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Thymidylate synthase Inhibitors (IC50, Ki)
Structure
Compound Name
Standard Type
Standard Values (in nM)
PemetrexedIC509500.0 [1]
PemetrexedKi1.3 [1], 340.0 [2]
RaltitrexedIC50380.0 [1]
10-Propargyl-5,8-dideazafolic acidIC5072.0 [1]
10-Propargyl-5,8-dideazafolic acidKi7.0 [1], 30.0 [2], 20000.0 [3]

References
This online resource may be cited as follows
MLA
"Quest DatabaseThymidylate synthase Inhibitors (IC50, Ki)." AAT Bioquest, Inc.5 Mar2026https://www.aatbio.com/data-sets/thymidylate-synthase-inhibitors-ic50-ki.
APA
AAT Bioquest, Inc. (2026March 5). Quest DatabaseThymidylate synthase Inhibitors (IC50, Ki). AAT Bioquest. https://www.aatbio.com/data-sets/thymidylate-synthase-inhibitors-ic50-ki.
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