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Thromboxane A2 receptor Inhibitors (IC50, Ki)

Structure
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Compound Name
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Standard Type
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Standard Values (in nM)
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▼
Benzenesulfonamide, N-(((1,1-dimethylethyl)amino)carbonyl)-2-((4-methylphenyl)amino)-5-nitro-IC5053.0 [1], 240.0 [2], 319.0 [3], 620.0 [4], 700.0 [5]
RamatrobanIC508.4 [1], 9.6 [2], 14.0 [3]
RamatrobanKi0.58 [1], 4.5 [2], 18.0 [3]
RidogrelIC501280.0 [1], 1700.0 [2], 2100.0 [3], 5200.0 [4]
1-[(3,4,5-Trimethoxyphenyl)methyl]-1,2,3,4-tetrahydroisoquinoline-6,7-diolIC50281.84 [1], 446.68 [2]
1-[(3,4,5-Trimethoxyphenyl)methyl]-1,2,3,4-tetrahydroisoquinoline-6,7-diolKi162.18 [1], 173.78 [2]
2-[(3R)-5-Acetyl-4-[(4-chlorophenyl)methyl]-7-methylsulfonyl-2,3-dihydro-1H-cyclopenta[b]indol-3-yl]acetic acidIC508400.0 [1]
2-[(3R)-5-Acetyl-4-[(4-chlorophenyl)methyl]-7-methylsulfonyl-2,3-dihydro-1H-cyclopenta[b]indol-3-yl]acetic acidKi1200.0 [1]
2-[(3R)-4-[(4-Chlorophenyl)methyl]-5-(1-hydroxyethyl)-7-methylsulfonyl-2,3-dihydro-1H-cyclopenta[b]indol-3-yl]acetic acidIC5043000.0 [1]
2-[(3R)-4-[(4-Chlorophenyl)methyl]-5-(1-hydroxyethyl)-7-methylsulfonyl-2,3-dihydro-1H-cyclopenta[b]indol-3-yl]acetic acidKi7100.0 [1]
2-[(3R)-3-[(4-Fluorophenyl)sulfonyl-methylamino]-1,2,3,4-tetrahydrocarbazol-9-yl]acetic acidIC5010000.0 [1]
2-[(3R)-3-[(4-Fluorophenyl)sulfonyl-methylamino]-1,2,3,4-tetrahydrocarbazol-9-yl]acetic acidKi6852.0 [1], 10000.0 [2]
SulotrobanKi650.0 [1], 1300.0 [2]
DaltrobanIC50150.0 [1], 460.0 [2]
DaltrobanKi63.0 [1]
MK-7246IC50100000.0 [1]
MK-7246Ki3804.0 [1]
(R,S)-8-((4-Chlorophenylsulfonyl)amino)-4-(3-(3-pyridinyl)propyl)octanoic acidIC506.0 [1], 18.0 [2]
Acetic acid, (3-(((1S)-2-(4,5-diphenyl-2-oxazolyl)-2-cyclohexen-1-yl)methyl)phenoxy)-, sodium saltKi1000.0 [1]
3-[3-[2-[(4-Chlorophenyl)sulfonylamino]ethyl]phenyl]propanoic acidIC5061.0 [1], 190.0 [2], 523.0 [3]
SamixogrelIC5019.0 [1]
Benzenesulfonamide, 2-((4-methylphenyl)amino)-5-nitro-N-((pentylamino)carbonyl)-IC5013.56 [1], 50.04 [2], 278.0 [3]
11-[2-(Benzenesulfonamido)ethylsulfanyl]-6,11-dihydrobenzo[c][1]benzoxepine-2-carboxylic acidKi32.0 [1]
11-[2-[[(E)-2-Phenylethenyl]sulfonylamino]ethylsulfanyl]-6,11-dihydrobenzo[c][1]benzoxepine-2-carboxylic acidKi4.2 [1], 6.5 [2]
1-[2-(4-Methylphenoxy)-5-nitrophenyl]sulfonyl-3-pentylureaIC5055.38 [1], 139.32 [2], 670.0 [3]
1-Tert-butyl-3-[2-(4-methylphenoxy)-5-nitrophenyl]sulfonylureaIC5057.63 [1], 58.34 [2], 300.0 [3]
1-Tert-butyl-3-[2-(4-methylphenyl)sulfanyl-5-nitrophenyl]sulfonylureaIC5055.17 [1], 293.54 [2], 800.0 [3]
N-[2-(4-Methylphenylamino)-5-nitrobenzenesulfonyl]-piperidine-1-carboxamideIC5038.52 [1], 64.81 [2], 900.0 [3]
1-Tert-butyl-3-[2-(2,6-dimethylanilino)-5-nitrophenyl]sulfonylureaIC5030.78 [1], 56.89 [2], 90.0 [3]
DinoprostIC500.0 [1], 10000.0 [2]
CAY10471 RacemateKi1394.0 [1], 10000.0 [2]
2-[2-Methyl-1-[4-[[(2S)-4-methyl-2,3-dihydro-1,4-benzoxazin-2-yl]methoxy]benzoyl]indol-4-yl]acetic acidKi260.0 [1]
2-[(11E)-11-[2-(Dimethylamino)ethylidene]-6H-benzo[c][1]benzoxepin-2-yl]acetic acidKi1000.0 [1]
2-Pyridinecarboxylic acid, 6-(5'-chloro-2'-(2-methylpropoxy)(1,1'-biphenyl)-2-yl)-, sodium saltIC501584.89 [1]
2-Pyridinecarboxylic acid, 6-(5'-chloro-2'-(2-methylpropoxy)(1,1'-biphenyl)-2-yl)-, sodium saltKi316.23 [1]
11-[2-(Pyridin-3-ylsulfonylamino)ethylsulfanyl]-6,11-dihydrobenzo[c][1]benzoxepine-2-carboxylic acidKi47.0 [1]
(Z)-6-[3-[(N'-Tert-butyl-N-cyanocarbamimidoyl)amino]phenyl]-6-pyridin-3-ylhex-5-enoic acidIC5011.0 [1], 2600.0 [2]
1-(4-Aminobenzyl)-1,2,3,4-tetrahydroisoquinoline-6,7-diolIC5089125.09 [1]
1-(4-Aminobenzyl)-1,2,3,4-tetrahydroisoquinoline-6,7-diolKi34673.69 [1]
1-(5-Nitro-2-(m-tolyloxy)phenylsulfonyl)-3-pentylureaIC50223.0 [1], 2530.0 [2]
1-(5-Nitro-2-(o-tolyloxy)phenylsulfonyl)-3-pentylureaIC50181.0 [1], 1630.0 [2]
2-(2-Benzoyl-3,4-dihydro-1H-pyrido[4,3-b]indol-5-yl)acetic acidIC5025000.0 [1]
7-[3,5-Dihydroxy-2-(3-hydroxy-5-phenyl-pentyl)-cyclopentyl]-heptanoic acidIC5010000.0 [1]
2-[(7R)-7-[(4-Fluorophenyl)sulfonyl-methylamino]-6,7,8,9-tetrahydropyrido[2,3-b]indolizin-10-yl]acetic acidIC50100000.0 [1]
2-[(7R)-7-[(4-Fluorophenyl)sulfonyl-methylamino]-6,7,8,9-tetrahydropyrido[2,3-b]indolizin-10-yl]acetic acidKi7000.0 [1]
3-(2-(Naphthalen-2-ylmethyl)phenyl)acrylic acidKi500.0 [1], 10000.0 [2]
2-[2-(Benzenesulfonamido)ethylsulfanyl]tricyclo[9.4.0.03,8]pentadeca-1(15),3(8),4,6,11,13-hexaene-5-carboxylic acidKi30.0 [1]
11-[2-[(3-Nitrophenyl)sulfonylamino]ethylsulfanyl]-6,11-dihydrobenzo[c][1]benzoxepine-2-carboxylic acidKi14.0 [1]
11-[2-[(3,4,5-Trimethoxybenzoyl)amino]ethylsulfanyl]-6,11-dihydrobenzo[c][1]benzoxepine-2-carboxylic acidKi92.0 [1]
11-((2-((Phenylsulfonyl)amino)ethyl)thio)-6,11-dihydrodibenzo(b,e)thiepin-2-carboxylic acidKi3.7 [1]
11-[2-[(2-Nitrophenyl)sulfonylamino]ethylsulfanyl]-6,11-dihydrobenzo[c][1]benzoxepine-2-carboxylic acidKi15.0 [1]
11-[2-[(3-Methylthiophene-2-carbonyl)amino]ethylsulfanyl]-6,11-dihydrobenzo[c][1]benzoxepine-2-carboxylic acidKi10.0 [1]
11-[2-[(2,3,4-Trimethoxybenzoyl)amino]ethylsulfanyl]-6,11-dihydrobenzo[c][1]benzoxepine-2-carboxylic acidKi18.0 [1]
11-[2-(Benzylcarbamothioylamino)ethylsulfanyl]-6,11-dihydrobenzo[c][1]benzoxepine-2-carboxylic acidKi6.1 [1]
11-[2-[(4-Methylphenyl)sulfonylamino]ethylsulfanyl]-6,11-dihydrobenzo[c][1]benzoxepine-2-carboxylic acidKi27.0 [1]
11-(2-Benzamidoethylsulfanyl)-6,11-dihydrobenzo[c][1]benzoxepine-2-carboxylic acidKi44.0 [1]
11-[2-(Phenylmethoxycarbonylamino)ethylsulfanyl]-6,11-dihydrobenzo[c][1]benzoxepine-2-carboxylic acidKi7.7 [1]
11-[2-[Benzenesulfonyl(methyl)amino]ethylsulfanyl]-6,11-dihydrobenzo[c][1]benzoxepine-2-carboxylic acidKi33.0 [1]
3-[alpha-[[2-[(Phenylsulfonyl)amino]ethyl]thio]benzyl]benzoic acidKi77.0 [1]
11-[2-[(4-Methoxyphenyl)sulfonylamino]ethylsulfanyl]-6,11-dihydrobenzo[c][1]benzoxepine-2-carboxylic acidKi17.0 [1]
2-[2-(Benzenesulfonamido)ethylsulfanyl]tricyclo[9.4.0.03,8]pentadeca-1(15),3(8),4,6,9,11,13-heptaene-5-carboxylic acidKi25.0 [1]
1-(3-Nitro-4-hydroxybenzyl)-1,2,3,4-tetrahydroisoquinoline-6,7-diolIC50870.96 [1]
1-(3-Nitro-4-hydroxybenzyl)-1,2,3,4-tetrahydroisoquinoline-6,7-diolKi338.84 [1]
1-(4-Nitrobenzyl)-1,2,3,4-tetrahydroisoquinoline-6,7-diolIC5025118.86 [1]
1-(4-Nitrobenzyl)-1,2,3,4-tetrahydroisoquinoline-6,7-diolKi9549.93 [1]
2-(2-Phenylethyl)-1-[(3,4,5-trimethoxyphenyl)methyl]-3,4-dihydro-1H-isoquinoline-6,7-diolIC5041686.94 [1]
2-(2-Phenylethyl)-1-[(3,4,5-trimethoxyphenyl)methyl]-3,4-dihydro-1H-isoquinoline-6,7-diolKi16218.1 [1]
2-[(3R)-5-Acetyl-4-[(4-chlorophenyl)methyl]-7-fluoro-2,3-dihydro-1H-cyclopenta[b]indol-3-yl]acetic acidIC501400.0 [1]
2-[(3R)-5-Acetyl-4-[(4-chlorophenyl)methyl]-7-fluoro-2,3-dihydro-1H-cyclopenta[b]indol-3-yl]acetic acidKi14.0 [1]
2-[(1R)-6-Fluoro-8-methylsulfonyl-9-[(1S)-1-[4-(trifluoromethyl)phenyl]ethyl]-1,2,3,4-tetrahydrocarbazol-1-yl]acetic acidIC5019400.0 [1]
2-[(1R)-6-Fluoro-8-methylsulfonyl-9-[(1S)-1-[4-(trifluoromethyl)phenyl]ethyl]-1,2,3,4-tetrahydrocarbazol-1-yl]acetic acidKi338.0 [1]
1-[2-(3-Methylanilino)-5-nitrophenyl]sulfonyl-3-pentylureaIC5045.53 [1], 60.39 [2]
1-Butyl-3-[2-(4-methylphenoxy)-5-nitrophenyl]sulfonylureaIC5052.89 [1], 558.04 [2]
[3-((R)-4-Fluoro-benzenesulfonylamino)-1,2,3,4-tetrahydro-carbazol-9-yl]-acetic acidIC501700.0 [1]
[3-((R)-4-Fluoro-benzenesulfonylamino)-1,2,3,4-tetrahydro-carbazol-9-yl]-acetic acidKi540.0 [1]
1-[2-(2,6-Dimethylanilino)-5-nitrophenyl]sulfonyl-3-pentylureaIC5047.1 [1], 80.72 [2]
1-Benzyl-3-[2-(4-methylanilino)-5-nitrophenyl]sulfonylureaIC5045.01 [1], 64.47 [2]
[(3R)-5-Bromo-4-(4-chlorobenzyl)-7-fluoro-1,2,3,4-tetrahydrocyclopenta[b]indol-3-yl]acetic acidIC5080.0 [1]
[(3R)-5-Bromo-4-(4-chlorobenzyl)-7-fluoro-1,2,3,4-tetrahydrocyclopenta[b]indol-3-yl]acetic acidKi0.84 [1]
1-[2-(Cyclohexylamino)-5-nitrophenyl]sulfonyl-3-hexylureaIC5046.17 [1], 81.22 [2]
1-[2-(4-Bromo-3-methylanilino)-5-nitrophenyl]sulfonyl-3-pentylureaIC5043.19 [1], 126.28 [2]
1-[2-(3,5-Dimethylanilino)-5-nitrophenyl]sulfonyl-3-pentylureaIC5076.5 [1], 537.86 [2]
1-Cyclohexyl-3-[2-(4-methylphenoxy)-5-nitrophenyl]sulfonylureaIC5070.15 [1], 600.71 [2]
1-[2-(Cyclohexylamino)-5-nitrophenyl]sulfonyl-3-heptylureaIC5055.55 [1], 92.9 [2]
1-Hexyl-3-[2-(4-methylphenoxy)-5-nitrophenyl]sulfonylureaIC5058.48 [1], 526.42 [2]
11-[2-(Naphthalen-2-ylsulfonylamino)ethylsulfanyl]-6,11-dihydrobenzo[c][1]benzoxepine-2-carboxylic acidKi14.0 [1]
11-[2-[[4-(Trifluoromethyl)phenyl]sulfonylamino]ethylsulfanyl]-6,11-dihydrobenzo[c][1]benzoxepine-2-carboxylic acidKi20.0 [1]
(Z)-7-[(1R,2S,3R)-3-(Hexylsulfanylmethyl)-7-oxabicyclo[2.2.1]heptan-2-yl]hept-5-enoic acidIC5083000.0 [1], 1000000.0 [2]
1-(3,4,5-Trimethoxyanilino)-3,4-dihydroisoquinoline-6,7-diolIC50275422.87 [1]
1-(3,4,5-Trimethoxyanilino)-3,4-dihydroisoquinoline-6,7-diolKi120226.44 [1]
1-Tert-butyl-3-[2-(3-methoxyphenoxy)-5-nitrophenyl]sulfonylureaIC5099.0 [1], 1970.0 [2]
1-Tert-butyl-3-[2-(2-methoxy-4-methylphenoxy)-5-nitrophenyl]sulfonylureaIC5052.0 [1], 528.0 [2]
1-[2-(2-Methylphenoxy)-5-nitrophenyl]sulfonyl-3-propan-2-ylureaIC50501.0 [1], 8750.0 [2]
1-Tert-butyl-3-[2-(2-methylphenoxy)-5-nitrophenyl]sulfonylureaIC50233.0 [1], 3760.0 [2]
1-Butyl-3-[2-(3-methylphenoxy)-5-nitrophenyl]sulfonylureaIC50155.0 [1], 1910.0 [2]
1-[2-(4-Methylphenoxy)-5-nitrophenyl]sulfonyl-3-propan-2-ylureaIC50843.0 [1], 8760.0 [2]
1-[2-(2-Bromophenoxy)-5-nitrophenyl]sulfonyl-3-tert-butylureaIC50151.0 [1], 2580.0 [2]
1-[2-(2-Bromophenoxy)-5-nitrophenyl]sulfonyl-3-pentylureaIC50423.0 [1], 3130.0 [2]
1-[2-(3-Bromophenoxy)-5-nitrophenyl]sulfonyl-3-pentylureaIC50413.0 [1], 5860.0 [2]
1-[2-(4-Bromophenoxy)-5-nitrophenyl]sulfonyl-3-pentylureaIC50120.0 [1], 1010.0 [2]
Items per page: 1 - 10 of 100
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References

This online tool may be cited as follows

MLA

"Quest Database™ Thromboxane A2 receptor Inhibitors (IC50, Ki)." AAT Bioquest, Inc., 9 May. 2024, https://www.aatbio.com/data-sets/thromboxane-a2-receptor-inhibitors-ic50-ki.

APA

AAT Bioquest, Inc. (2024, May 9). Quest Database™ Thromboxane A2 receptor Inhibitors (IC50, Ki). AAT Bioquest. https://www.aatbio.com/data-sets/thromboxane-a2-receptor-inhibitors-ic50-ki.
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