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Steryl-sulfatase Inhibitors (IC50, Ki)

Structure
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▼
Compound Name
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▼
Standard Type
▲
▼
Standard Values (in nM)
▲
▼
EmateIC5050.0 [1]
EmateKi470.0 [1], 670.0 [2]
IrosustatIC508.0 [1]
4-Methyl-2-oxo-2H-chromen-7-yl sulfamateIC501030.0 [1]
Sulfamic acid 2-adamantan-2-ylidenemethyl-benzooxazol-6-yl esterIC500.77 [1]
Sulfamic acid 2-adamantan-2-ylidenemethyl-benzooxazol-6-yl esterKi6000.0 [1]
(8R,9S,13S,14S,17R)-17-Benzyl-13-methyl-7,8,9,11,12,14,15,16-octahydro-6H-cyclopenta[a]phenanthrene-3,17-diolIC50230.0 [1], 310.0 [2], 325.0 [3]
(8R,9S,13S,14S,17R)-17-Benzyl-13-methyl-7,8,9,11,12,14,15,16-octahydro-6H-cyclopenta[a]phenanthrene-3,17-diolKi250.0 [1]
(8R,9S,13S,14S,17R)-17-[(4-Tert-butylphenyl)methyl]-13-methyl-7,8,9,11,12,14,15,16-octahydro-6H-cyclopenta[a]phenanthrene-3,17-diolIC508.3 [1], 12.0 [2], 14.0 [3], 28.0 [4]
[(1S,5R)-8-[[3,5-Bis(trifluoromethyl)phenyl]sulfonylcarbamoyl]-8-azabicyclo[3.2.1]octan-3-yl] 2-phenylacetateIC5084.0 [1], 1890.0 [2]
[(1S,5R)-8-[[3,5-Bis(trifluoromethyl)phenyl]sulfonylcarbamoyl]-8-azabicyclo[3.2.1]octan-3-yl] 2-phenylacetateKi76.0 [1]
Estrone-3-methylthiophosphonateIC5036000.0 [1], 43000.0 [2]
Estrone-3-methylthiophosphonateKi15000.0 [1], 33000.0 [2]
Sulfamic acid 2-adamantan-1-yl-4-oxo-4H-thiochromen-6-yl esterIC500.34 [1], 20.0 [2]
Sulfamic acid 2-adamantan-1-yl-4-oxo-4H-thiochromen-6-yl esterKi210.0 [1]
[(1S,5R)-8-[(4-Chlorophenyl)sulfonylcarbamoyl]-8-azabicyclo[3.2.1]octan-3-yl] 2-phenylacetateIC50910.0 [1], 6270.0 [2], 6720.0 [3]
[(1S,5R)-8-[(4-Chlorophenyl)sulfonylcarbamoyl]-8-azabicyclo[3.2.1]octan-3-yl] 2-phenylacetateKi2400.0 [1]
2-Adamantan-1-yl-4-oxo-4H-chromene-6-carboxylic acidIC50180.0 [1], 530.0 [2], 9400.0 [3]
2-Adamantan-1-yl-4-oxo-4H-chromene-6-carboxylic acidKi500.0 [1]
2-Adamantan-1-yl-4-oxo-4H-thiochromene-6-carboxylic acidIC50180.0 [1]
2-Adamantan-1-yl-4-oxo-4H-thiochromene-6-carboxylic acidKi500.0 [1], 530.0 [2]
[(8R,9S,13S,14S,17R)-17-[(4-Tert-butylphenyl)methyl]-17-hydroxy-13-methyl-7,8,9,11,12,14,15,16-octahydro-6H-cyclopenta[a]phenanthren-3-yl] sulfamateIC500.15 [1], 1.4 [2], 30.0 [3]
2-Adamantan-1-yl-4-oxo-4H-chromene-6-carbaldehydeIC50180.0 [1], 530.0 [2], 30000.0 [3]
2-Adamantan-1-yl-4-oxo-4H-chromene-6-carbaldehydeKi20000.0 [1]
(2-Adamantan-1-yl-4-oxo-4H-chromen-6-yl)-oxo-acetic acidIC50180.0 [1], 530.0 [2], 12300.0 [3]
(2-Adamantan-1-yl-4-oxo-4H-chromen-6-yl)-oxo-acetic acidKi2200.0 [1]
2-Adamantan-1-yl-4-oxo-4H-thiochromene-6-carbonitrileIC50180.0 [1], 530.0 [2], 30000.0 [3]
2-Adamantan-1-yl-4-oxo-4H-thiochromene-6-carbonitrileKi50000.0 [1]
2-Adamantan-1-yl-4-oxo-4H-chromene-6-carboxylic acid amideIC50180.0 [1], 530.0 [2], 30000.0 [3]
2-Adamantan-1-yl-4-oxo-4H-chromene-6-carboxylic acid amideKi50000.0 [1]
2-Adamantan-1-yl-6-hydroxymethyl-chromen-4-oneIC50180.0 [1], 530.0 [2], 30000.0 [3]
2-Adamantan-1-yl-6-hydroxymethyl-chromen-4-oneKi32000.0 [1]
(2-Adamantan-1-yl-4-oxo-4H-chromen-6-yl)-acetic acidIC50180.0 [1], 530.0 [2], 30000.0 [3]
(2-Adamantan-1-yl-4-oxo-4H-chromen-6-yl)-acetic acidKi50000.0 [1]
2-Adamantan-1-yl-4-oxo-4H-chromene-6-carboxylic acid methyl esterIC50180.0 [1], 530.0 [2], 30000.0 [3]
2-Adamantan-1-yl-4-oxo-4H-chromene-6-carboxylic acid methyl esterKi50000.0 [1]
2-Adamantan-1-yl-6-(2-hydroxy-acetyl)-chromen-4-oneIC50180.0 [1], 530.0 [2], 30000.0 [3]
2-Adamantan-1-yl-6-(2-hydroxy-acetyl)-chromen-4-oneKi3200.0 [1]
3-Bromo-N-[(8R,9S,13S,14S,17S)-3-hydroxy-13-methyl-6,7,8,9,11,12,14,15,16,17-decahydrocyclopenta[a]phenanthren-17-yl]benzenesulfonamideIC5025.0 [1]
3-Bromo-N-[(8R,9S,13S,14S,17S)-3-hydroxy-13-methyl-6,7,8,9,11,12,14,15,16,17-decahydrocyclopenta[a]phenanthren-17-yl]benzenesulfonamideKi23.0 [1], 108.0 [2]
Estrone sulfateIC507600.0 [1]
Estrone sulfateKi60000.0 [1]
4-{[(4-Cyanophenyl)(4H-1,2,4-triazol-4-YL)amino]methyl}phenyl sulfamateIC50227.0 [1], 277.0 [2]
(8R,9S,13S,14S,17R)-17-[(3-Bromophenyl)methyl]-13-methyl-7,8,9,11,12,14,15,16-octahydro-6H-cyclopenta[a]phenanthrene-3,17-diolIC5024.0 [1]
Sulfamic acid 4-[(E)-(3-phenyl-acryloyl)]-phenyl esterIC503400.0 [1], 263000.0 [2]
Sulfamic acid 4-benzoyl-phenyl esterIC505100.0 [1], 63000.0 [2]
Sulfamic acid 4-heptanoyl-phenyl esterIC503400.0 [1], 5000.0 [2]
4-Formylphenyl sulfamateIC503400.0 [1], 254000.0 [2]
Sulfamic acid 4-acetylphenyl esterIC503400.0 [1], 302000.0 [2]
[(8R,9S,13S,14S)-13-Methyl-2-methylsulfanyl-17-oxo-7,8,9,11,12,14,15,16-octahydro-6H-cyclopenta[a]phenanthren-3-yl] sulfamateIC5044.0 [1], 120.0 [2], 120000.0 [3]
(4-{[4-(Sulfamoyloxy)phenyl](1H-1,2,4-triazol-1-yl)methyl}phenyl) sulfamateIC5010000.0 [1]
{2-Bromo-4-[(4-cyanophenyl)(1H-1,2,4-triazol-1-yl)methyl]phenyl} sulfamateIC502600.0 [1]
Sulfamic acid 4-pentanoyl-phenyl esterIC503400.0 [1], 20900.0 [2]
Sulfamic acid 4-phenylacetyl-phenyl esterIC503400.0 [1], 33000.0 [2]
Sulfamic acid 4-butyryl-phenyl esterIC503400.0 [1], 39800.0 [2]
Sulfamic acid 4-decanoyl-phenyl esterIC503400.0 [1], 13000.0 [2]
3-Chloro-2'-Cyano-5'-(1h-1,2,4-Triazol-1-Ylmethyl)biphenyl-4-Yl SulfamateIC505.5 [1]
Sulfamic acid 4-octanoyl-phenyl esterIC503400.0 [1], 5600.0 [2]
Sulfamic acid 4-nonanoyl-phenyl esterIC503400.0 [1]
(9-Oxo-8-oxatricyclo[8.8.0.02,7]octadeca-1(10),2(7),3,5-tetraen-5-yl) sulfamateIC501.0 [1]
[(8R,9S,13S,14S,17R)-17-Benzyl-17-hydroxy-13-methyl-7,8,9,11,12,14,15,16-octahydro-6H-cyclopenta[a]phenanthren-3-yl] sulfamateIC500.39 [1], 1.4 [2], 4.1 [3]
[(8R,9S,13S,14S)-4-Bromo-13-methyl-17-oxo-7,8,9,11,12,14,15,16-octahydro-6H-cyclopenta[a]phenanthren-3-yl] sulfamateIC5042.0 [1], 1200.0 [2]
Sulfamic acid 2-adamantan-1-yl-4-oxo-4H-chromen-6-yl esterIC505.6 [1], 20.0 [2]
Sulfamic acid 2-adamantan-1-yl-4-oxo-4H-chromen-6-yl esterKi190.0 [1]
Tert-butyl 4-[(4-bromo-2,5-dichlorothiophen-3-yl)sulfonylcarbamoyl]piperidine-1-carboxylateIC5026.0 [1], 270.0 [2]
Tert-butyl 4-[(4-bromo-2,5-dichlorothiophen-3-yl)sulfonylcarbamoyl]piperidine-1-carboxylateKi12.0 [1]
[3-Chloro-4-[5-(2,6-difluoro-3-hydroxybenzoyl)thiophen-2-yl]phenyl] sulfamateIC503.4 [1], 3.9 [2], 19.4 [3]
[2-Chloro-4-[5-(2,6-difluoro-3-hydroxybenzoyl)thiophen-2-yl]phenyl] sulfamateIC5015.6 [1], 16.4 [2], 143.1 [3]
[4-[5-(2,6-Difluoro-3-hydroxybenzoyl)thiophen-2-yl]-3-fluorophenyl] sulfamateIC502.1 [1], 3.1 [2], 19.5 [3]
[4-[5-(2,6-Difluoro-3-hydroxybenzoyl)thiophen-2-yl]-2-fluorophenyl] sulfamateIC505.1 [1], 5.7 [2], 81.8 [3]
4-(4-Chloro-benzenesulfonylaminocarbonyl)-piperazine-1-carboxylic acid tert-butyl esterIC503600.0 [1], 12000.0 [2]
4-(4-Chloro-benzenesulfonylaminocarbonyl)-piperazine-1-carboxylic acid tert-butyl esterKi14500.0 [1]
4-(4-Chloro-benzenesulfonylaminocarbonyl)-piperidine-1-carboxylic acid tert-butyl esterIC508600.0 [1], 9800.0 [2]
4-(4-Chloro-benzenesulfonylaminocarbonyl)-piperidine-1-carboxylic acid tert-butyl esterKi16100.0 [1]
Tert-butyl 4-[[3,5-bis(trifluoromethyl)phenyl]sulfonylcarbamoyl]piperidine-1-carboxylateIC50210.0 [1], 780.0 [2]
Tert-butyl 4-[[3,5-bis(trifluoromethyl)phenyl]sulfonylcarbamoyl]piperidine-1-carboxylateKi220.0 [1]
EstradiolIC5084000.0 [1]
(9beta,13alpha,14beta,17alpha)-2-Methoxyestra-1,3,5(10)-Triene-3,17-Diyl DisulfamateIC5039.0 [1]
Phenyl sulfamateIC5010000000.0 [1], 100000000.0 [2]
Sulfamic acid, 4-(2-((1-oxotetradecyl)amino)ethyl)phenyl esterIC5055.8 [1]
2-MeOEMATEIC5030.0 [1], 42.0 [2]
Estradiol 3-sulfamateIC5016.0 [1]
[(4As,4bR,10bS,12aS)-12a-methyl-1,3-dioxo-2-propyl-4,4a,4b,5,6,10b,11,12-octahydronaphtho[2,1-f]isoquinolin-8-yl] sulfamateIC501.0 [1]
4-[(3-Bromo-4-O-sulfamoylbenzyl)(4-cyanophenyl)amino]-4H-[1,2,4]-triazoleIC5039.0 [1]
(9beta,14beta,17beta)-17-Hydroxy-2-Methoxyestra-1,3,5(10)-Trien-3-Yl SulfamateIC5016.0 [1], 34.0 [2]
4-Bromophenyl SulfamateIC50912000.0 [1]
Sulfamic acid 5,6,7,8-tetrahydro-naphthalen-2-yl esterIC501000.0 [1]
4-Chlorophenyl SulfamateIC501584800.0 [1], 1585000.0 [2]
(9beta)-2-Ethyl-17-Oxoestra-1(10),2,4-Trien-3-Yl SulfamateIC50820.0 [1], 1800.0 [2]
Sulfamic acid, 4-cyanophenyl esterIC50300000.0 [1]
4-{4-[(Aminosulfonyl)oxy]benzoyl}phenyl sulfamateIC50190.0 [1]
3-Nitrophenyl SulfamateIC50120000.0 [1]
[(8R,9S,13S,14S)-13-Methyl-17-oxo-7,8,9,11,12,14,15,16-octahydro-6H-cyclopenta[a]phenanthren-3-yl] formateIC50420.0 [1]
4-Nitrophenyl sulfamateIC50330000.0 [1]
4-Methylphenyl sulfamateIC5010000000.0 [1], 100000000.0 [2]
[(8R,9S,13S,14S,17R)-17-Benzyl-17-hydroxy-2-methoxy-13-methyl-7,8,9,11,12,14,15,16-octahydro-6H-cyclopenta[a]phenanthren-3-yl] sulfamateIC500.02 [1], 0.05 [2]
(8R,9S,13S,14S)-3-Hydroxy-13-methyl-17-oxo-7,8,9,11,12,14,15,16-octahydro-6H-cyclopenta[a]phenanthrene-4-carbaldehydeIC501500.0 [1]
(8R,9S,13S,14S)-3-Hydroxy-13-methyl-17-oxo-7,8,9,11,12,14,15,16-octahydro-6H-cyclopenta[a]phenanthrene-4-carbaldehydeKi1500.0 [1]
4-Fluorophenyl SulfamateIC50537000.0 [1], 100000000.0 [2]
(8R,9S,13S,14S,17R)-13-Methyl-17-[[3-(trifluoromethyl)phenyl]methyl]-7,8,9,11,12,14,15,16-octahydro-6H-cyclopenta[a]phenanthrene-3,17-diolIC50126.0 [1]
Items per page: 1 - 10 of 100
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References

This online tool may be cited as follows

MLA

"Quest Database™ Steryl-sulfatase Inhibitors (IC50, Ki)." AAT Bioquest, Inc., 9 May. 2024, https://www.aatbio.com/data-sets/steryl-sulfatase-inhibitors-ic50-ki.

APA

AAT Bioquest, Inc. (2024, May 9). Quest Database™ Steryl-sulfatase Inhibitors (IC50, Ki). AAT Bioquest. https://www.aatbio.com/data-sets/steryl-sulfatase-inhibitors-ic50-ki.
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