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Transmembrane protease serine 4 Inhibitors (IC50, Ki)

Structure
Compound Name
Standard Type
Standard Values (in nM)
4-(2-Aminoethyl)benzenesulfonyl fluoride hydrochlorideIC5039000.0 [1]
N-[3,5-Bis(trifluoromethyl)phenyl]-5-chloro-2-hydroxybenzamideIC5011000.0 [1]
5-Chloro-2-hydroxy-N-[4-(trifluoromethyl)phenyl]benzamideIC5016000.0 [1]
5-ChlorosalicylanilideIC5050000.0 [1]
5-Chloro-2-hydroxy-N-[3-(trifluoromethyl)phenyl]benzamideIC5013000.0 [1]
5-Chloro-N-(3,5-dichlorophenyl)-2-hydroxybenzamideIC5019000.0 [1]
Benzamide, 5-chloro-N-(4-cyanophenyl)-2-hydroxy-IC5076000.0 [1]
N-[3,5-Bis(trifluoromethyl)phenyl]-5-bromo-2-hydroxy-benzamideIC5013000.0 [1]
N-[3,5-Bis(trifluoromethyl)phenyl]-2-hydroxy-benzamideIC50100000.0 [1]
N-[3,5-Bis(trifluoromethyl)phenyl]-2-hydroxy-5-nitro-benzamideIC5012000.0 [1]
5-Chloro-N-(3,5-dimethylphenyl)-2-hydroxybenzamideIC5039000.0 [1]
N-[3,5-Bis(trifluoromethyl)phenyl]-5-fluoro-2-hydroxy-benzamideIC5029000.0 [1]
N-[3,5-Bis(trifluoromethyl)phenyl]-2-hydroxy-5-methyl-benzamideIC5028000.0 [1]
N-[3,5-Bis(trifluoromethyl)phenyl]-2-hydroxy-5-methoxy-benzamideIC5029000.0 [1]
CID 17860163IC5028000.0 [1]
5-Chloro-n-[4-chloro-3-(trifluoromethyl)phenyl]-2-hydroxybenzamideIC5035000.0 [1]
CID 23070355IC5012000.0 [1]
CID 23070359IC5020000.0 [1]
N-[[3,5-Bis(trifluoromethyl)phenyl]methyl]-5-chloro-2-hydroxybenzamideIC5018000.0 [1]
N-[4-Bromo-3-(trifluoromethyl)phenyl]-5-chloro-2-hydroxybenzamideIC5030000.0 [1]
5-Chloro-2-hydroxy-N-[3-methoxy-5-(trifluoromethyl)phenyl]benzamideIC5016000.0 [1]
N-[3,5-Bis(trifluoromethyl)phenyl]-5-chloro-2-phenylmethoxybenzamideIC50100000.0 [1]
N-[3,4-Bis(trifluoromethyl)phenyl]-5-chloro-2-hydroxybenzamideIC5013000.0 [1]
CID 71508779IC5010000.0 [1]
CID 71555039IC50100000.0 [1]
[2-[[3,5-Bis(trifluoromethyl)phenyl]carbamoyl]-4-chloro-phenyl] AcetateIC50100000.0 [1]
N-[3-Bromo-5-(trifluoromethyl)phenyl]-5-chloro-2-hydroxybenzamideIC5012000.0 [1]
5-Chloro-N-(6-chloropyridin-3-yl)-2-hydroxybenzamideIC50100000.0 [1]
5-Chloro-2-hydroxy-N-quinolin-3-ylbenzamideIC5085000.0 [1]
N-[3,5-Bis(trifluoromethyl)phenyl]-1-hydroxynaphthalene-2-carboxamideIC50100000.0 [1]
CID 17860285IC50100000.0 [1]
5-Chloro-2-hydroxy-N-pyrimidin-2-ylbenzamideIC50100000.0 [1]
N-[3,5-Bis(trifluoromethyl)phenyl]-4-oxo-1H-quinoline-3-carboxamideIC50100000.0 [1]
5-Chloro-N-(5-cyanopyridin-2-yl)-2-hydroxybenzamideIC5080000.0 [1]
N-[3,5-Bis(trifluoromethyl)phenyl]-3-chloro-2-hydroxybenzamideIC5012000.0 [1]
3-N-[3,5-Bis(trifluoromethyl)phenyl]-4-hydroxybenzene-1,3-dicarboxamideIC50100000.0 [1]
5-Chloro-2-hydroxy-N-[4-methoxy-3,5-bis(trifluoromethyl)phenyl]benzamideIC5012000.0 [1]
5-Chloro-2-hydroxy-N-[5-(trifluoromethyl)pyridin-2-yl]benzamideIC50100000.0 [1]
N-[4-Bromo-3,5-bis(trifluoromethyl)phenyl]-5-chloro-2-hydroxybenzamideIC506000.0 [1]
N-[3,5-Bis(trifluoromethyl)phenyl]-5-chloro-2-oxo-1H-pyridine-3-carboxamideIC50100000.0 [1]
CID 9976653IC5019000.0 [1]



References

This online tool may be cited as follows

MLA

"Quest Database™ Transmembrane protease serine 4 Inhibitors (IC50, Ki)." AAT Bioquest, Inc.9 May2024https://www.aatbio.com/data-sets/transmembrane-protease-serine-4-inhibitors-ic50-ki.

APA

AAT Bioquest, Inc. (2024May 9). Quest Database™ Transmembrane protease serine 4 Inhibitors (IC50, Ki). AAT Bioquest. https://www.aatbio.com/data-sets/transmembrane-protease-serine-4-inhibitors-ic50-ki.
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