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TAK1/TAB1 Inhibitors (IC50, Ki)

Structure
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Compound Name
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Standard Type
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Standard Values (in nM)
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DoramapimodIC50900.0 [1]
5Z-7-OxozeaenolIC508.0 [1]
3-[2-(4-Oxo-1,3-thiazol-2-yl)hydrazinyl]indol-2-oneIC505000.0 [1]
7-Chloro-3-oxo-8-(1,3-thiazol-5-ylmethylamino)-11,16-dioxa-2,4,19,21-tetrazatricyclo[15.3.1.05,10]henicosa-1(20),5,7,9,17(21),18-hexaene-18-carbonitrileKi1606.0 [1]
(3Z)-3-(2-Oxo-2-phenylethylidene)-1,3-dihydro-2H-indol-2-oneIC505000.0 [1]
1-[4-[4-[7-Amino-2-(1,2-benzothiazol-7-yl)furo[2,3-c]pyridin-4-yl]pyrazol-1-yl]piperidin-1-yl]ethanoneIC5023.0 [1]
1-[5-Tert-butyl-3-[4-[2-(dimethylamino)ethyl]-5-oxo-1,4-diazepane-1-carbonyl]thiophen-2-yl]-3-(2,3-dichlorophenyl)ureaIC5030000.0 [1]
1-[4-[4-(7-Amino-2-thieno[2,3-c]pyridin-3-ylfuro[2,3-c]pyridin-4-yl)pyrazol-1-yl]piperidin-1-yl]ethanoneIC5030.0 [1]
(2Z)-3-(4-Hydroxyphenyl)-2-[(Z)-(2-oxo-1H-indol-3-ylidene)hydrazinylidene]-1,3-thiazolidin-4-oneIC5046.0 [1]
(2Z)-2-[(Z)-(2-Oxo-1H-indol-3-ylidene)hydrazinylidene]-3-(pyridin-4-ylmethyl)-1,3-thiazolidin-4-oneIC508200.0 [1]
(2Z)-3-(2-Hydroxyphenyl)-2-[(Z)-(2-oxo-1H-indol-3-ylidene)hydrazinylidene]-1,3-thiazolidin-4-oneIC505800.0 [1]
(2Z)-3-(4-Methoxyphenyl)-2-[(Z)-(2-oxo-1H-indol-3-ylidene)hydrazinylidene]-1,3-thiazolidin-4-oneIC505000.0 [1]
(2Z)-2-[(Z)-(5-Fluoro-2-oxo-1H-indol-3-ylidene)hydrazinylidene]-3-(4-hydroxyphenyl)-1,3-thiazolidin-4-oneIC5099.0 [1]
(2Z)-2-[(Z)-(2-Oxo-1H-indol-3-ylidene)hydrazinylidene]-3-(pyrrolidin-2-ylmethyl)-1,3-thiazolidin-4-oneIC5030000.0 [1]
(2Z)-2-[(Z)-(5-Chloro-2-oxo-1H-indol-3-ylidene)hydrazinylidene]-5-ethyl-3-(4-hydroxyphenyl)-1,3-thiazolidin-4-oneIC505000.0 [1]
(2Z)-2-[(Z)-(5-Chloro-2-oxo-1H-indol-3-ylidene)hydrazinylidene]-3-(4-hydroxyphenyl)-1,3-thiazolidin-4-oneIC5021.0 [1]
(2Z)-3-(3-Hydroxyphenyl)-2-[(Z)-(2-oxo-1H-indol-3-ylidene)hydrazinylidene]-1,3-thiazolidin-4-oneIC5025000.0 [1]
(2Z)-2-[(Z)-(5-Chloro-2-oxo-1H-indol-3-ylidene)hydrazinylidene]-3-(4-hydroxyphenyl)-5-methyl-1,3-thiazolidin-4-oneIC50630.0 [1]
(2Z)-2-[(Z)-(2-Oxo-1H-indol-3-ylidene)hydrazinylidene]-3-(4-oxo-1H-pyridin-3-yl)-1,3-thiazolidin-4-oneIC5025000.0 [1]
(2Z)-2-[(Z)-(5-Chloro-2-oxo-1H-indol-3-ylidene)hydrazinylidene]-3-(4-hydroxyphenyl)-5-propan-2-yl-1,3-thiazolidin-4-oneIC505000.0 [1]
(2Z)-3-(4-Hydroxyphenyl)-2-[(Z)-(5-methyl-2-oxo-1H-indol-3-ylidene)hydrazinylidene]-1,3-thiazolidin-4-oneIC5042.0 [1]
(2Z)-2-[(Z)-(5-Bromo-2-oxo-1H-indol-3-ylidene)hydrazinylidene]-3-(4-hydroxyphenyl)-1,3-thiazolidin-4-oneIC508.9 [1]
(2Z)-3-(4-Hydroxyphenyl)-2-[(Z)-[2-oxo-5-(trifluoromethoxy)-1H-indol-3-ylidene]hydrazinylidene]-1,3-thiazolidin-4-oneIC503000.0 [1]
(2Z)-3-[4-(Dimethylamino)phenyl]-2-[(Z)-(2-oxo-1H-indol-3-ylidene)hydrazinylidene]-1,3-thiazolidin-4-oneIC5050000.0 [1]
1-[4-[4-[7-Amino-2-(4-hydroxyphenyl)furo[2,3-c]pyridin-4-yl]pyrazol-1-yl]piperidin-1-yl]ethanoneIC50270.0 [1]
1-[4-[4-[7-Amino-2-(1H-pyrazol-4-yl)furo[2,3-c]pyridin-4-yl]pyrazol-1-yl]piperidin-1-yl]ethanoneIC50130.0 [1]
1-[4-[4-[7-Amino-2-(3-methylsulfonylphenyl)furo[2,3-c]pyridin-4-yl]pyrazol-1-yl]piperidin-1-yl]ethanoneIC504900.0 [1]
3-[4-[1-(1-Acetylpiperidin-4-yl)pyrazol-4-yl]-7-aminofuro[2,3-c]pyridin-2-yl]benzenesulfonamideIC501800.0 [1]
1-[4-[4-[7-Amino-2-(3-nitrophenyl)furo[2,3-c]pyridin-4-yl]pyrazol-1-yl]piperidin-1-yl]ethanoneIC5089.0 [1]
1-[4-[4-[7-Amino-2-(4-methylsulfanylphenyl)furo[2,3-c]pyridin-4-yl]pyrazol-1-yl]piperidin-1-yl]ethanoneIC5017500.0 [1]
N-[4-[4-[1-(1-Acetylpiperidin-4-yl)pyrazol-4-yl]-7-aminofuro[2,3-c]pyridin-2-yl]phenyl]methanesulfonamideIC504900.0 [1]
3-[4-[1-(1-Acetylpiperidin-4-yl)pyrazol-4-yl]-7-aminofuro[2,3-c]pyridin-2-yl]benzamideIC50530.0 [1]
1-[4-[4-[7-Amino-2-(cyclohexen-1-yl)furo[2,3-c]pyridin-4-yl]pyrazol-1-yl]piperidin-1-yl]ethanoneIC50460.0 [1]
1-[4-[4-(7-Amino-2-cyclohexylfuro[2,3-c]pyridin-4-yl)pyrazol-1-yl]piperidin-1-yl]ethanoneIC50650.0 [1]
1-[4-[4-[7-Amino-2-[3-(trifluoromethoxy)phenyl]furo[2,3-c]pyridin-4-yl]pyrazol-1-yl]piperidin-1-yl]ethanoneIC503500.0 [1]
1-[4-[4-[7-Amino-2-[4-(trifluoromethoxy)phenyl]furo[2,3-c]pyridin-4-yl]pyrazol-1-yl]piperidin-1-yl]ethanoneIC503500.0 [1]
1-[4-[4-[7-Amino-2-[3-(aminomethyl)phenyl]furo[2,3-c]pyridin-4-yl]pyrazol-1-yl]piperidin-1-yl]ethanoneIC50790.0 [1]
1-[4-[4-[7-Amino-2-[3-(2-methoxyethoxy)phenyl]furo[2,3-c]pyridin-4-yl]pyrazol-1-yl]piperidin-1-yl]ethanoneIC503200.0 [1]
1-[4-[4-[7-Amino-2-(1,2,3-benzothiadiazol-7-yl)furo[2,3-c]pyridin-4-yl]pyrazol-1-yl]piperidin-1-yl]ethanoneIC504.0 [1]
1-[4-[4-[7-Amino-2-(1,3-benzothiazol-7-yl)furo[2,3-c]pyridin-4-yl]pyrazol-1-yl]piperidin-1-yl]ethanoneIC5013.0 [1]
2-Phenyl-4-(1-piperidin-4-ylpyrazol-4-yl)furo[2,3-c]pyridin-7-amineIC502700.0 [1]
2-(1-Benzothiophen-7-Yl)-4-[1-(Piperidin-4-Yl)-1h-Pyrazol-4-Yl]furo[2,3-C]pyridin-7-AmineIC501200.0 [1]
1-[4-[4-(7-Amino-2-imidazo[1,2-a]pyrazin-3-ylfuro[2,3-c]pyridin-4-yl)pyrazol-1-yl]piperidin-1-yl]ethanoneIC501400.0 [1]
(3E)-3-[(2,3,4-Trihydroxyphenyl)methylidene]-1H-indol-2-oneIC501700.0 [1]
(3Z)-3-[2-(3,4-Dihydroxyphenyl)-2-oxoethylidene]-1H-indol-2-oneIC50560.0 [1]
(3Z)-3-[2-(3-Hydroxyphenyl)-2-oxoethylidene]-1H-indol-2-oneIC504100.0 [1]
(3E)-3-[(3,4-Dihydroxyphenyl)methylidene]-1H-indol-2-oneIC505000.0 [1]
1-[4-[4-[7-Amino-2-[2-(hydroxymethyl)phenyl]furo[2,3-c]pyridin-4-yl]pyrazol-1-yl]piperidin-1-yl]ethanoneIC50750.0 [1]
2-Thieno[2,3-c]pyridin-3-yl-4-(1,3,5-trimethylpyrazol-4-yl)furo[2,3-c]pyridin-7-amineIC5023900.0 [1]
2-[4-[1-(1-Acetylpiperidin-4-yl)pyrazol-4-yl]-7-aminofuro[2,3-c]pyridin-2-yl]benzamideIC506000.0 [1]
1-[4-[4-(7-Amino-2-phenylfuro[2,3-c]pyridin-4-yl)pyrazol-1-yl]piperidin-1-yl]ethanoneIC501100.0 [1]
1-[4-[4-[7-Amino-2-(3-hydroxyphenyl)furo[2,3-c]pyridin-4-yl]pyrazol-1-yl]piperidin-1-yl]ethanoneIC5061.0 [1]
1-[2-[4-[1-(1-Acetylpiperidin-4-yl)pyrazol-4-yl]-7-aminofuro[2,3-c]pyridin-2-yl]phenyl]ethanoneIC505400.0 [1]
4-(3-Methoxy-1-methylpyrazol-4-yl)-2-thieno[2,3-c]pyridin-3-ylfuro[2,3-c]pyridin-7-amineIC50600.0 [1]
3-[4-[1-(1-Acetylpiperidin-4-yl)pyrazol-4-yl]-7-aminofuro[2,3-c]pyridin-2-yl]benzonitrileIC50250.0 [1]
4-[4-[1-(1-Acetylpiperidin-4-yl)pyrazol-4-yl]-7-aminofuro[2,3-c]pyridin-2-yl]-N,N-dimethylbenzamideIC5030000.0 [1]
N-[3-[4-[1-(1-Acetylpiperidin-4-yl)pyrazol-4-yl]-7-aminofuro[2,3-c]pyridin-2-yl]phenyl]acetamideIC503200.0 [1]
1-[4-[4-[7-Amino-2-(3-methylsulfanylphenyl)furo[2,3-c]pyridin-4-yl]pyrazol-1-yl]piperidin-1-yl]ethanoneIC504300.0 [1]
1-[4-[4-[7-Amino-2-[2-(trifluoromethyl)phenyl]furo[2,3-c]pyridin-4-yl]pyrazol-1-yl]piperidin-1-yl]ethanoneIC5030000.0 [1]
1-[4-[4-[7-Amino-2-[3-(hydroxymethyl)phenyl]furo[2,3-c]pyridin-4-yl]pyrazol-1-yl]piperidin-1-yl]ethanoneIC50850.0 [1]
1-[4-[4-[7-Amino-2-(1-benzothiophen-3-yl)furo[2,3-c]pyridin-4-yl]pyrazol-1-yl]piperidin-1-yl]ethanoneIC50340.0 [1]
4-(1-Methylpyrrol-3-yl)-2-thieno[2,3-c]pyridin-3-ylfuro[2,3-c]pyridin-7-amineIC504900.0 [1]
2-[4-[4-[1-(1-Acetylpiperidin-4-yl)pyrazol-4-yl]-7-aminofuro[2,3-c]pyridin-2-yl]phenyl]acetonitrileIC501500.0 [1]
1-[4-[4-[7-Amino-2-(1-methylpyrrolo[2,3-c]pyridin-3-yl)furo[2,3-c]pyridin-4-yl]pyrazol-1-yl]piperidin-1-yl]ethanoneIC5018.0 [1]
4-(1-Methylimidazol-4-yl)-2-thieno[2,3-c]pyridin-3-ylfuro[2,3-c]pyridin-7-amineIC5012700.0 [1]
4-(1,3-Thiazol-4-yl)-2-thieno[2,3-c]pyridin-3-ylfuro[2,3-c]pyridin-7-amineIC501400.0 [1]
N-[2-[4-[1-(1-Acetylpiperidin-4-yl)pyrazol-4-yl]-7-aminofuro[2,3-c]pyridin-2-yl]phenyl]acetamideIC5030000.0 [1]
1-[4-[4-[7-Amino-2-[2-(methoxymethyl)phenyl]furo[2,3-c]pyridin-4-yl]pyrazol-1-yl]piperidin-1-yl]ethanoneIC501400.0 [1]
1-{4-[4-(7-Amino-2-cyclopentylfuro[2,3-c]pyridin-4-yl)-1H-pyrazol-1-yl]piperidin-1-yl}ethanoneIC502100.0 [1]
2-[4-[1-(1-Acetylpiperidin-4-yl)pyrazol-4-yl]-7-aminofuro[2,3-c]pyridin-2-yl]benzonitrileIC50560.0 [1]
1-[4-[4-[7-Amino-2-(3-aminophenyl)furo[2,3-c]pyridin-4-yl]pyrazol-1-yl]piperidin-1-yl]ethanoneIC50770.0 [1]
1-[4-[4-(7-Amino-2-naphthalen-1-ylfuro[2,3-c]pyridin-4-yl)pyrazol-1-yl]piperidin-1-yl]ethanoneIC501000.0 [1]
2-Thieno[2,3-c]pyridin-3-yl-4-thiophen-3-ylfuro[2,3-c]pyridin-7-amineIC502200.0 [1]
Tak1 inhibitorIC5028.0 [1]
1-[4-[4-[7-Amino-2-(4-aminophenyl)furo[2,3-c]pyridin-4-yl]pyrazol-1-yl]piperidin-1-yl]ethanoneIC501800.0 [1]
3-[4-[1-(1-Acetylpiperidin-4-yl)pyrazol-4-yl]-7-aminofuro[2,3-c]pyridin-2-yl]-N,N-dimethylbenzenesulfonamideIC501400.0 [1]
1-{4-[4-(7-Amino-2-cyclopent-1-enyl-furo[2,3-c]pyridin-4-yl)-pyrazol-1-yl]-piperidin-1-yl}-ethanoneIC501200.0 [1]
1-[4-[4-[7-Amino-2-(2-methylsulfanylphenyl)furo[2,3-c]pyridin-4-yl]pyrazol-1-yl]piperidin-1-yl]ethanoneIC50430.0 [1]
1-[3-[4-[1-(1-Acetylpiperidin-4-yl)pyrazol-4-yl]-7-aminofuro[2,3-c]pyridin-2-yl]phenyl]ethanoneIC502800.0 [1]
1-[4-[4-[7-Amino-2-(4-methylsulfonylphenyl)furo[2,3-c]pyridin-4-yl]pyrazol-1-yl]piperidin-1-yl]ethanoneIC5025700.0 [1]
1-[4-[4-(7-Amino-2-thiophen-3-ylfuro[2,3-c]pyridin-4-yl)pyrazol-1-yl]piperidin-1-yl]ethanoneIC50480.0 [1]
1-[4-[4-[7-Amino-2-[3-(trifluoromethyl)phenyl]furo[2,3-c]pyridin-4-yl]pyrazol-1-yl]piperidin-1-yl]ethanoneIC502800.0 [1]
4-(2-Methyl-1,3-thiazol-5-yl)-2-thieno[2,3-c]pyridin-3-ylfuro[2,3-c]pyridin-7-amineIC50230.0 [1]
1-[4-[4-[7-Amino-2-[4-(hydroxymethyl)phenyl]furo[2,3-c]pyridin-4-yl]pyrazol-1-yl]piperidin-1-yl]ethanoneIC502800.0 [1]
2-[2-[4-[1-(1-Acetylpiperidin-4-yl)pyrazol-4-yl]-7-aminofuro[2,3-c]pyridin-2-yl]phenyl]acetonitrileIC50250.0 [1]
4-(Furan-3-yl)-2-thieno[2,3-c]pyridin-3-ylfuro[2,3-c]pyridin-7-amineIC50560.0 [1]
4-[4-[7-Amino-2-(1,2,3-benzothiadiazol-7-yl)furo[2,3-c]pyridin-4-yl]pyrazol-1-yl]cyclohexan-1-olIC509.0 [1]
4-(7-Amino-2-thieno[2,3-c]pyridin-3-ylfuro[2,3-c]pyridin-4-yl)-1-methylpyrazole-3-carbonitrileIC5022800.0 [1]
4-[4-[1-(1-Acetylpiperidin-4-yl)pyrazol-4-yl]-7-aminofuro[2,3-c]pyridin-2-yl]benzonitrileIC502500.0 [1]
4-(1,5-Dimethylpyrazol-4-yl)-2-thieno[2,3-c]pyridin-3-ylfuro[2,3-c]pyridin-7-amineIC504100.0 [1]
4-(5-Methylthiophen-2-yl)-2-thieno[2,3-c]pyridin-3-ylfuro[2,3-c]pyridin-7-amineIC504600.0 [1]
4-(1-Methylpyrazol-4-yl)-2-thieno[2,3-c]pyridin-3-ylfuro[2,3-c]pyridin-7-amineIC50150.0 [1]
4-(1,3-Dimethylpyrazol-4-yl)-2-thieno[2,3-c]pyridin-3-ylfuro[2,3-c]pyridin-7-amineIC503500.0 [1]
1-[4-[4-[7-Amino-2-(1,2,3,6-tetrahydropyridin-4-yl)furo[2,3-c]pyridin-4-yl]pyrazol-1-yl]piperidin-1-yl]ethanoneIC50800.0 [1]
1-[4-[4-[7-Amino-2-[3-(dimethylamino)phenyl]furo[2,3-c]pyridin-4-yl]pyrazol-1-yl]piperidin-1-yl]ethanoneIC502400.0 [1]
1-[4-[4-[7-Amino-2-(3-methoxyphenyl)furo[2,3-c]pyridin-4-yl]pyrazol-1-yl]piperidin-1-yl]ethanoneIC501800.0 [1]
4-(5-Methylfuran-2-yl)-2-thieno[2,3-c]pyridin-3-ylfuro[2,3-c]pyridin-7-amineIC502100.0 [1]
1-[4-[4-(7-Amino-2-pyridin-3-ylfuro[2,3-c]pyridin-4-yl)pyrazol-1-yl]piperidin-1-yl]ethanoneIC50710.0 [1]
1-[4-[4-[7-Amino-2-(1-methylpyrazol-4-yl)furo[2,3-c]pyridin-4-yl]pyrazol-1-yl]piperidin-1-yl]ethanoneIC501600.0 [1]
1-[4-[4-[7-Amino-2-(1,3-oxazol-5-yl)furo[2,3-c]pyridin-4-yl]pyrazol-1-yl]piperidin-1-yl]ethanoneIC501200.0 [1]
Items per page: 1 - 10 of 100
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References

This online tool may be cited as follows

MLA

"Quest Database™ TAK1/TAB1 Inhibitors (IC50, Ki)." AAT Bioquest, Inc., 9 May. 2024, https://www.aatbio.com/data-sets/tak1-tab1-inhibitors-ic50-ki.

APA

AAT Bioquest, Inc. (2024, May 9). Quest Database™ TAK1/TAB1 Inhibitors (IC50, Ki). AAT Bioquest. https://www.aatbio.com/data-sets/tak1-tab1-inhibitors-ic50-ki.
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