Transcription initiation factor IIA alpha and bTranscription initiation factor IIA alpha and beta chains Inhibitors (IC50, Ki)

Structure ▲ ▼	Compound Name ▲ ▼	Standard Type ▲ ▼	Standard Values (in nM) ▲ ▼
	(2R)-2-(Benzylsulfonylamino)-N-[(2S)-1-[(4-carbamimidoylphenyl)methylamino]-1-oxo-4-piperidin-4-ylbutan-2-yl]-5-phenylpentanamide	Ki	240.0 [1]
	(2R)-2-(Benzylsulfonylamino)-N-[(2S)-1-[(4-carbamimidoylphenyl)methylamino]-1-oxo-4-piperidin-4-ylbutan-2-yl]-5-pyridin-4-ylpentanamide	Ki	1200.0 [1]
	(2R)-2-(Benzylsulfonylamino)-N-[(2S)-1-[(4-carbamimidoylphenyl)methylamino]-1-oxo-4-piperidin-4-ylbutan-2-yl]-5-(tetrazol-1-yl)pentanamide	Ki	4700.0 [1]
	(2S)-2-[[(2R)-2-(Benzylsulfonylamino)-2-phenylacetyl]amino]-N-[(4-carbamimidoylphenyl)methyl]-4-piperidin-4-ylbutanamide	Ki	1700.0 [1]
	(2S)-2-[[(2R)-2-(Benzylsulfonylamino)-4-pyridin-4-ylbutanoyl]amino]-N-[(4-carbamimidoylphenyl)methyl]-4-piperidin-4-ylbutanamide	Ki	3900.0 [1]
	(2S)-2-[[(2R)-2-(Benzylsulfonylamino)-4-(1-oxidopyridin-1-ium-4-yl)butanoyl]amino]-N-[(4-carbamimidoylphenyl)methyl]-4-piperidin-4-ylbutanamide	Ki	9000.0 [1]
	Methyl 3-[[(2R)-1-[[(2S)-1-[(4-carbamimidoylphenyl)methylamino]-1-oxo-4-piperidin-4-ylbutan-2-yl]amino]-1-oxo-5-phenylpentan-2-yl]sulfamoylmethyl]benzoate	Ki	920.0 [1]
	3-[[(2R)-1-[[(2S)-1-[(4-Carbamimidoylphenyl)methylamino]-1-oxo-4-piperidin-4-ylbutan-2-yl]amino]-1-oxo-5-phenylpentan-2-yl]sulfamoylmethyl]benzoic acid	Ki	4400.0 [1]
	(2S)-2-[[(2R)-4-(1-Acetylpiperidin-4-yl)-2-(benzylsulfonylamino)butanoyl]amino]-N-[(4-carbamimidoylphenyl)methyl]-4-piperidin-4-ylbutanamide	Ki	8000.0 [1]
	Methyl 4-[(3R)-3-(benzylsulfonylamino)-4-[[(2S)-1-[(4-carbamimidoylphenyl)methylamino]-1-oxo-4-piperidin-4-ylbutan-2-yl]amino]-4-oxobutyl]piperidine-1-carboxylate	Ki	13000.0 [1]
	(2S)-2-[[(2R)-2-(Benzylsulfonylamino)-4-[1-(2-methoxyacetyl)piperidin-4-yl]butanoyl]amino]-N-[(4-carbamimidoylphenyl)methyl]-4-piperidin-4-ylbutanamide	Ki	4500.0 [1]
	4-[(3R)-3-(Benzylsulfonylamino)-4-[[(2S)-1-[(4-carbamimidoylphenyl)methylamino]-1-oxo-4-piperidin-4-ylbutan-2-yl]amino]-4-oxobutyl]-N-methylpiperidine-1-carboxamide	Ki	4800.0 [1]
	4-[(3R)-3-(Benzylsulfonylamino)-4-[[(2S)-1-[(4-carbamimidoylphenyl)methylamino]-1-oxo-4-piperidin-4-ylbutan-2-yl]amino]-4-oxobutyl]-N,N-dimethylpiperidine-1-carboxamide	Ki	13000.0 [1]
	(2S)-2-[[(2R)-2-(Benzylsulfonylamino)-4-[1-(cyclopropanecarbonyl)piperidin-4-yl]butanoyl]amino]-N-[(4-carbamimidoylphenyl)methyl]-4-piperidin-4-ylbutanamide	Ki	8500.0 [1]
	(2S)-2-[[(2R)-2-(Benzylsulfonylamino)-4-(1-butanoylpiperidin-4-yl)butanoyl]amino]-N-[(4-carbamimidoylphenyl)methyl]-4-piperidin-4-ylbutanamide	Ki	5500.0 [1]
	(2S)-2-[[(2R)-2-(Benzylsulfonylamino)-4-[1-(2-methylpropanoyl)piperidin-4-yl]butanoyl]amino]-N-[(4-carbamimidoylphenyl)methyl]-4-piperidin-4-ylbutanamide	Ki	13000.0 [1]
	(2R)-2-(Benzylsulfonylamino)-N-[(2S)-1-[(4-carbamimidoylphenyl)methylamino]-1-oxo-4-piperidin-4-ylbutan-2-yl]-5-piperidin-4-ylpentanamide	Ki	800.0 [1]
	(2R)-5-(1-Acetylpiperidin-4-yl)-2-(benzylsulfonylamino)-N-[(2S)-1-[(4-carbamimidoylphenyl)methylamino]-1-oxo-4-piperidin-4-ylbutan-2-yl]pentanamide	Ki	3800.0 [1]
	Methyl 4-[(4R)-4-(benzylsulfonylamino)-5-[[(2S)-1-[(4-carbamimidoylphenyl)methylamino]-1-oxo-4-piperidin-4-ylbutan-2-yl]amino]-5-oxopentyl]piperidine-1-carboxylate	Ki	3600.0 [1]
	(2S)-2-[[(2R)-2-(Benzylsulfonylamino)-4-(1-propanoylpiperidin-4-yl)butanoyl]amino]-N-[(4-carbamimidoylphenyl)methyl]-4-piperidin-4-ylbutanamide	Ki	5600.0 [1]
	(2S)-2-[[(2R)-2-(Benzylsulfonylamino)-4-piperidin-4-ylbutanoyl]amino]-N-[(4-carbamimidoylphenyl)methyl]-4-piperidin-4-ylbutanamide	Ki	4200.0 [1]
	(2R)-2-(Benzylsulfonylamino)-N-[(2S)-1-[(4-carbamimidoylphenyl)methylamino]-1-oxo-4-piperidin-4-ylbutan-2-yl]-5-(1-oxidopyridin-1-ium-4-yl)pentanamide	Ki	4900.0 [1]

Entire TableStructureCompound NameStandard TypeStandard Values (in nM)

Items per page: 510All1 - 10 of 22 ⟨⟩

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References

This online tool may be cited as follows

MLA	"Quest Database™ Transcription initiation factor IIA alpha and bTranscription initiation factor IIA alpha and beta chains Inhibitors (IC50, Ki)." AAT Bioquest, Inc., 8 May. 2024, https://www.aatbio.com/data-sets/transcription-initiation-factor-iia-alpha-and-btranscription-initiation-factor-iia-alpha-and-beta-chains-inhibitors-ic50-ki.
APA	AAT Bioquest, Inc. (2024, May 8). Quest Database™ Transcription initiation factor IIA alpha and bTranscription initiation factor IIA alpha and beta chains Inhibitors (IC50, Ki). AAT Bioquest. https://www.aatbio.com/data-sets/transcription-initiation-factor-iia-alpha-and-btranscription-initiation-factor-iia-alpha-and-beta-chains-inhibitors-ic50-ki.
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