-naphthylmethyl)amino]propyl]thioureaKi16.0 [1]
1-[(R)-1-(4-Phenyl-1H-imidazole-2-yl)-2-(1H-indole-3-yl)ethyl]-3-(2,4-difluorophenyl)ureaKi10000.0 [1]
3-[3-(1H-Imidazole-4-yl)propyl]-1-[2-[(5-bromo-2-pyridinyl)(3,4-dichlorobenzyl)amino]ethyl]ureaKi14.0 [1]
3-(3-Aminopropyl)-1-[2-[(5-bromo-2-pyridinyl)(3,4-dichlorobenzyl)amino]ethyl]thioureaKi4200.0 [1]
3-[3-(1H-Imidazole-1-yl)propyl]-1-[3-[(2-pyridinyl)(4-bromobenzyl)amino]propyl]thioureaKi7000.0 [1]
3-[3-(1H-Imidazole-4-yl)propyl]-1-[4-[(5-bromo-2-pyridinyl)(3,4-dichlorobenzyl)amino]butyl]thioureaKi53.0 [1]
(4R,7S,10S,13R,16S,19S)-10-(4-Aminobutyl)-N-[(2S,3R)-1-amino-3-hydroxy-1-oxobutan-2-yl]-19-[[(2R)-2-amino-3-phenylpropanoyl]amino]-7-ethyl-16-[(4-hydroxyphenyl)methyl]-13-(1H-indol-3-ylmethyl)-6,9,12,15,18-pentaoxo-1,2-dithia-5,8,11,14,17-pentazacycloicosane-4-carboxamideIC501000.0 [1]
3-[3-(1H-Imidazole-1-yl)propyl]-1-[4-[(2-pyridinyl)(3,4-dichlorobenzyl)amino]butyl]thioureaKi4000.0 [1]
3-(1H-Benzotriazole-5-yl)-1-[2-[(5-bromo-2-pyridinyl)(3,4-dichlorobenzyl)amino]ethyl]thioureaKi1000.0 [1]
5-[[(2R,3S,5R,6R)-5-(1H-Imidazol-5-ylmethoxy)-6-[2-(1H-indol-3-yl)ethoxy]-3-phenylmethoxyoxan-2-yl]methoxy]pentan-1-amineKi3000.0 [1]
1-[2-[(5-Bromopyridin-2-yl)-[(3,4-dichlorophenyl)methyl]amino]ethyl]-3-(3-pyrrolidin-1-ylpropyl)thioureaKi477.0 [1]
N'-[[(2R,3R,4S,5R,6R)-6-[2-(1H-Indol-3-yl)ethoxy]-3,4,5-tris(phenylmethoxy)oxan-2-yl]methyl]pentane-1,5-diamineKi500.0 [1]
3-(4-Aminobutyl)-1-[3-[(5-bromo-2-pyridinyl)(1-naphthylmethyl)amino]propyl]thioureaKi2000.0 [1]
3-[2-(1H-Imidazole-4-yl)ethyl]-1-[2-[(5-bromo-2-pyridinyl)(3,4-dichlorobenzyl)amino]ethyl]thioureaKi476.0 [1]
3-(1H-Benzimidazole-2-ylmethyl)-1-[2-[(5-bromo-2-pyridinyl)(3,4-dichlorobenzyl)amino]ethyl]thioureaKi1200.0 [1]
3-[3-(1H-Imidazole-4-yl)propyl]-1-[2-[(5-nitro-2-pyridinyl)(3,4-dichlorobenzyl)amino]ethyl]thioureaKi176.0 [1]
3-(4-Aminobutyl)-1-[3-[(5-bromo-2-pyridinyl)(3,4-dichlorobenzyl)amino]propyl]thioureaKi1000.0 [1]
3-[3-(1H-Imidazole-1-yl)propyl]-1-[3-[(5-bromo-2-pyridinyl)(3,4-dichlorobenzyl)amino]propyl]thioureaKi1700.0 [1]
3-[3-(1H-Imidazole-4-yl)propyl]-1-[5-[(5-bromo-2-pyridinyl)(3,4-dichlorobenzyl)amino]pentyl]thioureaKi132.0 [1]
3-[3-(2-Pyridinylamino)propyl]-1-[3-[(5-bromo-2-pyridinyl)(3,4-dichlorobenzyl)amino]propyl]thioureaKi185.0 [1]
3-(4-Piperidinophenyl)-1-[2-[(5-bromo-2-pyridinyl)(3,4-dichlorobenzyl)amino]ethyl]thioureaKi15000.0 [1]
5-[[(2S,3S,4R,5S,6S)-6-[2-(1H-Indol-3-yl)ethoxy]-3,4,5-tris(phenylmethoxy)oxan-2-yl]methoxy]pentan-1-amineKi2000.0 [1]
(4R,7S,10S,13R,16S,19S)-10-(4-Aminobutyl)-N-[(2S,3R)-1-amino-3-hydroxy-1-oxobutan-2-yl]-19-[[(2S)-2-amino-3-phenylpropanoyl]amino]-7-[(1R)-1-hydroxyethyl]-13-(1H-indol-3-ylmethyl)-6,9,12,15,18-pentaoxo-16-(pyridin-3-ylmethyl)-1,2-dithia-5,8,11,14,17-pentazacycloicosane-4-carboxamideIC501000.0 [1]
3-[3-(1H-Imidazole-1-yl)propyl]-1-[4-[(2-pyridinyl)(4-bromobenzyl)amino]butyl]thioureaKi7000.0 [1]
(4R,7S,10S,13R,16S,19S)-10-(4-Aminobutyl)-N-[(2S,3R)-1-amino-3-hydroxy-1-oxobutan-2-yl]-19-[[(2S)-2-amino-3-(4-hydroxyphenyl)propanoyl]amino]-7-[(1R)-1-hydroxyethyl]-13-(1H-indol-3-ylmethyl)-6,9,12,15,18-pentaoxo-16-(pyridin-3-ylmethyl)-1,2-dithia-5,8,11,14,17-pentazacycloicosane-4-carboxamideIC501000.0 [1]
(4R,7S,10S,13R,16S,19S)-10-(4-Aminobutyl)-N-[(2S,3R)-1-amino-3-hydroxy-1-oxobutan-2-yl]-19-[[(2R)-2-amino-3-naphthalen-2-ylpropanoyl]amino]-16-[(4-hydroxyphenyl)methyl]-13-(1H-indol-3-ylmethyl)-6,9,12,15,18-pentaoxo-7-propan-2-yl-1,2-dithia-5,8,11,14,17-pentazacycloicosane-4-carboxamideIC501000.0 [1]
Items per page: 1 - 10 of 100
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References

This online tool may be cited as follows

MLA

"Quest Database™ Somatostatin receptor 4 Inhibitors (IC50, Ki)." AAT Bioquest, Inc., 9 May. 2024, https://www.aatbio.com/data-sets/somatostatin-receptor-4-inhibitors-ic50-ki.

APA

AAT Bioquest, Inc. (2024, May 9). Quest Database™ Somatostatin receptor 4 Inhibitors (IC50, Ki). AAT Bioquest. https://www.aatbio.com/data-sets/somatostatin-receptor-4-inhibitors-ic50-ki.
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