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Sulfonylurea receptors; K-ATP channels Inhibitors (IC50, Ki)

Structure
▲
▼
Compound Name
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▼
Standard Type
▲
▼
Standard Values (in nM)
▲
▼
N-[4-(Benzenesulfonyl)phenyl]-3,3,3-trifluoro-2-hydroxy-2-methylpropanamideIC5044.0 [1], 470.0 [2]
N-(4-Benzoylphenyl)-3,3,3-trifluoro-2-hydroxy-2-methylpropanamideIC5082.0 [1], 3000.0 [2], 3800.0 [3]
CromakalimIC50500.0 [1], 1500.0 [2]
(+/-)-CromakalimIC5020.0 [1], 570.0 [2]
3,3,3-Trifluoro-2-hydroxy-2-methyl-N-(4-pyridin-3-ylsulfonylphenyl)propanamideIC50130.0 [1], 3500.0 [2]
3,3,3-Trifluoro-2-hydroxy-N-[4-[(Z)-N-methoxy-C-phenylcarbonimidoyl]phenyl]-2-methylpropanamideIC5030000.0 [1]
3,3,3-Trifluoro-2-hydroxy-2-methyl-N-(4-pyridin-4-ylsulfonylphenyl)propanamideIC50540.0 [1], 2700.0 [2]
3,3,3-Trifluoro-2-hydroxy-2-methyl-N-[4-[methyl(phenyl)sulfamoyl]phenyl]propanamideIC501970.0 [1], 2000.0 [2]
N-[4-(Diphenylsulfamoyl)phenyl]-3,3,3-trifluoro-2-hydroxy-2-methylpropanamideIC5030000.0 [1]
(2S)-N-(4-Benzoylphenyl)-3,3,3-trifluoro-2-hydroxy-2-methylpropanamideIC501600.0 [1]
N-(4-Benzoyl-2-chlorophenyl)-3,3,3-trifluoro-2-hydroxy-2-methylpropanamideIC5030000.0 [1]
3,3,3-Trifluoro-2-hydroxy-2-methyl-N-(4-nitro-3-phenylsulfanylphenyl)propanamideIC5016000.0 [1]
3,3,3-Trifluoro-2-hydroxy-N-[4-(4-hydroxyphenyl)sulfonylphenyl]-2-methylpropanamideIC5030000.0 [1]
N-[3-(Benzenesulfonyl)-4-cyanophenyl]-3,3,3-trifluoro-2-hydroxy-2-methylpropanamideIC502600.0 [1]
3,3,3-Trifluoro-N-[4-(3-fluorobenzoyl)phenyl]-2-hydroxy-2-methylpropanamideIC502600.0 [1]
3,3,3-Trifluoro-N-[4-(3-fluorophenyl)sulfonylphenyl]-2-hydroxy-2-methylpropanamideIC503400.0 [1]
3,3,3-Trifluoro-N-[4-(2-fluorobenzoyl)phenyl]-2-hydroxy-2-methylpropanamideIC502300.0 [1]
3,3,3-Trifluoro-2-hydroxy-2-methyl-N-[4-(1,3-thiazol-2-ylsulfonyl)phenyl]propanamideIC501400.0 [1]
5-(Benzenesulfonyl)-2-[(3,3,3-trifluoro-2-hydroxy-2-methylpropanoyl)amino]benzoic acidIC5030000.0 [1]
3,3,3-Trifluoro-2-hydroxy-2-methyl-N-[4-(3-methylbenzoyl)phenyl]propanamideIC5030000.0 [1]
N-(9,10-Dioxoanthracen-2-yl)-3,3,3-trifluoro-2-hydroxy-2-methylpropanamideIC5030000.0 [1]
3,3,3-Trifluoro-2-hydroxy-2-methyl-N-(4-pyrimidin-5-ylsulfonylphenyl)propanamideIC5030000.0 [1]
3,3,3-Trifluoro-2-hydroxy-N-[4-(3-hydroxyphenyl)sulfonylphenyl]-2-methylpropanamideIC5018000.0 [1]
3,3,3-Trifluoro-N-[4-(4-fluorophenyl)sulfonylphenyl]-2-hydroxy-2-methylpropanamideIC508600.0 [1]
2-(Benzenesulfonyl)-5-[(3,3,3-trifluoro-2-hydroxy-2-methylpropanoyl)amino]benzoic acidIC5030000.0 [1]
N-(4-Diphenylphosphorylphenyl)-3,3,3-trifluoro-2-hydroxy-2-methylpropanamideIC5030000.0 [1]
3,3,3-Trifluoro-2-hydroxy-N-(3-hydroxy-4-pyridin-4-ylsulfonylphenyl)-2-methylpropanamideIC501300.0 [1]
N-[4-(Benzenesulfonyl)-3-cyanophenyl]-3,3,3-trifluoro-2-hydroxy-2-methylpropanamideIC503800.0 [1]
N-[4-(Benzenesulfonyl)-3-chlorophenyl]-3,3,3-trifluoro-2-hydroxy-2-methylpropanamideIC502200.0 [1]
N-[4-(Benzenesulfonyl)-2-nitrophenyl]-3,3,3-trifluoro-2-hydroxy-2-methylpropanamideIC507900.0 [1]
(2R)-N-(4-Benzoylphenyl)-3,3,3-trifluoro-2-hydroxy-2-methylpropanamideIC5030000.0 [1]
N-[3-(Benzenesulfonyl)phenyl]-3,3,3-trifluoro-2-hydroxy-2-methylpropanamideIC5030000.0 [1]
N-[5-(Benzenesulfonyl)pyridin-2-yl]-3,3,3-trifluoro-2-hydroxy-2-methylpropanamideIC506200.0 [1]
3,3,3-Trifluoro-N-[4-(2-fluorophenyl)sulfonylphenyl]-2-hydroxy-2-methylpropanamideIC501300.0 [1]
3,3,3-Trifluoro-2-hydroxy-N-[4-(2-methoxyphenyl)sulfonylphenyl]-2-methylpropanamideIC501600.0 [1]
3,3,3-Trifluoro-2-hydroxy-2-methyl-N-[4-(4-nitrophenyl)sulfonylphenyl]propanamideIC5030000.0 [1]
3,3,3-Trifluoro-2-hydroxy-2-methyl-N-(4-pyridin-2-ylsulfonylphenyl)propanamideIC50600.0 [1]
3,3,3-Trifluoro-2-hydroxy-2-methyl-N-[4-(2-methylphenyl)sulfonylphenyl]propanamideIC505100.0 [1]
3,3,3-Trifluoro-2-hydroxy-2-methyl-N-[4-(3-methylphenyl)sulfonylphenyl]propanamideIC502200.0 [1]
N-[4-(4-Cyanophenyl)sulfonylphenyl]-3,3,3-trifluoro-2-hydroxy-2-methylpropanamideIC5030000.0 [1]
N-[4-(Benzenesulfonyl)-3-nitrophenyl]-3,3,3-trifluoro-2-hydroxy-2-methylpropanamideIC5030000.0 [1]
N-(5,5-Dioxodibenzothiophen-2-yl)-3,3,3-trifluoro-2-hydroxy-2-methylpropanamideIC5024000.0 [1]
N-[4-(2-Cyanophenyl)sulfonylphenyl]-3,3,3-trifluoro-2-hydroxy-2-methylpropanamideIC501100.0 [1]
N-[4-(Benzenesulfonyl)-3-(trifluoromethyl)phenyl]-3,3,3-trifluoro-2-hydroxy-2-methylpropanamideIC5030000.0 [1]
N-(5-Benzoylthiophen-2-yl)-3,3,3-trifluoro-2-hydroxy-2-methylpropanamideIC5030000.0 [1]
3,3,3-Trifluoro-N-[4-(4-fluorobenzoyl)phenyl]-2-hydroxy-2-methylpropanamideIC5014000.0 [1]
3,3,3-Trifluoro-2-hydroxy-2-methyl-N-[4-(4-methylphenyl)sulfonylphenyl]propanamideIC5030000.0 [1]
N-[4-(4-Bromophenyl)sulfonylphenyl]-3,3,3-trifluoro-2-hydroxy-2-methylpropanamideIC5030000.0 [1]
N-(4-Cyano-3-phenylsulfanylphenyl)-3,3,3-trifluoro-2-hydroxy-2-methylpropanamideIC508300.0 [1]
3,3,3-Trifluoro-2-hydroxy-2-methyl-N-[4-(1,3-thiazol-5-ylsulfonyl)phenyl]propanamideIC507700.0 [1]
3,3,3-Trifluoro-2-hydroxy-2-methyl-N-[4-[3-(trifluoromethyl)phenyl]sulfonylphenyl]propanamideIC5030000.0 [1]
N-(4-Benzoyl-3-hydroxyphenyl)-3,3,3-trifluoro-2-hydroxy-2-methylpropanamideIC504200.0 [1]
3,3,3-Trifluoro-2-hydroxy-2-methyl-N-(4-pyrazin-2-ylsulfonylphenyl)propanamideIC5012000.0 [1]
3,3,3-Trifluoro-2-hydroxy-2-methyl-N-(9,10,10-trioxothioxanthen-3-yl)propanamideIC5030000.0 [1]
N-(4-Benzoyl-3-fluorophenyl)-3,3,3-trifluoro-2-hydroxy-2-methylpropanamideIC502700.0 [1]
N-[4-(Benzenesulfonyl)-3-methoxyphenyl]-3,3,3-trifluoro-2-hydroxy-2-methylpropanamideIC505900.0 [1]
N-[4-(2-Chlorophenyl)sulfonylphenyl]-3,3,3-trifluoro-2-hydroxy-2-methylpropanamideIC502300.0 [1]
N-[3-(Benzenesulfonyl)-4-nitrophenyl]-3,3,3-trifluoro-2-hydroxy-2-methylpropanamideIC5030000.0 [1]
N-[4-(3-Chlorobenzoyl)phenyl]-3,3,3-trifluoro-2-hydroxy-2-methylpropanamideIC5030000.0 [1]
N-[4-(Benzenesulfonyl)-3-methylphenyl]-3,3,3-trifluoro-2-hydroxy-2-methylpropanamideIC501600.0 [1]
3,3,3-Trifluoro-2-hydroxy-N-[4-(2-hydroxyphenyl)sulfonylphenyl]-2-methylpropanamideIC503090.0 [1]
N-[4-(3-Chlorophenyl)sulfonylphenyl]-3,3,3-trifluoro-2-hydroxy-2-methylpropanamideIC5010000.0 [1]
N-(4-Benzoyl-2-hydroxyphenyl)-3,3,3-trifluoro-2-hydroxy-2-methylpropanamideIC5015000.0 [1]
N-[4-(Benzenesulfonyl)-3-hydroxyphenyl]-3,3,3-trifluoro-2-hydroxy-2-methylpropanamideIC50430.0 [1]
N-[4-(Benzenesulfonyl)-3-fluorophenyl]-3,3,3-trifluoro-2-hydroxy-2-methylpropanamideIC501800.0 [1]
3,3,3-Trifluoro-2-hydroxy-N-[4-(3-methoxyphenyl)sulfonylphenyl]-2-methylpropanamideIC5016000.0 [1]
3,3,3-Trifluoro-2-hydroxy-N-[4-(4-methoxyphenyl)sulfonylphenyl]-2-methylpropanamideIC5030000.0 [1]
3,3,3-Trifluoro-2-hydroxy-N-[4-[hydroxy(phenyl)methyl]phenyl]-2-methylpropanamideIC5030000.0 [1]
(2S)-N-(4-Benzoyl-2-methylphenyl)-3,3,3-trifluoro-2-hydroxy-2-methylpropanamideIC502600.0 [1]
(2R)-3,3,3-Trifluoro-2-hydroxy-2-methyl-N-(4-pyridin-4-ylsulfonylphenyl)propanamideIC5030000.0 [1]
(2S)-3,3,3-Trifluoro-2-hydroxy-2-methyl-N-(4-pyridin-4-ylsulfonylphenyl)propanamideIC501600.0 [1]
3,3,3-Trifluoro-2-hydroxy-2-methyl-N-(2-methyl-1,1,3-trioxo-1,2-benzothiazol-5-yl)propanamideIC5026000.0 [1]
3,3,3-Trifluoro-2-hydroxy-2-methyl-N-(1,1,3-trioxo-1,2-benzothiazol-5-yl)propanamideIC5030000.0 [1]
N-(4-Benzoyl-2,6-dimethylphenyl)-3,3,3-trifluoro-2-hydroxy-2-methylpropanamideIC5030000.0 [1]
N-(4-Benzoyl-2-methoxyphenyl)-3,3,3-trifluoro-2-hydroxy-2-methylpropanamideIC506100.0 [1]
CID 9819831IC505000.0 [1]
CID 9841562IC5011000.0 [1]
3,3,3-Trifluoro-2-hydroxy-2-methyl-N-(4-piperidin-1-ylsulfonylphenyl)propanamideIC509250.0 [1]
N-(4-Benzoyl-2-bromophenyl)-3,3,3-trifluoro-2-hydroxy-2-methylpropanamideIC5030000.0 [1]
3,3,3-Trifluoro-2-hydroxy-2-methyl-N-(4-sulfamoylphenyl)propanamideIC5012800.0 [1]
N-(4-Benzoyl-2-cyanophenyl)-3,3,3-trifluoro-2-hydroxy-2-methylpropanamideIC503800.0 [1]
N-[4-[Bis(2-methylpropyl)sulfamoyl]phenyl]-3,3,3-trifluoro-2-hydroxy-2-methylpropanamideIC5030000.0 [1]
N-[4-[Di(butan-2-yl)sulfamoyl]phenyl]-3,3,3-trifluoro-2-hydroxy-2-methylpropanamideIC5030000.0 [1]
3,3,3-Trifluoro-2-hydroxy-2-methyl-N-[4-(phenylsulfamoyl)phenyl]propanamideIC5030000.0 [1]
3,3,3-Trifluoro-2-hydroxy-2-methyl-N-(4-piperazin-1-ylsulfonylphenyl)propanamideIC5030000.0 [1]
3,3,3-Trifluoro-2-hydroxy-2-methyl-N-(4-morpholin-4-ylsulfonylphenyl)propanamideIC505850.0 [1]
3,3,3-Trifluoro-2-hydroxy-N-[4-[(R)-hydroxy(phenyl)methyl]phenyl]-2-methylpropanamideIC5030000.0 [1]
N,N-Diethyl-4-[(3,3,3-trifluoro-2-hydroxy-2-methylpropanoyl)amino]benzamideIC5030000.0 [1]
3,3,3-Trifluoro-2-hydroxy-2-methyl-N-(4-phenylsulfanylphenyl)propanamideIC5030000.0 [1]
3,3,3-Trifluoro-2-hydroxy-N-[4-[(Z)-N-hydroxy-C-phenylcarbonimidoyl]phenyl]-2-methylpropanamideIC5030000.0 [1]
3,3,3-Trifluoro-2-hydroxy-2-methyl-N-[4-(1-methyltetrazol-5-yl)phenyl]propanamideIC5030900.0 [1]
3,3,3-Trifluoro-2-hydroxy-2-methyl-N-[4-(2H-tetrazol-5-yl)phenyl]propanamideIC5030000.0 [1]
3,3,3-Trifluoro-2-hydroxy-N-[4-[(S)-hydroxy(phenyl)methyl]phenyl]-2-methylpropanamideIC5030000.0 [1]
N-[4-(Diethylsulfamoyl)phenyl]-3,3,3-trifluoro-2-hydroxy-2-methylpropanamideIC50810.0 [1]
N-[4-(Dipropylsulfamoyl)phenyl]-3,3,3-trifluoro-2-hydroxy-2-methylpropanamideIC506440.0 [1]
N-[4-(Dimethylsulfamoyl)phenyl]-3,3,3-trifluoro-2-hydroxy-2-methylpropanamideIC50480.0 [1]
2,2-Dimethyl-4-(1-oxidopyridin-1-ium-2-yl)-6-(1,1,2,2,2-pentafluoroethyl)naphthalen-1-oneIC502520.0 [1]
3,3,3-Trifluoro-2-hydroxy-2-methyl-N-(4-thiomorpholin-4-ylsulfonylphenyl)propanamideIC504580.0 [1]
3,3,3-Trifluoro-2-hydroxy-2-methyl-N-(4-pyrrolidin-1-ylsulfonylphenyl)propanamideIC50880.0 [1]
2-(3,3-Dimethyl-4-oxo-7-cyano-3,4-dihydronaphthalene-1-yl)pyridine 1-oxideIC503600.0 [1]
Items per page: 1 - 10 of 100
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References

This online tool may be cited as follows

MLA

"Quest Database™ Sulfonylurea receptors; K-ATP channels Inhibitors (IC50, Ki)." AAT Bioquest, Inc., 10 May. 2024, https://www.aatbio.com/data-sets/sulfonylurea-receptors-k-atp-channels-inhibitors-ic50-ki.

APA

AAT Bioquest, Inc. (2024, May 10). Quest Database™ Sulfonylurea receptors; K-ATP channels Inhibitors (IC50, Ki). AAT Bioquest. https://www.aatbio.com/data-sets/sulfonylurea-receptors-k-atp-channels-inhibitors-ic50-ki.
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