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TNF-alpha Inhibitors (IC50, Ki)
Structure
Compound Name
Standard Type
Standard Values (in nM)
6,7-Dimethyl-3-[[methyl-[2-[methyl-[[1-[3-(trifluoromethyl)phenyl]indol-3-yl]methyl]amino]ethyl]amino]methyl]chromen-4-oneIC505000.0 [1], 15000.0 [2], 22000.0 [3]
RolipramIC50200.0 [1], 500.0 [2], 12000.0 [3]
MesalamineIC5020000.0 [1], 20600000.0 [2]
1-Propyl-2,4-dioxo-1,4-dihydropteridine-3(2H)-butyric acid ethyl esterIC503000.0 [1], 5000.0 [2]
4-N-Benzyl-4-N-[2-[3-(2-piperazin-1-ylpyrimidin-5-yl)phenyl]phenyl]pyrimidine-2,4-diamineIC501100.0 [1], 1200.0 [2]

References
This online resource may be cited as follows
MLA
"Quest DatabaseTNF-alpha Inhibitors (IC50, Ki)." AAT Bioquest, Inc.13 Jan2026https://www.aatbio.com/data-sets/tnf-alpha-inhibitors-ic50-ki.
APA
AAT Bioquest, Inc. (2026January 13). Quest DatabaseTNF-alpha Inhibitors (IC50, Ki). AAT Bioquest. https://www.aatbio.com/data-sets/tnf-alpha-inhibitors-ic50-ki.
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