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T-cell protein-tyrosine phosphatase Inhibitors (IC50, Ki)

Structure
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Compound Name
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Standard Type
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Standard Values (in nM)
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Oleanolic acidIC505460.0 [1]
5-{2-Fluoro-5-[3-(3-hydroxy-2-methoxycarbonyl-phenoxy)-propenyl]-phenyl}-isoxazole-3-carboxylic acidIC50164000.0 [1]
5-{2-Fluoro-5-[3-(3-hydroxy-2-methoxycarbonyl-phenoxy)-propenyl]-phenyl}-isoxazole-3-carboxylic acidKi164000.0 [1]
2-(Oxalyl-amino)-4,5,6,7-tetrahydro-thieno[2,3-C]pyridine-3-carboxylic acidKi290.0 [1], 710.0 [2], 9400.0 [3], 10000.0 [4]
Ursolic acidIC502400.0 [1], 3330.0 [2], 6700.0 [3]
(3S)-4-[[(2S)-1-Amino-3-[4-[difluoro(phosphono)methyl]phenyl]-1-oxopropan-2-yl]amino]-3-[[2-[4-[difluoro(phosphono)methyl]phenyl]acetyl]amino]-4-oxobutanoic acidKi24.0 [1], 26.0 [2]
2-[4-[[4-[(4-Oxalophenoxy)methyl]phenyl]methoxy]phenyl]-2-oxoacetic acidIC505350.0 [1], 6240.0 [2]
2-[4-[(2S)-2-Acetamido-3-[4-(3-hydroxy-2-methoxycarbonylphenoxy)butylamino]-3-oxopropyl]-2-hydroxyphenoxy]acetic acidKi182000.0 [1]
4-Bromo-3-(carboxymethoxy)-5-phenylthiophene-2-carboxylic acidKi320.0 [1], 1300.0 [2], 3200.0 [3]
[3-[3-[(3S)-3-(Methylcarbamoyl)-7-(sulfoamino)-3,4-dihydro-1H-isoquinolin-2-yl]-3-oxopropyl]phenyl]sulfamic acidIC509400.0 [1], 9900.0 [2]
2-[4-[2-Acetamido-3-[4-(3-hydroxy-2-methoxycarbonylphenoxy)butylamino]-3-oxopropyl]-2-ethyl-N-oxaloanilino]benzoic acidKi65.0 [1]
5-(3-(3-(3-Hydroxy-2-(methoxycarbonyl)phenoxy)prop-1-enyl)phenyl)isoxazole-3-carboxylic acidKi202000.0 [1]
5-[(3-Carboxy-4-hydroxy-5-phenylphenyl)methyl]-2-hydroxy-3-phenylbenzoic acidIC50291000.0 [1]
5-[(3-Carboxy-4-hydroxy-5-phenylphenyl)methyl]-2-hydroxy-3-phenylbenzoic acidKi64000.0 [1]
4-Amino-5-[3-[(E)-3-(3-hydroxy-2-methoxycarbonylphenoxy)prop-1-enyl]phenyl]-1,2-oxazole-3-carboxylic acidIC5030000.0 [1]
4-Amino-5-[3-[(E)-3-(3-hydroxy-2-methoxycarbonylphenoxy)prop-1-enyl]phenyl]-1,2-oxazole-3-carboxylic acidKi30000.0 [1]
[6-[4-[2-(Benzotriazol-1-yl)-3-[4-[difluoro(phosphono)methyl]phenyl]-2-phenylpropyl]phenyl]-2-(1-methoxy-3-methylbutyl)quinolin-8-yl]phosphonic acidIC5036.0 [1], 930.0 [2]
5-[3-[(1-Benzylsulfonylpiperidin-4-yl)amino]phenyl]-4-bromo-3-(carboxymethoxy)thiophene-2-carboxylic acidKi5.0 [1]
4-Bromo-3-(carboxymethoxy)-5-[4-[[oxo(3-pyridinyl)methyl]amino]phenyl]-2-thiophenecarboxylic acidKi680.0 [1], 820.0 [2]
3-[(3-Carboxy-2-hydroxy-5-phenylphenyl)methyl]-2-hydroxy-5-phenylbenzoic acidIC50156000.0 [1]
3-[(3-Carboxy-2-hydroxy-5-phenylphenyl)methyl]-2-hydroxy-5-phenylbenzoic acidKi89000.0 [1]
[3-[4-[2-(Benzotriazol-1-yl)-3-[4-[difluoro(phosphono)methyl]phenyl]-2-phenylpropyl]phenyl]phenyl]phosphonic acidIC503.0 [1]
4-Bromo-5-[4-[(2-carboxyacetyl)amino]phenyl]-3-(carboxymethoxy)thiophene-2-carboxylic acidKi140.0 [1], 180.0 [2]
4-Bromo-3-(carboxymethoxy)-5-[3-[(3,3,5,5-tetramethylcyclohexyl)amino]phenyl]thiophene-2-carboxylic acidKi26.0 [1], 36.0 [2]
4-Bromo-3-(carboxymethoxy)-5-[4-(dimethylamino)phenyl]thiophene-2-carboxylic acidKi1000.0 [1], 1600.0 [2]
Isochroman mono-carboxylic acidIC501821.0 [1]
5-[3-[(E)-3-(3-Hydroxy-2-methoxycarbonylphenoxy)prop-1-enyl]phenyl]-4-(hydroxymethyl)-1,2-oxazole-3-carboxylic acidIC5019200.0 [1]
5-[3-[(E)-3-(3-Hydroxy-2-methoxycarbonylphenoxy)prop-1-enyl]phenyl]-4-(hydroxymethyl)-1,2-oxazole-3-carboxylic acidKi19200.0 [1]
7-(Biphenyl-4-yl)-4-oxo-4H-chromene-3-carbaldehydeKi4300.0 [1], 51000.0 [2]
EnoxoloneIC5020000.0 [1]
Chlorogenic acidIC5077900.0 [1]
Lithocholic acidIC5020450.0 [1]
Maslinic acidIC5019470.0 [1]
CryptotanshinoneIC5055700.0 [1]
Asiatic acidIC5020000.0 [1]
beta-Boswellic acidIC5020000.0 [1]
alpha-TocopherolquinoneIC5035090.0 [1]
Corosolic acidIC5011310.0 [1]
[(2R,3R,4S,5R,6R)-3,4,5,6-Tetrakis[(3,4,5-trihydroxybenzoyl)oxy]oxan-2-yl]methyl 3,4,5-trihydroxybenzoateIC5070.0 [1]
11-Keto-beta-boswellic acidIC509450.0 [1]
Oleanonic acidIC505630.0 [1]
Madecassic acidIC5020000.0 [1]
(5R)-3-Hexadecanoyl-4-hydroxy-5-(hydroxymethyl)furan-2(5H)-oneIC505100.0 [1]
5-((E)-2-{4-[(E)-2-(3-Carboxy-4-hydroxyphenyl)vinyl]-phenyl}vinyl)-2-hydroxybenzoic acidIC5027000.0 [1]
2-(Oxalyl-amino)-benzoic acidKi23000.0 [1]
(4As,6aR,6aS,6bR,8aR,10S,12aR,14bS)-10-(3-carboxy-3-methylbutanoyl)oxy-2,2,6a,6b,9,9,12a-heptamethyl-1,3,4,5,6,6a,7,8,8a,10,11,12,13,14b-tetradecahydropicene-4a-carboxylic acidIC501380.0 [1]
3,4,6-Tribromo-5-[(2,3,6-tribromo-4,5-dihydroxyphenyl)methyl]benzene-1,2-diolIC5050000.0 [1]
3-Epioleanolic acidIC505100.0 [1]
Succinyl oleanolic acidIC505360.0 [1]
CID 71734765IC5011300.0 [1]
5-Iodo-2-(oxaloamino)benzoic acidKi14000.0 [1]
[(3-Bromo-7-cyano-2-naphthalenyl)-difluoromethyl]phosphonic acidIC50120.0 [1]
6-Hydroxy-3-[1-[2-(4-morpholin-4-ylanilino)-2-oxoethyl]triazol-4-yl]-2-phenyl-1-benzofuran-5-carboxylic acidIC5022000.0 [1]
6-(Oxalyl-amino)-1H-indole-5-carboxylic acidKi14000.0 [1]
2-(Oxalyl-amino)-4,7-dihydro-5H-thieno[2,3-C]pyran-3-carboxylic acidKi14000.0 [1]
2-(Carboxyformamido)-4,5,6,7-tetrahydrobenzo[b]thiophene-3-carboxylic acidKi8100.0 [1]
1-Oxobenzo[f]chromene-2-carbaldehydeIC50780000.0 [1]
(2-Bromo-4-(3-oxo-2,3-diphenylpropyl)phenyl)difluoromethylphosphonic acidIC50120.0 [1]
2-[4-[2-Acetamido-3-[[5-[[(1S)-1-carboxy-3-methylsulfanylpropyl]amino]-5-oxopentyl]amino]-3-oxopropyl]-2-ethyl-N-oxaloanilino]benzoic acidKi380.0 [1]
4-[4-(2,4-Dihydroxy-6-propylbenzoyl)oxy-2-hydroxy-6-propylbenzoyl]oxy-2-hydroxy-6-propylbenzoic acidIC5017680.0 [1]
CID 10348668IC505000.0 [1]
1H-Indole-7-carboxylic acid, 6-[(carboxycarbonyl)amino]-Ki8000.0 [1]
2-(Carboxyformamido)thiophene-3-carboxylic acidKi62000.0 [1]
3-(Carboxyformamido)thiophene-2-carboxylic acidKi58000.0 [1]
Furospongin-1IC509600.0 [1]
2-[4-[(2S)-3-[4-(3-Hydroxy-2-methoxycarbonylphenoxy)butylamino]-3-oxo-2-(prop-2-enoxycarbonylamino)propyl]-N-oxaloanilino]benzoic acidKi470.0 [1]
2-[4-[2-Acetamido-3-oxo-3-(pentylamino)propyl]-2-ethyl-N-oxaloanilino]benzoic acidKi900.0 [1]
(1R,2R,11R,14R,15S,18S,23S)-2,10,10,14,15,21,21-Heptamethyl-5,8-diazahexacyclo[12.12.0.02,11.04,9.015,24.018,23]hexacosa-4,6,8,24-tetraene-18-carboxylic acidIC508310.0 [1]
(1R,2R,15R,18R,19S,22S,27S)-2,14,14,18,19,25,25-Heptamethyl-5,12-diazaheptacyclo[16.12.0.02,15.04,13.06,11.019,28.022,27]triaconta-4,6,8,10,12,28-hexaene-22-carboxylic acidIC505880.0 [1]
(1R,2R,14R,17R,18S,21S,26S)-2,13,13,17,18,24,24-Heptamethyl-11-azaheptacyclo[15.12.0.02,14.04,12.05,10.018,27.021,26]nonacosa-4(12),5,7,9,27-pentaene-21-carboxylic acidIC501600.0 [1]
N-[(1S)-1-(1H-Benzimidazol-2-yl)-2-[3-methyl-4-(1,1,4-trioxo-1,2,5-thiadiazolidin-2-yl)phenyl]ethyl]benzenesulfonamideIC50150.0 [1]
5-(13-(3-Furanyl)-2,6,10-trimethyl-6,10-tridecadienylidene)-4-hydroxy-3-methyl-2(5H)-furanoneIC50800.0 [1]
[4-[(2S)-3-(Methylamino)-2-[(2-methylpropan-2-yl)oxycarbonylamino]-3-oxopropyl]phenyl]sulfamic acidIC5080100.0 [1]
2-[4-[(2S)-2-Acetamido-3-[4-(3-hydroxy-2-methoxycarbonylphenoxy)butylamino]-3-oxopropyl]-2-ethyl-N-oxaloanilino]benzoic acidKi65.0 [1]
(4As,6aR,6aS,6bR,8aR,10S,12aR,14bS)-2,2,6a,6b,9,9,12a-heptamethyl-10-oxalooxy-1,3,4,5,6,6a,7,8,8a,10,11,12,13,14b-tetradecahydropicene-4a-carboxylic acidIC504550.0 [1]
N-[(1S)-1-(1H-Benzimidazol-2-yl)-2-[3-methyl-4-[(5S)-1,1,3-trioxo-1,2-thiazolidin-5-yl]phenyl]ethyl]benzenesulfonamideIC5025.0 [1]
[[17-(Diphosphonomethyl)-26,28-dihydroxy-25,27-dipropoxy-5-pentacyclo[19.3.1.13,7.19,13.115,19]octacosa-1(25),3,5,7(28),9(27),10,12,15(26),16,18,21,23-dodecaenyl]-phosphonomethyl]phosphonic acidIC504900.0 [1]
[(26,28-Dihydroxy-25,27-dipropoxy-5-pentacyclo[19.3.1.13,7.19,13.115,19]octacosa-1(24),3,5,7(28),9,11,13(27),15(26),16,18,21(25),22-dodecaenyl)-phosphonomethyl]phosphonic acidIC509300.0 [1]
4-[5-[5-(1H-Indol-3-ylmethyl)-1,2,4-oxadiazol-3-yl]thiophen-2-yl]anilineIC50120000.0 [1]
4-[3-[5-(1H-Indol-3-ylmethyl)-1,2,4-oxadiazol-3-yl]phenyl]anilineIC50120000.0 [1]
5-[[2,5-Diethoxy-4-(methanesulfonamido)phenyl]methylcarbamoylamino]-2-ethoxy-N-(4-methylphenyl)benzamideIC50870.0 [1]
2-[4-[[3-Bromo-4-[difluoro(phosphono)methyl]phenyl]methyl-[[4-(dimethylsulfamoyl)phenyl]methyl]sulfamoyl]phenoxy]acetic acidIC5028.0 [1]
4-[5-(4-Benzyloxybenzylidene)-2,4-dioxothiazolidin-3-yl]methylbenzoic acidIC501300.0 [1]
2,4-Dihydroxy-6-propylbenzoic acidIC5020000.0 [1]
N-[1-(1H-Benzimidazol-2-yl)-2-[4-(1,1,3-trioxo-1,2-thiazolidin-5-yl)phenyl]ethyl]-3-(trifluoromethyl)benzenesulfonamideIC5043.0 [1]
(5Z)-3-(3-Chlorophenyl)-5-(4-hydroxy-3-methoxy-5-nitrobenzylidene)-2-thioxo-1,3-thiazolidin-4-oneIC505300.0 [1]
[(4As,5R,6S,8aR)-5-[(E)-5-(6-amino-9-methylpurin-9-ium-7-yl)-3-methylpent-3-enyl]-5,6,8a-trimethyl-3,4,4a,6,7,8-hexahydronaphthalen-1-yl]methyl 4-bromo-1H-pyrrole-2-carboxylateIC5016000.0 [1]
2-[4-[2-Acetamido-3-[[5-[[(1S)-1-carboxy-2-phenylethyl]amino]-5-oxopentyl]amino]-3-oxopropyl]-2-ethyl-N-oxaloanilino]benzoic acidKi160.0 [1]
2-[4-[2-Acetamido-3-[[5-[[(1S)-4-amino-1-carboxy-4-oxobutyl]amino]-5-oxopentyl]amino]-3-oxopropyl]-2-ethyl-N-oxaloanilino]benzoic acidKi270.0 [1]
2-[4-[2-Acetamido-3-[[5-[[(1S)-5-amino-1-carboxypentyl]amino]-5-oxopentyl]amino]-3-oxopropyl]-2-ethyl-N-oxaloanilino]benzoic acidKi820.0 [1]
2-[4-[2-Acetamido-3-[[5-[[(1S)-1-carboxypentyl]amino]-5-oxopentyl]amino]-3-oxopropyl]-2-ethyl-N-oxaloanilino]benzoic acidKi240.0 [1]
2-[4-[2-Acetamido-3-[[5-[[(1S)-1-carboxy-3-methylsulfonylpropyl]amino]-5-oxopentyl]amino]-3-oxopropyl]-2-ethyl-N-oxaloanilino]benzoic acidKi370.0 [1]
2-[4-[2-Acetamido-3-[[5-[[(1S)-1-carboxy-3-ethylsulfanylpropyl]amino]-5-oxopentyl]amino]-3-oxopropyl]-2-ethyl-N-oxaloanilino]benzoic acidKi510.0 [1]
2-[4-[(2S)-3-[4-(3-Hydroxy-2-methoxycarbonylphenoxy)butylamino]-2-[(2-methylpropan-2-yl)oxycarbonylamino]-3-oxopropyl]phenoxy]acetic acidKi200000.0 [1]
2-[4-[[3-Bromo-4-[difluoro(phosphono)methyl]phenyl]methyl-[[4-(thiadiazol-4-yl)phenyl]methyl]sulfamoyl]phenoxy]acetic acidIC50750.0 [1]
2-[5-[(4Ar,6aR,6aS,6bR,8aR,10S,12aR,14bR)-10-hydroxy-2,2,6a,6b,9,9,12a-heptamethyl-1,3,4,5,6,6a,7,8,8a,10,11,12,13,14b-tetradecahydropicen-4a-yl]pentanoylamino]-3-(2-chlorophenyl)propanoic acidIC50550.0 [1]
2-[5-[(4Ar,6aR,6aS,6bR,8aR,10S,12aR,14bR)-10-hydroxy-2,2,6a,6b,9,9,12a-heptamethyl-1,3,4,5,6,6a,7,8,8a,10,11,12,13,14b-tetradecahydropicen-4a-yl]pentanoylamino]-3-(2-methoxyphenyl)propanoic acidIC50450.0 [1]
2-[5-[(4Ar,6aR,6aS,6bR,8aR,10S,12aR,14bR)-10-hydroxy-2,2,6a,6b,9,9,12a-heptamethyl-1,3,4,5,6,6a,7,8,8a,10,11,12,13,14b-tetradecahydropicen-4a-yl]pentanoylamino]-3-(2,3-dimethoxyphenyl)propanoic acidIC50750.0 [1]
2-[5-[(4Ar,6aR,6aS,6bR,8aR,10S,12aR,14bR)-10-hydroxy-2,2,6a,6b,9,9,12a-heptamethyl-1,3,4,5,6,6a,7,8,8a,10,11,12,13,14b-tetradecahydropicen-4a-yl]pentanoylamino]-3-(3,5-dimethoxyphenyl)propanoic acidIC50850.0 [1]
(4As,6aR,6aS,6bR,8aR,10S,12aR,14bS)-2,2,6a,6b,9,9,12a-heptamethyl-10-phenylmethoxy-1,3,4,5,6,6a,7,8,8a,10,11,12,13,14b-tetradecahydropicene-4a-carboxylic acidIC502750.0 [1]
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References

This online tool may be cited as follows

MLA

"Quest Database™ T-cell protein-tyrosine phosphatase Inhibitors (IC50, Ki)." AAT Bioquest, Inc., 8 May. 2024, https://www.aatbio.com/data-sets/t-cell-protein-tyrosine-phosphatase-inhibitors-ic50-ki.

APA

AAT Bioquest, Inc. (2024, May 8). Quest Database™ T-cell protein-tyrosine phosphatase Inhibitors (IC50, Ki). AAT Bioquest. https://www.aatbio.com/data-sets/t-cell-protein-tyrosine-phosphatase-inhibitors-ic50-ki.
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