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Transient receptor potential cation channel subfamily M member 8 Inhibitors (IC50, Ki)

Structure
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Compound Name
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Standard Type
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Standard Values (in nM)
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▼
CID 16095384IC504.0 [1], 160.0 [2], 190.0 [3]
MentholIC5019000.0 [1], 92000.0 [2], 520000.0 [3]
4-({[4-Fluoro-3-(trifluoromethyl)phenyl]methyl}(3-methyl-1-benzothiophen-2-yl)sulfamoyl)benzoic acidIC504.0 [1], 5.0 [2]
5-MethoxytryptamineIC5011600.0 [1], 12400.0 [2]
BctcIC50475.0 [1], 800.0 [2]
5-FluorotryptamineIC5012300.0 [1], 13100.0 [2]
5-BenzyloxytryptamineIC50340.0 [1], 660.0 [2]
5-ChlorotryptamineIC5021500.0 [1], 32200.0 [2]
5-BromotryptamineIC5022700.0 [1], 30400.0 [2]
3-[4-(Trifluoromethyl)-6-[2-(trifluoromethyl)phenyl]-1H-benzimidazol-2-yl]-1-oxa-2-azaspiro[4.5]dec-2-eneIC500.41 [1], 3.0 [2]
7-BenzyloxytryptamineIC503340.0 [1], 8930.0 [2]
1H-Indole-3-ethanamine, N,N'-dimethyl-5-(phenylmethoxy)-IC505630.0 [1], 5960.0 [2]
CID 60195662IC50103.0 [1], 181.0 [2]
Ethyl {2-[5-(benzyloxy)-1H-indol-3-yl]ethyl}carbamateIC5021600.0 [1], 28800.0 [2]
2-(5-Benzyloxy-2-methyl-1H-indol-3-yl)-ethylamineIC501500.0 [1], 2360.0 [2]
4-[(3-Methyl-1-benzothiophen-2-yl)-[[4-(trifluoromethoxy)phenyl]methyl]sulfamoyl]benzoic acidIC501.4 [1], 1.8 [2]
CapsazepineIC5018000.0 [1]
2-(1,3-Dimethyl-2,6-dioxo-1,2,3,6-tetrahydro-7H-purin-7-yl)-N-(4-isopropylphenyl)acetamideIC5030000.0 [1]
N-(p-Amylcinnamoyl)anthranilic acidIC503900.0 [1]
7-Bromo-N-(1-phenylcyclopropyl)-3-[(4-piperidin-1-ylpiperidin-1-yl)methyl]-2-[3-(trifluoromethyl)phenyl]quinoline-4-carboxamideIC5025000.0 [1]
N-[2-Methyl-3-[[4-[4-[[4-(trifluoromethoxy)phenyl]methoxy]piperidin-1-yl]-1,3,5-triazin-2-yl]amino]phenyl]acetamideIC5020000.0 [1]
CID 121513880IC5030000.0 [1]
CID 49783953IC508.3 [1]
(8R)-8-[4-(Trifluoromethyl)phenyl]-N-[(2S)-1,1,1-trifluoropropan-2-yl]-6,8-dihydro-5H-1,7-naphthyridine-7-carboxamideIC5025.0 [1]
(R)-8-{5-[3-Methyl-4-(trifluoromethyl)phenyl]oxazol-2-ylamino}-1,2,3,4-tetrahydronaphthalen-2-olIC5044000.0 [1]
(1R)-N-(4-Fluorophenyl)-1-[4-(trifluoromethyl)phenyl]-3,4-dihydro-1H-isoquinoline-2-carboxamideIC5036.0 [1]
N-[(1R)-2-Amino-2-oxo-1-phenylethyl]-N-[(3-methylphenyl)methyl]benzamideIC50870.0 [1]
N-[(1R)-2-Amino-2-oxo-1-phenylethyl]-N-[[3-(trifluoromethyl)phenyl]methyl]benzamideIC505000.0 [1]
N-[(1R)-2-Amino-2-oxo-1-phenylethyl]-N-[(1R)-1-(3-methoxyphenyl)ethyl]benzamideIC50240.0 [1]
N-[(1R)-2-Amino-2-oxo-1-phenylethyl]-N-[(1R)-1-(3-chlorophenyl)ethyl]benzamideIC50400.0 [1]
N-[(1R)-2-Amino-2-oxo-1-phenylethyl]-N-[(1S)-1-(3-methoxyphenyl)ethyl]benzamideIC5043000.0 [1]
N-[(1R)-2-Amino-2-oxo-1-phenylethyl]-N-[(1R)-1-phenylpropyl]benzamideIC5019000.0 [1]
N-[(1R)-2-Amino-2-oxo-1-phenylethyl]-N-[(1R)-1-(3,5-difluorophenyl)ethyl]benzamideIC5080.0 [1]
N-[(1R)-2-Amino-2-oxo-1-phenylethyl]-N-[(2-chlorophenyl)methyl]benzamideIC505600.0 [1]
N-[(1R)-2-Amino-2-oxo-1-phenylethyl]-N-[(4-chlorophenyl)methyl]benzamideIC5028000.0 [1]
N-[(1R)-2-Amino-2-oxo-1-phenylethyl]-N-[(1R)-1-(3-chlorophenyl)ethyl]-2-hydroxybenzamideIC50100.0 [1]
(2R)-2-[(3-Methoxyphenyl)methyl-(2-phenylacetyl)amino]-2-phenylacetamideIC5019000.0 [1]
N-[(1R)-2-Amino-2-oxo-1-phenylethyl]-N-[(3-fluorophenyl)methyl]benzamideIC508100.0 [1]
N-[(1R)-2-Amino-2-oxo-1-phenylethyl]-N-benzylbenzamideIC5011000.0 [1]
N-[(1R)-2-Amino-2-oxo-1-pyridin-3-ylethyl]-N-[(1R)-1-(3-chlorophenyl)ethyl]benzamideIC504100.0 [1]
N-[(1R)-2-Amino-2-oxo-1-phenylethyl]-N-[(1R)-1-(3-chlorophenyl)ethyl]-3-methylbenzamideIC502100.0 [1]
N-[(1R)-2-Amino-2-oxo-1-phenylethyl]-N-[(1R)-1-(3-chlorophenyl)ethyl]-4-methylbenzamideIC50850.0 [1]
N-[(2R)-1-Amino-1-oxo-3-phenylpropan-2-yl]-N-[(3-methoxyphenyl)methyl]thiophene-2-carboxamideIC5037000.0 [1]
N-[(1R)-2-Amino-2-oxo-1-phenylethyl]-N-[(3-methoxyphenyl)methyl]thiophene-2-carboxamideIC501700.0 [1]
N-[(1R)-2-Amino-2-oxo-1-phenylethyl]-N-[[3-(trifluoromethoxy)phenyl]methyl]benzamideIC504700.0 [1]
N-[(1S)-2-Amino-2-oxo-1-phenylethyl]-N-[(3-methoxyphenyl)methyl]thiophene-2-carboxamideIC5054000.0 [1]
N-[(1R)-2-Amino-2-oxo-1-phenylethyl]-N-[(1R)-1-(3-chlorophenyl)ethyl]-2-methylbenzamideIC50390.0 [1]
N-[(1R)-2-Amino-2-oxo-1-phenylethyl]-N-[(3-chlorophenyl)methyl]benzamideIC503000.0 [1]
N-[(1R)-2-Amino-2-oxo-1-phenylethyl]-N-[(1R)-1-(3-chloro-5-fluorophenyl)ethyl]benzamideIC50180.0 [1]
2-[Benzyl-[3-chloro-5-(trifluoromethyl)pyridin-2-yl]sulfamoyl]benzoic acidIC5015974.0 [1]
4-[Benzyl-(3-chloro-5-cyanopyridin-2-yl)sulfamoyl]benzoic acidIC5023782.0 [1]
4-[Benzyl-[3-cyano-5-(trifluoromethyl)pyridin-2-yl]sulfamoyl]benzoic acidIC502472.0 [1]
4-[Benzyl-[5-chloro-3-(trifluoromethyl)pyridin-2-yl]sulfamoyl]benzoic acidIC501562.0 [1]
4-[(4-Acetamidophenyl)methyl-[3-chloro-5-(trifluoromethyl)pyridin-2-yl]sulfamoyl]benzoic acidIC5018216.0 [1]
3-[[[2-(3-Chlorophenyl)acetyl]-[(1R)-1-(4-fluorophenyl)ethyl]amino]methyl]benzoic acidIC5010000.0 [1]
3-[[[(1R)-1-(4-Fluorophenyl)ethyl]-(3-phenylbenzoyl)amino]methyl]benzoic acidIC50837.0 [1]
3-[[[(1R)-1-(4-Fluorophenyl)ethyl]-(1H-pyrrolo[2,3-c]pyridine-5-carbonyl)amino]methyl]benzoic acidIC50951.0 [1]
3-[[Cinnoline-3-carbonyl-[(1R)-1-(4-fluorophenyl)ethyl]amino]methyl]benzoic acidIC50340.0 [1]
3-[[[(1R)-1-(4-Fluorophenyl)ethyl]-(imidazo[1,2-a]pyridine-2-carbonyl)amino]methyl]benzoic acidIC50307.0 [1]
3-[[[(1R)-1-(4-Fluorophenyl)ethyl]-(4-phenoxybenzoyl)amino]methyl]benzoic acidIC506166.0 [1]
5-[[[(1R)-1-(4-Fluorophenyl)ethyl]-(quinoline-3-carbonyl)amino]methyl]-2-methylbenzoic acidIC507820.0 [1]
2-[3-[[[(1R)-1-(4-Fluorophenyl)ethyl]-(quinoline-3-carbonyl)amino]methyl]phenyl]acetic acidIC503249.0 [1]
N-[(1R)-1-(4-Fluorophenyl)ethyl]-N-[[3-(2H-tetrazol-5-yl)phenyl]methyl]quinoline-3-carboxamideIC501613.0 [1]
3-[[(4-Fluorophenyl)methyl-(quinoline-3-carbonyl)amino]methyl]benzoic acidIC509356.0 [1]
3-[[[(1S)-2-Hydroxy-1-phenylethyl]-(quinoline-3-carbonyl)amino]methyl]benzoic acidIC506863.0 [1]
3-[[[(1R)-1-(2,4-Difluorophenyl)ethyl]-(quinoline-3-carbonyl)amino]methyl]benzoic acidIC50288.0 [1]
3-[[2-(4-Fluorophenyl)propan-2-yl-(quinoline-3-carbonyl)amino]methyl]benzoic acidIC5010000.0 [1]
3-[[1-(4-Methoxyphenyl)ethyl-(quinoline-3-carbonyl)amino]methyl]benzoic acidIC506104.0 [1]
6-[[[(1R)-1-(2,4-Difluorophenyl)ethyl]-(isoquinoline-3-carbonyl)amino]methyl]pyridine-2-carboxylic acidIC50190.0 [1]
(2S,4R,5S)-4-Fluoro-1-(4-fluorophenyl)sulfonyl-N-[[5-fluoro-2-[2-(trifluoromethyl)pyrimidin-5-yl]pyridin-4-yl]methyl]-5-methylpyrrolidine-2-carboxamideIC5020000.0 [1]
2-Amino-N-[(1R)-2-amino-2-oxo-1-phenylethyl]-N-[(1R)-1-(3-chlorophenyl)ethyl]benzamideIC50420.0 [1]
2-[Benzoyl-[(3-methoxyphenyl)methyl]amino]-2-phenylacetic acidIC5059000.0 [1]
N-[(1R)-2-(Dimethylamino)-2-oxo-1-phenylethyl]-N-[(3-methoxyphenyl)methyl]benzamideIC5086000.0 [1]
N-[(1R)-2-Amino-2-oxo-1-phenylethyl]-N-[(1R)-1-(3-chlorophenyl)ethyl]pyridine-3-carboxamideIC502500.0 [1]
N-[(2R)-1-Amino-1-oxopropan-2-yl]-N-[(3-methoxyphenyl)methyl]benzamideIC50100000.0 [1]
N-[(1R)-2-Amino-2-oxo-1-phenylethyl]-N-[[4-[(4-fluorophenyl)methoxy]-3-methoxyphenyl]methyl]thiophene-2-carboxamideIC50100000.0 [1]
N-(2-Amino-2-oxoethyl)-N-[[4-[(4-fluorophenyl)methoxy]-3-methoxyphenyl]methyl]thiophene-2-carboxamideIC509100.0 [1]
N-[(3-Methoxyphenyl)methyl]-N-[(1R)-2-(methylamino)-2-oxo-1-phenylethyl]benzamideIC5010000.0 [1]
Methyl (2R)-2-[benzoyl-[(3-methoxyphenyl)methyl]amino]-2-phenylacetateIC50210.0 [1]
4-[(3S,4R)-1-(2,4-Dichlorophenyl)sulfonyl-4-hydroxy-4-(hydroxymethyl)pyrrolidin-3-yl]oxy-2-fluorobenzonitrileIC5010000.0 [1]
N-[(S)-(2-Methylphenyl)-[3-(trifluoromethyl)pyridin-2-yl]methyl]quinoline-7-carboxamideIC5020000.0 [1]
N-[(R)-1,3-Thiazol-2-yl-[3-(trifluoromethyl)pyridin-2-yl]methyl]quinoline-7-carboxamideIC5010000.0 [1]
N-[(S)-Pyridin-2-yl-[3-(trifluoromethyl)pyridin-2-yl]methyl]quinoline-7-carboxamideIC5010000.0 [1]
Quinolin-6-yl-[(1R)-1-[4-(trifluoromethyl)phenyl]-3,4-dihydro-1H-isoquinolin-2-yl]methanoneIC50390.0 [1]
N-[(S)-[3-Fluoro-4-(trifluoromethyl)phenyl]-[2-(trifluoromethyl)phenyl]methyl]quinoline-7-carboxamideIC50109.0 [1]
N-[(S)-Cyclohexyl-[3-(trifluoromethyl)pyridin-2-yl]methyl]quinoline-7-carboxamideIC50301.0 [1]
N-[(S)-[4-(Trifluoromethyl)phenyl]-[4-(trifluoromethyl)pyridin-3-yl]methyl]quinoline-7-carboxamideIC50311.0 [1]
N-[(1S)-2-Phenyl-1-[3-(trifluoromethyl)pyridin-2-yl]ethyl]quinoline-7-carboxamideIC501140.0 [1]
(5R)-N-(4-Fluorophenyl)-5-[4-(trifluoromethyl)phenyl]-7,8-dihydro-5H-1,6-naphthyridine-6-carboxamideIC50391.0 [1]
(8R)-N-(4-Fluorophenyl)-8-[4-(trifluoromethyl)phenyl]-6,8-dihydro-5H-1,7-naphthyridine-7-carboxamideIC5014.0 [1]
(8R)-N-Pyridin-3-yl-8-[4-(trifluoromethyl)phenyl]-6,8-dihydro-5H-1,7-naphthyridine-7-carboxamideIC5024.0 [1]
(5R)-N-(4-Fluorophenyl)-5-[4-(trifluoromethyl)phenyl]-7,8-dihydro-5H-pyrido[3,4-b]pyrazine-6-carboxamideIC50200.0 [1]
N-(4-Fluorophenyl)-1-[4-(trifluoromethyl)phenyl]-3,4-dihydro-1H-2,6-naphthyridine-2-carboxamideIC501262.0 [1]
N-(4-Fluorophenyl)-1-[4-(trifluoromethyl)phenyl]-3,4-dihydro-1H-2,7-naphthyridine-2-carboxamideIC50463.0 [1]
N-(4-Fluorophenyl)-8-[4-(trifluoromethyl)phenyl]-6,8-dihydro-5H-pyrido[3,4-d]pyrimidine-7-carboxamideIC50786.0 [1]
N-Benzyl-N-[3-chloro-5-(trifluoromethyl)pyridin-2-yl]benzenesulfonamideIC50183.0 [1]
(1R)-1-[4-(Trifluoromethyl)phenyl]-N-[(2R)-1,1,1-trifluoropropan-2-yl]-3,4-dihydro-1H-isoquinoline-2-carboxamideIC5052.0 [1]
(1R)-N-Pyridin-2-yl-1-[4-(trifluoromethyl)phenyl]-3,4-dihydro-1H-isoquinoline-2-carboxamideIC50171.0 [1]
(8R)-8-[3-Fluoro-4-(trifluoromethyl)phenyl]-N-[(2S)-1,1,1-trifluoropropan-2-yl]-6,8-dihydro-5H-1,7-naphthyridine-7-carboxamideIC5012.0 [1]
8-Bromo-N-[4-(trifluoromethyl)phenyl]spiro[3,4-dihydrochromene-2,4'-piperidine]-1'-carboxamideIC5018.9 [1]
Items per page: 1 - 10 of 100
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References

This online tool may be cited as follows

MLA

"Quest Database™ Transient receptor potential cation channel subfamily M member 8 Inhibitors (IC50, Ki)." AAT Bioquest, Inc., 9 May. 2024, https://www.aatbio.com/data-sets/transient-receptor-potential-cation-channel-subfamily-m-member-8-inhibitors-ic50-ki.

APA

AAT Bioquest, Inc. (2024, May 9). Quest Database™ Transient receptor potential cation channel subfamily M member 8 Inhibitors (IC50, Ki). AAT Bioquest. https://www.aatbio.com/data-sets/transient-receptor-potential-cation-channel-subfamily-m-member-8-inhibitors-ic50-ki.
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