Transmembrane protease serine 11D Inhibitors (IC50, Ki)

Name: Transmembrane protease serine 11D Inhibitors (IC50, Ki)
Creator: AAT Bioquest
License: https://www.aatbio.com/tou.html

Structure ▲ ▼	Compound Name ▲ ▼	Standard Type ▲ ▼	Standard Values (in nM) ▲ ▼
	N-(Benzylsulfonyl)seryl-N~1~-{4-[(Z)-amino(imino)methyl]benzyl}serinamide	Ki	78.0 ^[1]
	CID 46899577	Ki	19.0 ^[1]
	N-(Benzylsulfonyl)-3-Cyclohexyl-D-Alanyl-N-(4-Carbamimidoylbenzyl)-L-Prolinamide	Ki	108.0 ^[1]
	N-(Benzylsulfonyl)-D-Valyl-N-(4-Carbamimidoylbenzyl)-L-Prolinamide	Ki	76.0 ^[1]
	N-(Benzylsulfonyl)-D-Leucyl-N-(4-Carbamimidoylbenzyl)-L-Prolinamide	Ki	120.0 ^[1]
	Inhibitor 1 [Colombo et al., 2012]	Ki	8.4 ^[1]
	(2S)-2-[[(2S)-2-[[(2S)-5-Amino-2-[[(2S)-2-[(2-aminobenzoyl)amino]-5-(diaminomethylideneamino)pentanoyl]amino]-5-oxopentanoyl]amino]-3-carboxypropanoyl]amino]-5-(diaminomethylideneamino)pentanoic acid	Ki	54.3 ^[1]
	(2S)-6-Amino-2-[[(2S)-2-[[(2S)-5-amino-2-[[(2S)-2-[(2-aminobenzoyl)amino]-5-(diaminomethylideneamino)pentanoyl]amino]-5-oxopentanoyl]amino]-3-carboxypropanoyl]amino]hexanoic acid	Ki	112.3 ^[1]
	(2S)-1-[(2R)-6-Amino-2-(benzylsulfonylamino)hexanoyl]-N-[(4-carbamimidoylphenyl)methyl]pyrrolidine-2-carboxamide	Ki	40.0 ^[1]
	N~2~-(Benzylsulfonyl)-D-Arginyl-N-(4-Carbamimidoylbenzyl)glycinamide	Ki	430.0 ^[1]
	Benzyl N-[(5S)-5-[[(2R)-2-(benzylsulfonylamino)-3-hydroxypropanoyl]amino]-6-[(4-carbamimidoylphenyl)methylamino]-6-oxohexyl]carbamate	Ki	51.0 ^[1]
	(2S)-1-[(2R)-2-(Benzylsulfonylamino)-3-phenylpropanoyl]-N-[(4-carbamimidoylphenyl)methyl]pyrrolidine-2-carboxamide	Ki	98.0 ^[1]
	(2S)-1-[(2R)-2-(Benzylsulfonylamino)-4-phenylbutanoyl]-N-[(4-carbamimidoylphenyl)methyl]pyrrolidine-2-carboxamide	Ki	63.0 ^[1]
	Benzyl N-[(5R)-5-(benzylsulfonylamino)-6-[(2S)-2-[(4-carbamimidoylphenyl)methylcarbamoyl]pyrrolidin-1-yl]-6-oxohexyl]carbamate	Ki	53.0 ^[1]
	(2S)-1-[(2R)-2-(Benzylsulfonylamino)-6-(diaminomethylideneamino)hexanoyl]-N-[(4-carbamimidoylphenyl)methyl]pyrrolidine-2-carboxamide	Ki	13.0 ^[1]
	(2S)-1-[(2R)-2-(Benzylsulfonylamino)-3-(4-cyanophenyl)propanoyl]-N-[(4-carbamimidoylphenyl)methyl]pyrrolidine-2-carboxamide	Ki	311.0 ^[1]
	(2S)-1-[(2R)-2-(Benzylsulfonylamino)-3-(4-carbamimidoylphenyl)propanoyl]-N-[(4-carbamimidoylphenyl)methyl]pyrrolidine-2-carboxamide	Ki	168.0 ^[1]
	(2S)-1-[(2R)-2-(Benzylsulfonylamino)-5-oxo-5-(4-pyrimidin-2-ylpiperazin-1-yl)pentanoyl]-N-[(4-carbamimidoylphenyl)methyl]pyrrolidine-2-carboxamide	Ki	17.0 ^[1]
	Benzyl 4-[(3R)-3-(benzylsulfonylamino)-4-[(2S)-2-[(4-carbamimidoylphenyl)methylcarbamoyl]pyrrolidin-1-yl]-4-oxobutanoyl]piperazine-1-carboxylate	Ki	135.0 ^[1]
	(2S)-1-[(2R)-2-(Benzylsulfonylamino)-4-[4-[3-(dimethylamino)propyl]piperazin-1-yl]-4-oxobutanoyl]-N-[(4-carbamimidoylphenyl)methyl]pyrrolidine-2-carboxamide	Ki	149.0 ^[1]
	4-[[[(2S,4R)-4-(Benzylsulfonylamino)-7-(diaminomethylideneamino)-3-oxoheptan-2-yl]amino]methyl]benzenecarboximidamide	Ki	30.0 ^[1]
	4-[[[(2S,4R)-4-(Benzylsulfonylamino)-7-(diaminomethylideneamino)-3-oxo-1-phenylheptan-2-yl]amino]methyl]benzenecarboximidamide	Ki	57.0 ^[1]
	(3S,5R)-5-(Benzylsulfonylamino)-3-[(4-carbamimidoylphenyl)methylamino]-8-(diaminomethylideneamino)-4-oxooctanoic acid	Ki	422.0 ^[1]
	(2S)-1-[(2R)-4-(4-Benzylpiperazin-1-yl)-2-(benzylsulfonylamino)-4-oxobutanoyl]-N-[(4-carbamimidoylphenyl)methyl]pyrrolidine-2-carboxamide	Ki	158.0 ^[1]
	(2S)-1-[(2R)-2-(Benzylsulfonylamino)-4-oxo-4-(4-propan-2-ylpiperazin-1-yl)butanoyl]-N-[(4-carbamimidoylphenyl)methyl]pyrrolidine-2-carboxamide	Ki	221.0 ^[1]
	4-[[[(4S,6R)-6-(Benzylsulfonylamino)-9-(diaminomethylideneamino)-5-oxononan-4-yl]amino]methyl]benzenecarboximidamide	Ki	15.0 ^[1]
	(2S)-1-[(2R)-2-(Benzylsulfonylamino)-4-[4-(2,5-dimethylphenyl)piperazin-1-yl]-4-oxobutanoyl]-N-[(4-carbamimidoylphenyl)methyl]pyrrolidine-2-carboxamide	Ki	73.0 ^[1]
	(2S)-1-[(2R)-2-(Benzylsulfonylamino)-4-[4-(2-hydroxyethyl)piperazin-1-yl]-4-oxobutanoyl]-N-[(4-carbamimidoylphenyl)methyl]pyrrolidine-2-carboxamide	Ki	210.0 ^[1]
	Benzyl N-[(5S,7R)-7-(benzylsulfonylamino)-5-[(4-carbamimidoylphenyl)methylamino]-10-(diaminomethylideneamino)-6-oxodecyl]carbamate	Ki	34.0 ^[1]
	4-[[[(4S,6R)-6-(Benzylsulfonylamino)-9-(diaminomethylideneamino)-2-methyl-5-oxononan-4-yl]amino]methyl]benzenecarboximidamide	Ki	47.0 ^[1]
	Tert-butyl (4R)-4-(benzylsulfonylamino)-5-[(2S)-2-[(4-carbamimidoylphenyl)methylcarbamoyl]pyrrolidin-1-yl]-5-oxopentanoate	Ki	36.0 ^[1]
	(3R)-3-(Benzylsulfonylamino)-4-[(2S)-2-[(4-carbamimidoylphenyl)methylcarbamoyl]pyrrolidin-1-yl]-4-oxobutanoic acid	Ki	1425.0 ^[1]
	4-[[[(3S,5R)-5-(Benzylsulfonylamino)-8-(diaminomethylideneamino)-2-methyl-4-oxooctan-3-yl]amino]methyl]benzenecarboximidamide	Ki	22.0 ^[1]
	4-[[[(2S,4R)-4-(Benzylsulfonylamino)-7-(diaminomethylideneamino)-1-hydroxy-3-oxoheptan-2-yl]amino]methyl]benzenecarboximidamide	Ki	34.0 ^[1]
	Tert-butyl (3S,5R)-5-(benzylsulfonylamino)-3-[(4-carbamimidoylphenyl)methylamino]-8-(diaminomethylideneamino)-4-oxooctanoate	Ki	512.0 ^[1]
	Tert-butyl (3R)-3-(benzylsulfonylamino)-4-[(2S)-2-[(4-carbamimidoylphenyl)methylcarbamoyl]pyrrolidin-1-yl]-4-oxobutanoate	Ki	38.0 ^[1]
	(2S)-1-[(2R)-2-(Benzylsulfonylamino)-5-oxo-5-piperazin-1-ylpentanoyl]-N-[(4-carbamimidoylphenyl)methyl]pyrrolidine-2-carboxamide	Ki	68.0 ^[1]
	4-[[[(5R)-5-(Benzylsulfonylamino)-8-(diaminomethylideneamino)-4-oxooctan-3-yl]amino]methyl]benzenecarboximidamide	Ki	14.0 ^[1]
	4-[[[(3S,4S,6R)-6-(Benzylsulfonylamino)-9-(diaminomethylideneamino)-3-methyl-5-oxononan-4-yl]amino]methyl]benzenecarboximidamide	Ki	23.0 ^[1]
	Benzyl 4-[(4R)-4-(benzylsulfonylamino)-5-[(2S)-2-[(4-carbamimidoylphenyl)methylcarbamoyl]pyrrolidin-1-yl]-5-oxopentanoyl]piperazine-1-carboxylate	Ki	38.0 ^[1]
	(2S)-1-[(2R)-2-(Benzylsulfonylamino)-4-oxo-4-(4-pyrimidin-2-ylpiperazin-1-yl)butanoyl]-N-[(4-carbamimidoylphenyl)methyl]pyrrolidine-2-carboxamide	Ki	43.0 ^[1]
	(2S)-1-[(2R)-2-(Benzylsulfonylamino)-4-morpholin-4-yl-4-oxobutanoyl]-N-[(4-carbamimidoylphenyl)methyl]pyrrolidine-2-carboxamide	Ki	183.0 ^[1]
	(2S)-1-[(2R)-2-(Benzylsulfonylamino)-4-oxo-4-piperazin-1-ylbutanoyl]-N-[(4-carbamimidoylphenyl)methyl]pyrrolidine-2-carboxamide	Ki	202.0 ^[1]
	4-[[[(4S,6R)-6-(Benzylsulfonylamino)-1,9-bis(diaminomethylideneamino)-5-oxononan-4-yl]amino]methyl]benzenecarboximidamide	Ki	457.0 ^[1]

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MLA	"Quest Database™ Transmembrane protease serine 11D Inhibitors (IC50, Ki)." AAT Bioquest, Inc., 8 May. 2024, https://www.aatbio.com/data-sets/transmembrane-protease-serine-11d-inhibitors-ic50-ki.
APA	AAT Bioquest, Inc. (2024, May 8). Quest Database™ Transmembrane protease serine 11D Inhibitors (IC50, Ki). AAT Bioquest. https://www.aatbio.com/data-sets/transmembrane-protease-serine-11d-inhibitors-ic50-ki.
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Transmembrane protease serine 11D Inhibitors (IC50, Ki)

References

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