Transcriptional regulator ERG Inhibitors (IC50, Ki)

Name: Transcriptional regulator ERG Inhibitors (IC50, Ki)
Creator: AAT Bioquest
License: https://www.aatbio.com/tou.html

Structure ▲ ▼	Compound Name ▲ ▼	Standard Type ▲ ▼	Standard Values (in nM) ▲ ▼
	N-(Cyclopropylmethyl)-7-[2,6-dimethoxy-4-(methoxymethyl)phenyl]-2-ethyl-N-(oxan-4-ylmethyl)pyrazolo[1,5-a]pyridin-3-amine;4-methylbenzenesulfonic acid	IC50	16300.0 ^[1]
	(1R,2R)-N-(1-Cyanocyclopropyl)-2-(6-methoxy-1,3,4,5-tetrahydropyrido[4,3-b]indole-2-carbonyl)cyclohexane-1-carboxamide	IC50	100000.0 ^[1]
	N-(4,4-Difluorocyclohexyl)-4-(3-quinolin-2-yl-1,2,4-oxadiazol-5-yl)piperazine-1-carboxamide	IC50	30000.0 ^[1]
	N-(2-Chlorophenyl)-4-(3-quinolin-2-yl-1,2,4-oxadiazol-5-yl)piperazine-1-carboxamide	IC50	12000.0 ^[1]
	N-(2-Chlorophenyl)-4-[3-(1-methylbenzimidazol-2-yl)-1,2,4-oxadiazol-5-yl]piperidine-1-carboxamide	IC50	32000.0 ^[1]
	N-Cyclohexyl-4-(3-quinolin-2-yl-1,2,4-oxadiazol-5-yl)piperazine-1-carboxamide	IC50	30000.0 ^[1]
	(2S)-N-[2-(4-Cyanophenyl)ethyl]-1-[6-(4-methylpiperazin-1-yl)-2-(trifluoromethyl)pyrimidin-4-yl]piperidine-2-carboxamide	IC50	2300.0 ^[1]
	(2S)-N-[2-(4-Cyanophenyl)ethyl]-1-[6-(4-methylpiperazin-1-yl)-2-(trifluoromethyl)pyrimidin-4-yl]pyrrolidine-2-carboxamide	IC50	13000.0 ^[1]
	(2R)-N-[2-(4-Cyanophenyl)ethyl]-1-[6-(4-methylpiperazin-1-yl)-2-(trifluoromethyl)pyrimidin-4-yl]pyrrolidine-2-carboxamide	IC50	5500.0 ^[1]
	(2S)-N-[2-(4-Cyanophenyl)ethyl]-1-[6-(4-methylpiperazin-1-yl)-2-(trifluoromethyl)pyrimidin-4-yl]azetidine-2-carboxamide	IC50	9800.0 ^[1]
	(2R)-N-[2-(4-Cyanophenyl)ethyl]-1-[6-(4-methylpiperazin-1-yl)-2-(trifluoromethyl)pyrimidin-4-yl]azetidine-2-carboxamide	IC50	6000.0 ^[1]
	(2S)-N-[2-(6-Cyanopyridin-3-yl)ethyl]-1-[6-(4-ethylpiperazin-1-yl)-2-(trifluoromethyl)pyrimidin-4-yl]azetidine-2-carboxamide	IC50	30000.0 ^[1]
	(3R)-N-[2-(4-Cyanophenyl)ethyl]-1-[4-methyl-6-(4-methylpiperazin-1-yl)pyrimidin-2-yl]piperidine-3-carboxamide	IC50	3100.0 ^[1]
	(3R)-N-[2-(4-Cyanophenyl)ethyl]-1-[4-(4-methylpiperazin-1-yl)-6-(trifluoromethyl)pyrimidin-2-yl]piperidine-3-carboxamide	IC50	2100.0 ^[1]
	(3R)-N-[2-(4-Cyanophenyl)ethyl]-1-[6-(4-methylpiperazin-1-yl)-2-(trifluoromethyl)pyrimidin-4-yl]piperidine-3-carboxamide	IC50	3200.0 ^[1]
	(3R)-N-[2-(4-Cyanophenyl)ethyl]-1-[6-piperazin-1-yl-2-(trifluoromethyl)pyrimidin-4-yl]piperidine-3-carboxamide	IC50	3500.0 ^[1]
	(3R)-N-[2-(4-Cyanophenyl)ethyl]-1-[6-[4-(oxetan-3-yl)piperazin-1-yl]-2-(trifluoromethyl)pyrimidin-4-yl]piperidine-3-carboxamide	IC50	30000.0 ^[1]
	(3R)-N-[2-(6-Cyanopyridin-3-yl)ethyl]-1-[6-(4-methylpiperazin-1-yl)-2-(trifluoromethyl)pyrimidin-4-yl]piperidine-3-carboxamide	IC50	25000.0 ^[1]
	(3R)-N-[2-(6-Cyanopyridin-3-yl)ethyl]-1-[6-piperazin-1-yl-2-(trifluoromethyl)pyrimidin-4-yl]piperidine-3-carboxamide	IC50	20000.0 ^[1]
	(3R)-N-[2-(2-Cyanopyrimidin-5-yl)ethyl]-1-[6-(4-ethylpiperazin-1-yl)-2-(trifluoromethyl)pyrimidin-4-yl]piperidine-3-carboxamide	IC50	18000.0 ^[1]
	4-[4-[6-[(2S)-2-[2-(4-Cyanophenyl)ethylcarbamoyl]azetidin-1-yl]-2-(trifluoromethyl)pyrimidin-4-yl]phenyl]cyclohexane-1-carboxylic acid	IC50	30000.0 ^[1]

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References

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MLA	"Quest Database™ Transcriptional regulator ERG Inhibitors (IC50, Ki)." AAT Bioquest, Inc., 8 May. 2024, https://www.aatbio.com/data-sets/transcriptional-regulator-erg-inhibitors-ic50-ki.
APA	AAT Bioquest, Inc. (2024, May 8). Quest Database™ Transcriptional regulator ERG Inhibitors (IC50, Ki). AAT Bioquest. https://www.aatbio.com/data-sets/transcriptional-regulator-erg-inhibitors-ic50-ki.
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Transcriptional regulator ERG Inhibitors (IC50, Ki)

References

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