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Thymidylate kinase Inhibitors (IC50, Ki)

Structure
▲
▼
Compound Name
▲
▼
Standard Type
▲
▼
Standard Values (in nM)
▲
▼
ThymidineKi180000.0 [1]
5-Bromo-2'-deoxyuridineKi214000.0 [1]
5,5'-Dithiobis(2-nitrobenzoic acid)IC501530.0 [1]
1-(4-Aminomethyl-5-hydroxymethyl-tetrahydro-furan-2-yl)-5-methyl-1H-pyrimidine-2,4-dioneKi220000.0 [1]
p1-(5'-Adenosyl)p5-(5'-thymidyl)pentaphosphateIC508000.0 [1]
1-[(4Ar,5S,7R,7aR)-5-(hydroxymethyl)-2-sulfanylidene-3,4,4a,5,7,7a-hexahydrofuro[3,4-e][1,3]oxazin-7-yl]-5-methylpyrimidine-2,4-dioneKi700000.0 [1]
P(1)-(Adenosine-5')-P(5)-(thymidine-5')-pentaphosphateIC50290000.0 [1]
1-[4-Chloro-3-(trifluoromethyl)phenyl]-3-[(2S,3S,5R)-2-(hydroxymethyl)-5-(5-methyl-2,4-dioxopyrimidin-1-yl)oxolan-3-yl]ureaKi95000.0 [1]
4-[4-[(5-Methyl-2,4-dioxo-pyrimidin-1-yl)methyl]phenyl]butanoic acidKi252000.0 [1]
4-[4-[(5-Bromo-2,4-dioxo-pyrimidin-1-yl)methyl]phenyl]butanoic acidKi293000.0 [1]
1-[(4Ar,5S,7R,7aR)-5-(hydroxymethyl)-2-oxo-3,4,4a,5,7,7a-hexahydrofuro[3,4-e][1,3]oxazin-7-yl]-5-methylpyrimidine-2,4-dioneKi1100000.0 [1]
1-Methyl-6-Phenyl-1,3-Dihydro-2h-Imidazo[4,5-B]pyridin-2-OneIC50200000.0 [1]
2-(3-Bromophenoxy)-4-[(1R)-3,3-dimethyl-1-[(3S)-3-(5-methyl-2,4-dioxopyrimidin-1-yl)piperidin-1-yl]butyl]benzoic acidIC5062000.0 [1]
2-(3-Chlorophenoxy)-4-[(1R)-1-[(3S)-3-(5-methyl-2,4-dioxopyrimidin-1-yl)piperidin-1-yl]butyl]benzoic acidIC50150000.0 [1]
4-[4-[(5-Chloro-2,4-dioxo-pyrimidin-1-yl)methyl]phenyl]butanoic AcidKi790000.0 [1]
6-[4-[(5-Bromo-2,4-dioxo-pyrimidin-1-yl)methyl]phenyl]hexanoic AcidKi92000.0 [1]
[(2S,3R,5R)-2-(Hydroxymethyl)-5-(5-methyl-2,4-dioxopyrimidin-1-yl)oxolan-3-yl]methylimino-iminoazaniumKi1040000.0 [1]
5-[4-[(5-Chloro-2,4-dioxo-pyrimidin-1-yl)methyl]phenyl]pentanoic acidKi122000.0 [1]
[[(2R,3S,4R)-5-(6-Aminopurin-9-yl)-3,4-dihydroxyoxolan-2-yl]methoxy-hydroxyphosphoryl] [hydroxy-[hydroxy-[hydroxy-[hydroxy-[[(2R,3S)-3-hydroxy-5-(5-methyl-2,4-dioxopyrimidin-1-yl)oxolan-2-yl]methoxy]phosphoryl]oxyphosphoryl]oxyphosphoryl]oxyphosphoryl] hydrogen phosphateIC506000.0 [1]
[[(2R,3S,4R)-5-(6-Aminopurin-9-yl)-3,4-dihydroxyoxolan-2-yl]methoxy-hydroxyphosphoryl] [hydroxy-[[(2R,3S)-3-hydroxy-5-(5-methyl-2,4-dioxopyrimidin-1-yl)oxolan-2-yl]methoxy]phosphoryl] hydrogen phosphateIC501230000.0 [1]
[[[[(2R,3S,4R)-5-(6-Aminopurin-9-yl)-3,4-dihydroxyoxolan-2-yl]methoxy-hydroxyphosphoryl]oxy-hydroxyphosphoryl]oxy-hydroxyphosphoryl]oxy-[[hydroxy-[[(2R,3S)-3-hydroxy-5-(5-methyl-2,4-dioxopyrimidin-1-yl)oxolan-2-yl]methoxy]phosphoryl]methyl]phosphinic acidIC506000.0 [1]
[[(2R,3S,4R)-5-(6-Aminopurin-9-yl)-3,4-dihydroxyoxolan-2-yl]methoxy-hydroxyphosphoryl]oxy-[[hydroxy-[[(2R,3S)-3-hydroxy-5-(5-methyl-2,4-dioxopyrimidin-1-yl)oxolan-2-yl]methoxy]phosphoryl]methyl]phosphinic acidIC50730000.0 [1]
Bis[[[[(2R,3S,4R)-5-(6-aminopurin-9-yl)-3,4-dihydroxyoxolan-2-yl]methoxy-dihydroxyphosphaniumyl]oxy-dihydroxyphosphaniumyl]oxy]-dihydroxyphosphaniumIC501000000.0 [1]
[[[[[(2R,3S,4R)-5-(6-Aminopurin-9-yl)-3,4-dihydroxyoxolan-2-yl]methoxy-hydroxyphosphoryl]oxy-hydroxyphosphoryl]oxy-hydroxyphosphoryl]oxy-hydroxyphosphoryl]oxy-[[hydroxy-[[(2R,3S)-3-hydroxy-5-(5-methyl-2,4-dioxopyrimidin-1-yl)oxolan-2-yl]methoxy]phosphoryl]methyl]phosphinic acidIC504000.0 [1]
[[[(2R,3S,4R)-5-(6-Aminopurin-9-yl)-3,4-dihydroxyoxolan-2-yl]methoxy-hydroxyphosphoryl]oxy-hydroxyphosphoryl]oxy-[[hydroxy-[[(2R,3S)-3-hydroxy-5-(5-methyl-2,4-dioxopyrimidin-1-yl)oxolan-2-yl]methoxy]phosphoryl]methyl]phosphinic acidIC50340000.0 [1]
3-(1-Methyl-2-Oxo-2,3-Dihydro-1h-Imidazo[4,5-B]pyridin-6-Yl)benzamideIC50200000.0 [1]
3-(1-Methyl-2-oxo-3H-imidazo[4,5-b]pyridin-6-yl)-N-(3-phenylpropyl)benzamideIC50200000.0 [1]
N-[3-(4-Fluorophenyl)propyl]-3-(1-methyl-2-oxo-3H-imidazo[4,5-b]pyridin-6-yl)benzamideIC50123000.0 [1]
3-(1-Methyl-2-oxo-3H-imidazo[4,5-b]pyridin-6-yl)-N-[3-[4-(trifluoromethyl)phenyl]propyl]benzamideIC50124000.0 [1]
4-[[(3S)-3-(5-Methyl-2,4-dioxopyrimidin-1-yl)piperidin-1-yl]methyl]-2-[3-(trifluoromethyl)phenoxy]benzoic acidIC50200000.0 [1]
1-[(3S)-1-[3-(3-Chlorophenoxy)-4-hydroxyphenyl]sulfonylpiperidin-3-yl]-5-methylpyrimidine-2,4-dioneIC50200000.0 [1]
2-(3-Chlorophenoxy)-4-[(1R)-1-[(3S)-3-(5-methyl-2,4-dioxopyrimidin-1-yl)piperidin-1-yl]ethyl]benzoic acidIC50150000.0 [1]
2-(3-Bromophenoxy)-4-[(1R)-1-[(3S)-3-(5-methyl-2,4-dioxopyrimidin-1-yl)piperidin-1-yl]hexyl]benzoic acidIC5032000.0 [1]
2-(3-Chlorophenoxy)-4-[(1R)-3,3-dimethyl-1-[(3S)-3-(5-methyl-2,4-dioxopyrimidin-1-yl)piperidin-1-yl]pentyl]benzoic acidIC5043400.0 [1]
Items per page: 1 - 10 of 34
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References

This online tool may be cited as follows

MLA

"Quest Database™ Thymidylate kinase Inhibitors (IC50, Ki)." AAT Bioquest, Inc., 8 May. 2024, https://www.aatbio.com/data-sets/thymidylate-kinase-inhibitors-ic50-ki.

APA

AAT Bioquest, Inc. (2024, May 8). Quest Database™ Thymidylate kinase Inhibitors (IC50, Ki). AAT Bioquest. https://www.aatbio.com/data-sets/thymidylate-kinase-inhibitors-ic50-ki.
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