 | Finasteride | IC50 | 150.0 [1] |
| Finasteride | Ki | 100.0 [1], 150.0 [2], 366.0 [3] |
 | Epristeride | IC50 | 1000.0 [1], 1100.0 [2], 1600.0 [3], 7500.0 [4] |
| Epristeride | Ki | 410.0 [1], 1600.0 [2], 5000.0 [3] |
 | Bexlosteride | IC50 | 2.3 [1], 8.0 [2], 8.6 [3] |
| Bexlosteride | Ki | 4.0 [1] |
 | 1,2,5,6-Tetrahydro pyrido[1,2-a]quinolin-3-one | IC50 | 295.12 [1], 298.0 [2] |
 | 4-Methyl-8-chloro-1,2,5,6-tetrahydrobenzo[f]quinolin-3(4H)-one | IC50 | 30.0 [1], 173.78 [2] |
| 4-Methyl-8-chloro-1,2,5,6-tetrahydrobenzo[f]quinolin-3(4H)-one | Ki | 17.0 [1] |
 | 3H-Benzo(C)quinolizin-3-one, 1,2,5,6-tetrahydro-4,8-dimethyl- | IC50 | 19.95 [1], 20.0 [2], 41.0 [3] |
| 3H-Benzo(C)quinolizin-3-one, 1,2,5,6-tetrahydro-4,8-dimethyl- | Ki | 5.8 [1] |
 | 4-Methyl-8-chloro-1,2,5,6-tetrahydro pyrido[1,2-a]quinolin-3-one | IC50 | 5.62 [1], 5.8 [2], 7.6 [3], 41.0 [4] |
| 4-Methyl-8-chloro-1,2,5,6-tetrahydro pyrido[1,2-a]quinolin-3-one | Ki | 2.7 [1] |
 | 17-N,N-Diethylcarbamoyl-4-methyl-4-azaandrostane-3-one | IC50 | 1.7 [1], 4.14 [2] |
| 17-N,N-Diethylcarbamoyl-4-methyl-4-azaandrostane-3-one | Ki | 3.0 [1], 5.0 [2] |
 | (1R,4S,9Ar,11aR)-4,6,9a,11a-tetramethyl-1-(6-methylheptan-2-yl)-2,3,3a,3b,4,5,5a,8,9,9b,10,11-dodecahydro-1H-indeno[5,4-f]quinolin-7-one | IC50 | 0.5 [1], 0.9 [2] |
 | 8-Chloro-1,2,5,6-tetrahydro-3H-benzo[c]quinolizine-3-one | IC50 | 48.98 [1], 49.0 [2] |
 | (4Ar,10bR)-8-chloro-4,10b-dimethyl-2,4a,5,6-tetrahydro-1H-benzo[f]quinolin-3-one | IC50 | 17.0 [1] |
| (4Ar,10bR)-8-chloro-4,10b-dimethyl-2,4a,5,6-tetrahydro-1H-benzo[f]quinolin-3-one | Ki | 9.0 [1] |
 | Methyl (1S,9aR,11aS)-9a,11a-dimethyl-7-oxo-1,2,3,3a,3b,4,5,8,9,9b,10,11-dodecahydrocyclopenta[i]phenanthridine-1-carboxylate | Ki | 150.0 [1] |
 | 3,4,5,6-Tetrahydrobenzo[c]quinolizin-3-(4aH)-one | IC50 | 5130.0 [1] |
 | (1S,9Ar,11aS)-N-benzhydryl-9a,11a-dimethyl-7-oxo-1,2,3,3a,3b,4,5,8,9,9b,10,11-dodecahydrocyclopenta[i]phenanthridine-1-carboxamide | Ki | 30.0 [1] |
 | (1S,9Ar,11aS)-N-[bis(4-chlorophenyl)methyl]-9a,11a-dimethyl-7-oxo-1,2,3,3a,3b,4,5,8,9,9b,10,11-dodecahydrocyclopenta[i]phenanthridine-1-carboxamide | Ki | 20.0 [1] |
 | (1S,9Ar,11aS)-9a,11a-dimethyl-1-(morpholine-4-carbonyl)-1,2,3,3a,3b,4,5,8,9,9b,10,11-dodecahydrocyclopenta[i]phenanthridin-7-one | Ki | 2200.0 [1] |
 | 7-Bromo-9,10-dihydrophenanthrene-2-carboxylic Acid | IC50 | 26.0 [1] |
| 7-Bromo-9,10-dihydrophenanthrene-2-carboxylic Acid | Ki | 26.0 [1] |
 | 8-Methyl-1,2,5,6-tetrahydro-3H-benzo[c]quinolizine-3-one | IC50 | 376.0 [1], 380.19 [2] |
 | 4-Methyl-1,2,5,6-tetrahydro pyrido[1,2-a]quinolin-3-one | IC50 | 185.0 [1], 186.21 [2] |
 | Ethyl 4-methyl-3-oxo-1,2,5,6-tetrahydrobenzo[c]quinolizine-8-carboxylate | IC50 | 218.78 [1], 221.0 [2] |
 | Phenyl 4-methyl-3-oxo-1,2,5,6-tetrahydrobenzo[c]quinolizine-8-carboxylate | IC50 | 933.25 [1], 942.0 [2] |
 | Methyl 4-methyl-3-oxo-1,2,5,6-tetrahydrobenzo[c]quinolizine-8-carboxylate | IC50 | 117.0 [1], 117.49 [2] |
 | Tert-butyl 4-methyl-3-oxo-1,2,5,6-tetrahydrobenzo[c]quinolizine-8-carboxylate | IC50 | 1000.0 [1] |
 | (4-Methylphenyl) 4-methyl-3-oxo-1,2,5,6-tetrahydrobenzo[c]quinolizine-8-carboxylate | IC50 | 102.0 [1], 1047.13 [2], 1050.0 [3] |
 | (3-Methoxycarbonylphenyl) 4-methyl-3-oxo-1,2,5,6-tetrahydrobenzo[c]quinolizine-8-carboxylate | IC50 | 954.99 [1], 965.0 [2] |
 | (4-Tert-butylphenyl) 4-methyl-3-oxo-1,2,5,6-tetrahydrobenzo[c]quinolizine-8-carboxylate | IC50 | 560.0 [1], 562.34 [2] |
 | Propan-2-yl 4-methyl-3-oxo-1,2,5,6-tetrahydrobenzo[c]quinolizine-8-carboxylate | IC50 | 724.44 [1], 731.0 [2] |
 | (4-Methoxycarbonylphenyl) 4-methyl-3-oxo-1,2,5,6-tetrahydrobenzo[c]quinolizine-8-carboxylate | IC50 | 120.23 [1], 121.0 [2], 129.0 [3] |
 | Benzyl 4-methyl-3-oxo-1,2,5,6-tetrahydrobenzo[c]quinolizine-8-carboxylate | IC50 | 96.8 [1], 97.0 [2], 97.72 [3] |
 | (1S,9Ar,11aS)-9a,11a-dimethyl-1-(3-methylbutanoyl)-1,2,3,3a,3b,4,5,8,9,9b,10,11-dodecahydrocyclopenta[i]phenanthridin-7-one | Ki | 9.0 [1] |
 | (1S,9Ar,11aS)-N-tert-butyl-9a,11a-dimethyl-7-oxo-1,2,3,3a,3b,4,5,8,9,9b,10,11-dodecahydrocyclopenta[i]phenanthridine-1-carboxamide | Ki | 820.0 [1] |
 | 4-[3-[3-[Bis[4-(2-methylpropyl)phenyl]methylamino]benzoyl]indol-1-yl]butanoic acid | IC50 | 3.0 [1], 38.0 [2] |
 | 5-(Benzyloxy)-1H-indole-2-carboxylic acid | Ki | 2500.0 [1] |
 | 4-Methyl-1,4,4a,5,6,10b-hexahydro-2H-benzo[f]quinolin-3-one | IC50 | 560.0 [1] |
 | 2-Adamantyl (1S,3aS,3bS,9aR,9bS,11aS)-9a,11a-dimethyl-7-oxo-1,2,3,3a,3b,4,5,8,9,9b,10,11-dodecahydrocyclopenta[i]phenanthridine-1-carboxylate | Ki | 6.9 [1] |
 | (10R,13S,17S)-N-Tert-butyl-4-chloro-10,13-dimethyl-3-oxo-1,2,6,7,8,9,11,12,14,15,16,17-dodecahydrocyclopenta[a]phenanthrene-17-carboxamide | IC50 | 1000.0 [1] |
 | 8-Chloro-1,2,5,6-tetrahydrobenzo[f]quinolin-3(4H)-one | IC50 | 460.0 [1] |
 | 1,4,5,6-Tetrahydro-2H-benzo[f]quinolin-3-one | IC50 | 6500.0 [1] |
 | (1S,9Ar,11aS)-6-chloro-N-(4-chlorophenyl)-N-cyclopentyl-9a,11a-dimethyl-7-oxo-1,2,3,3a,3b,4,5,8,9,9b,10,11-dodecahydrocyclopenta[i]phenanthridine-1-carboxamide | Ki | 0.6 [1] |
 | (1S,9Ar,11aS)-N-(4-chlorophenyl)-N-cyclopentyl-6,9a,11a-trimethyl-7-oxo-1,2,3,3a,3b,4,5,8,9,9b,10,11-dodecahydrocyclopenta[i]phenanthridine-1-carboxamide | Ki | 0.3 [1] |
 | (10Br)-8-chloro-4,10b-dimethyl-2,4a,5,6-tetrahydro-1H-benzo[f]quinolin-3-one | IC50 | 17.0 [1] |
| (10Br)-8-chloro-4,10b-dimethyl-2,4a,5,6-tetrahydro-1H-benzo[f]quinolin-3-one | Ki | 9.0 [1] |
 | (10R,13S,17S)-4-Bromo-N-tert-butyl-10,13-dimethyl-3-oxo-1,2,6,7,8,9,11,12,14,15,16,17-dodecahydrocyclopenta[a]phenanthrene-17-carboxamide | IC50 | 981.0 [1] |
 | (10R,13S,17S)-N-Tert-butyl-10,13-dimethyl-3-oxo-4-sulfanyl-1,2,6,7,8,9,11,12,14,15,16,17-dodecahydrocyclopenta[a]phenanthrene-17-carboxamide | IC50 | 709.0 [1] |
 | (1S,9Ar,11aS)-9a,11a-dimethyl-7-oxo-N-phenyl-1,2,3,3a,3b,4,5,8,9,9b,10,11-dodecahydrocyclopenta[i]phenanthridine-1-carboxamide | Ki | 240.0 [1] |
 | (1S,9Ar,11aS)-N-(3,5-ditert-butylphenyl)-9a,11a-dimethyl-7-oxo-1,2,3,3a,3b,4,5,8,9,9b,10,11-dodecahydrocyclopenta[i]phenanthridine-1-carboxamide | Ki | 8.0 [1] |
 | CID 44275674 | Ki | 8.8 [1] |
 | (4Ar,10bR)-4,10b-dimethyl-8-[(E)-2-phenylethenyl]-2,4a,5,6-tetrahydro-1H-benzo[f]quinolin-3-one | IC50 | 23.0 [1] |
 | (1S,9Ar,11aS)-9a,11a-dimethyl-7-oxo-N',N'-diphenyl-1,2,3,3a,3b,4,5,8,9,9b,10,11-dodecahydrocyclopenta[i]phenanthridine-1-carbohydrazide | Ki | 14.0 [1] |
 | (1S,9Ar,11aS)-9a,11a-dimethyl-7-oxo-N-trityl-1,2,3,3a,3b,4,5,8,9,9b,10,11-dodecahydrocyclopenta[i]phenanthridine-1-carboxamide | Ki | 8.2 [1] |
 | (1S,9Ar,11aS)-N,N-diethyl-9a,11a-dimethyl-7-oxo-1,2,3,3a,3b,4,5,8,9,9b,10,11-dodecahydrocyclopenta[i]phenanthridine-1-carboxamide | Ki | 750.0 [1] |
 | (1S,9Ar,11aS)-N-(dicyclohexylmethyl)-9a,11a-dimethyl-7-oxo-1,2,3,3a,3b,4,5,8,9,9b,10,11-dodecahydrocyclopenta[i]phenanthridine-1-carboxamide | Ki | 20.0 [1] |
 | (1S,9Ar,11aS)-9a,11a-dimethyl-1-(piperazine-1-carbonyl)-1,2,3,3a,3b,4,5,8,9,9b,10,11-dodecahydrocyclopenta[i]phenanthridin-7-one | Ki | 8600.0 [1] |
 | (1S,9Ar,11aS)-9a,11a-dimethyl-1-(thiomorpholine-4-carbonyl)-1,2,3,3a,3b,4,5,8,9,9b,10,11-dodecahydrocyclopenta[i]phenanthridin-7-one | Ki | 570.0 [1] |
 | (1S,9Ar,11aS)-N-methoxy-N,9a,11a-trimethyl-7-oxo-1,2,3,3a,3b,4,5,8,9,9b,10,11-dodecahydrocyclopenta[i]phenanthridine-1-carboxamide | Ki | 2300.0 [1] |
 | (1S,9Ar,11aS)-N-[bis(4-fluorophenyl)methyl]-9a,11a-dimethyl-7-oxo-1,2,3,3a,3b,4,5,8,9,9b,10,11-dodecahydrocyclopenta[i]phenanthridine-1-carboxamide | Ki | 20.0 [1] |
 | (1S,9Ar,11aS)-N-(1-adamantyl)-9a,11a-dimethyl-7-oxo-1,2,3,3a,3b,4,5,8,9,9b,10,11-dodecahydrocyclopenta[i]phenanthridine-1-carboxamide | Ki | 11.0 [1] |
 | (9Ar,11aS)-N-benzhydryl-9a,11a-dimethyl-7-oxo-1,2,3,3a,3b,4,5,8,9,9b,10,11-dodecahydrocyclopenta[i]phenanthridine-1-carboxamide | IC50 | 186.0 [1] |
 | (4As)-7-chloro-4a-methyl-4,9-dihydro-3H-phenanthrene-2-carboxylic acid | Ki | 1200.0 [1] |
 | (10Br)-8-chloro-4,10b-dimethyl-1,2,5,6-tetrahydrophenanthridin-3-one | Ki | 920.0 [1] |
 | 8-Chloro-4-methyl-1,4,4a,5,6,10b-hexahydro-2H-benzo[f]quinolin-3-one | IC50 | 41.0 [1] |
| 8-Chloro-4-methyl-1,4,4a,5,6,10b-hexahydro-2H-benzo[f]quinolin-3-one | Ki | 15.0 [1] |
 | 8-Bromo-4-methyl-1,2,5,6-tetrahydrobenzo[f]quinolizin-3-one | IC50 | 8.1 [1], 8.13 [2] |
 | 8-Methoxy-4-methyl-1,2,5,6-tetrahydro-pyrido[1,2-a]quinolin-3-one | IC50 | 178.0 [1], 181.97 [2] |
 | 4-Methyl-8-vinyl-1,2,5,6-tetrahydro-pyrido[1,2-a]quinolin-3-one | IC50 | 21.38 [1], 21.6 [2] |
 | 4-Methyl-8-thiophen-2-yl-1,2,5,6-tetrahydrobenzo[f]quinolizin-3-one | IC50 | 79.0 [1], 79.43 [2] |
 | 4-Methyl-8-[(Z)-2-phenylethenyl]-1,2,5,6-tetrahydrobenzo[f]quinolizin-3-one | IC50 | 14.13 [1], 14.2 [2] |
 | 4-Methyl-8-phenyl-1,2,5,6-tetrahydrobenzo[f]quinolizin-3-one | IC50 | 128.0 [1], 128.82 [2] |
 | 4-Methyl-8-(2-phenylethynyl)-1,2,5,6-tetrahydrobenzo[f]quinolizin-3-one | IC50 | 8.71 [1], 8.75 [2] |
 | 8-[(2-Chlorophenyl)methoxy]-4-methyl-1,2,5,6-tetrahydrobenzo[f]quinolizin-3-one | IC50 | 194.0 [1], 194.98 [2] |
 | 4-Methyl-8-phenylmethoxy-1,2,5,6-tetrahydrobenzo[f]quinolizin-3-one | IC50 | 111.0 [1], 112.2 [2] |
 | 8-[[2,5-Bis(trifluoromethyl)phenyl]methoxy]-4-methyl-1,2,5,6-tetrahydrobenzo[f]quinolizin-3-one | IC50 | 389.05 [1], 393.0 [2] |
 | 8-[(4-Chlorophenyl)methoxy]-4-methyl-1,2,5,6-tetrahydrobenzo[f]quinolizin-3-one | IC50 | 92.9 [1], 93.33 [2] |
 | 8-[(3-Chlorophenyl)methoxy]-4-methyl-1,2,5,6-tetrahydrobenzo[f]quinolizin-3-one | IC50 | 93.0 [1], 93.33 [2] |
 | 4-Methyl-8-[[4-(trifluoromethyl)phenyl]methoxy]-1,2,5,6-tetrahydrobenzo[f]quinolizin-3-one | IC50 | 83.18 [1], 83.7 [2] |
 | 8-[[2,4-Bis(trifluoromethyl)phenyl]methoxy]-4-methyl-1,2,5,6-tetrahydrobenzo[f]quinolizin-3-one | IC50 | 147.91 [1], 149.0 [2] |
 | 4-Methyl-8-[(E)-2-phenylethenyl]-1,2,5,6-tetrahydrobenzo[f]quinolizin-3-one | IC50 | 380.0 [1], 380.19 [2] |
 | 8-(Furan-2-yl)-4-methyl-1,2,5,6-tetrahydrobenzo[f]quinolizin-3-one | IC50 | 131.83 [1], 133.0 [2] |
 | 4-Methyl-8-pyridin-3-yl-1,2,5,6-tetrahydrobenzo[f]quinolizin-3-one | IC50 | 169.82 [1], 170.0 [2] |
 | 8-Ethyl-4-methyl-1,2,5,6-tetrahydro-pyrido[1,2-a]quinolin-3-one | IC50 | 14.0 [1], 14.13 [2] |
 | (R)-8-Chloro-4,10b-dimethyl-1,4,6,10b-tetrahydro-2H-benzo[f]quinolin-3-one | IC50 | 120.0 [1] |
| (R)-8-Chloro-4,10b-dimethyl-1,4,6,10b-tetrahydro-2H-benzo[f]quinolin-3-one | Ki | 180.0 [1] |
 | 17-[(2E)-2-Hydroxyiminoethyl]-10,13-dimethyl-1,2,6,7,8,9,11,12,14,15,16,17-dodecahydrocyclopenta[a]phenanthren-3-one | IC50 | 1950.0 [1], 2440.0 [2] |
 | (17S)-17-[(Z)-N-Hydroxy-C-methylcarbonimidoyl]-10,13-dimethyl-1,2,6,7,8,9,11,12,14,15,16,17-dodecahydrocyclopenta[a]phenanthren-3-one | IC50 | 1630.0 [1], 1770.0 [2] |
 | 17-[(2E)-2-Hydroxyiminopropyl]-10,13-dimethyl-2,7,8,9,11,12,14,15,16,17-decahydro-1H-cyclopenta[a]phenanthrene-3,6-dione | IC50 | 900.0 [1], 2900.0 [2] |
 | 8-Chloro-4,10b-dimethyl-2,4a,5,6-tetrahydro-1H-benzo[f]quinolin-3-one | IC50 | 32.36 [1] |
| 8-Chloro-4,10b-dimethyl-2,4a,5,6-tetrahydro-1H-benzo[f]quinolin-3-one | Ki | 20.0 [1] |
 | (10R,13S)-17-(Benzimidazol-1-yl)-10,13-dimethyl-1,2,6,7,8,9,11,12,14,15-decahydrocyclopenta[a]phenanthren-3-one | IC50 | 770.0 [1] |
 | 17-(N-t-Butylcarboxamide)estra-1,3,5(10)-triene-3-carboxylic acid | Ki | 1600.0 [1] |
 | 6-(Benzyloxy)-5-methoxy-1H-indole-2-carboxylic acid | Ki | 460.0 [1] |
 | 4-(Benzyloxy)-1H-indole-2-carboxylic acid | Ki | 2500.0 [1] |
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