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Thyroid hormone receptor beta-1 Inhibitors (IC50, Ki)
StructureCompound NameStandard TypeStandard Values (in nM)
LiothyronineIC500.26 [1], 2.9 [2]
LiothyronineKi0.08 [1], 0.55 [2], 0.68 [3], 2.29 [4]
{3,5-Dichloro-4-[4-Hydroxy-3-(Propan-2-Yl)phenoxy]phenyl}acetic AcidIC501.1 [1]
{3,5-Dichloro-4-[4-Hydroxy-3-(Propan-2-Yl)phenoxy]phenyl}acetic AcidKi0.24 [1], 0.37 [2]
2-Methyl-3-(3,5-diiodo-4-carboxymethoxybenzyl)benzofuranIC504100.0 [1], 5100.0 [2], 5128.61 [3]

References
This online resource may be cited as follows
MLA
"Quest DatabaseThyroid hormone receptor beta-1 Inhibitors (IC50, Ki)." AAT Bioquest, Inc.11 Oct2025https://www.aatbio.com/data-sets/thyroid-hormone-receptor-beta-1-inhibitors-ic50-ki.
APA
AAT Bioquest, Inc. (2025October 11). Quest DatabaseThyroid hormone receptor beta-1 Inhibitors (IC50, Ki). AAT Bioquest. https://www.aatbio.com/data-sets/thyroid-hormone-receptor-beta-1-inhibitors-ic50-ki.
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