Structure | Compound Name | Standard Type | Standard Values (in nM) |
|---|---|---|---|
| 6,7-Dimethyl-3-[[methyl-[2-[methyl-[[1-[3-(trifluoromethyl)phenyl]indol-3-yl]methyl]amino]ethyl]amino]methyl]chromen-4-one | IC50 | 5000.0 [1], 15000.0 [2], 22000.0 [3] | |
| Rolipram | IC50 | 200.0 [1], 500.0 [2], 12000.0 [3] | |
| Mesalamine | IC50 | 20000.0 [1], 20600000.0 [2] | |
| 1-Propyl-2,4-dioxo-1,4-dihydropteridine-3(2H)-butyric acid ethyl ester | IC50 | 3000.0 [1], 5000.0 [2] | |
| 4-N-Benzyl-4-N-[2-[3-(2-piperazin-1-ylpyrimidin-5-yl)phenyl]phenyl]pyrimidine-2,4-diamine | IC50 | 1100.0 [1], 1200.0 [2] | |
MLA | "Quest Database™ TNF-alpha Inhibitors (IC50, Ki)." AAT Bioquest, Inc., 13 Jan. 2026, https://www.aatbio.com/data-sets/tnf-alpha-inhibitors-ic50-ki. | |
APA | AAT Bioquest, Inc. (2026, January 13). Quest Database™ TNF-alpha Inhibitors (IC50, Ki). AAT Bioquest. https://www.aatbio.com/data-sets/tnf-alpha-inhibitors-ic50-ki. | |
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