Name: Transcriptional regulator ERG Inhibitors (IC50, Ki)
Creator: AAT Bioquest
License: https://www.aatbio.com/tou.html

Transcriptional regulator ERG Inhibitors (IC50, Ki)

Structure	Compound Name	Standard Type	Standard Values (in nM)
	N-(Cyclopropylmethyl)-7-[2,6-dimethoxy-4-(methoxymethyl)phenyl]-2-ethyl-N-(oxan-4-ylmethyl)pyrazolo[1,5-a]pyridin-3-amine;4-methylbenzenesulfonic acid	IC50	16300.0 ^[1]
	(1R,2R)-N-(1-Cyanocyclopropyl)-2-(6-methoxy-1,3,4,5-tetrahydropyrido[4,3-b]indole-2-carbonyl)cyclohexane-1-carboxamide	IC50	100000.0 ^[1]
	N-(4,4-Difluorocyclohexyl)-4-(3-quinolin-2-yl-1,2,4-oxadiazol-5-yl)piperazine-1-carboxamide	IC50	30000.0 ^[1]
	N-(2-Chlorophenyl)-4-(3-quinolin-2-yl-1,2,4-oxadiazol-5-yl)piperazine-1-carboxamide	IC50	12000.0 ^[1]
	N-(2-Chlorophenyl)-4-[3-(1-methylbenzimidazol-2-yl)-1,2,4-oxadiazol-5-yl]piperidine-1-carboxamide	IC50	32000.0 ^[1]
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References

This online resource may be cited as follows

MLA	"Quest Database™ Transcriptional regulator ERG Inhibitors (IC50, Ki)." AAT Bioquest, Inc., 15 Dec. 2025, https://www.aatbio.com/data-sets/transcriptional-regulator-erg-inhibitors-ic50-ki.
APA	AAT Bioquest, Inc. (2025, December 15). Quest Database™ Transcriptional regulator ERG Inhibitors (IC50, Ki). AAT Bioquest. https://www.aatbio.com/data-sets/transcriptional-regulator-erg-inhibitors-ic50-ki.
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