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Trypsin Inhibitors (IC50, Ki)

Structure
▲
▼
Compound Name
▲
▼
Standard Type
▲
▼
Standard Values (in nM)
▲
▼
RazaxabanKi4200.0 [1], 10000.0 [2]
QuercetinIC5015400.0 [1], 19000.0 [2]
QuercetinKi13100.0 [1]
Bis(5-amidino-2-benzimidazolyl)methaneIC504400.0 [1]
Bis(5-amidino-2-benzimidazolyl)methaneKi90.0 [1], 19000.0 [2]
(2S)-3-(7-Carbamimidoylnaphthalen-2-yl)-2-[4-[(3S)-1-ethanimidoylpyrrolidin-3-yl]oxyphenyl]propanoic acidIC503200.0 [1]
(2S)-3-(7-Carbamimidoylnaphthalen-2-yl)-2-[4-[(3S)-1-ethanimidoylpyrrolidin-3-yl]oxyphenyl]propanoic acidKi620.0 [1]
N-[(6-Amino-2-methylpyridin-3-yl)methyl]-2-[6-methyl-2-oxo-3-(2-phenylethylamino)pyrazin-1-yl]acetamideIC501800.0 [1]
N-[(6-Amino-2-methylpyridin-3-yl)methyl]-2-[6-methyl-2-oxo-3-(2-phenylethylamino)pyrazin-1-yl]acetamideKi1800.0 [1]
Phenylmethylsulfonyl fluorideIC50110000.0 [1]
Phenylmethylsulfonyl fluorideKi10010.0 [1]
DabigatranKi50.0 [1], 50.3 [2]
RutinIC5016000.0 [1]
RutinKi17500.0 [1]
MelagatranIC5011.9 [1]
MelagatranKi4.3 [1]
2-[3-(Aminomethyl)phenyl]-N-[2-fluoro-4-(2-methylsulfonylphenyl)phenyl]-5-(trifluoromethyl)pyrazole-3-carboxamideKi60.0 [1]
2-[3-(Aminomethyl)phenyl]-N-[2-fluoro-4-(2-methylsulfonylphenyl)phenyl]-5-(trifluoromethyl)pyrazole-3-carboxamide;hydrochlorideIC50100000.0 [1]
2-[3-(Aminomethyl)phenyl]-N-[2-fluoro-4-(2-methylsulfonylphenyl)phenyl]-5-(trifluoromethyl)pyrazole-3-carboxamide;hydrochlorideKi60.0 [1]
Bms-740808Ki2800.0 [1]
2-(3-Carbamimidoylphenyl)-5-methyl-N-[4-(2-sulfamoylphenyl)phenyl]pyrazole-3-carboxamideKi16.0 [1]
Benzamidine hydrochloride hydrateKi5011.87 [1], 7943.28 [2]
2-[6-Cyano-3-[(2,2-difluoro-2-pyridin-2-ylethyl)amino]-2-oxopyrazin-1-yl]-N-[(3-fluoropyridin-2-yl)methyl]acetamideIC50213.0 [1]
2-[6-Cyano-3-[(2,2-difluoro-2-pyridin-2-ylethyl)amino]-2-oxopyrazin-1-yl]-N-[(3-fluoropyridin-2-yl)methyl]acetamideKi213000.0 [1]
2-[3-(Aminomethyl)phenyl]-5-methyl-N-[4-(2-sulfamoylphenyl)phenyl]pyrazole-3-carboxamideKi248.0 [1], 250.0 [2]
N-[(6-Amino-2-methylpyridin-3-yl)methyl]-2-[3-[(2,2-difluoro-2-pyridin-2-ylethyl)amino]-6-methyl-2-oxopyrazin-1-yl]acetamideIC50800.0 [1]
N-[(6-Amino-2-methylpyridin-3-yl)methyl]-2-[3-[(2,2-difluoro-2-pyridin-2-ylethyl)amino]-6-methyl-2-oxopyrazin-1-yl]acetamideKi800.0 [1]
Ethyl N-[(2S)-6-amino-1-oxo-1-[5-[[4-(2-phenylethoxy)phenyl]methyl]-1,2,4-oxadiazol-3-yl]hexan-2-yl]carbamateKi190.0 [1]
(2S)-3-(7-Carbamimidoylnaphthalen-2-yl)-2-[4-[(3S)-1-ethanimidoylpyrrolidin-3-yl]oxyphenyl]propanoic acid;hydrochlorideKi620.0 [1], 2000.0 [2]
(2S)-2-[[(2S)-2-[[(1R)-1-(4-Bromophenyl)ethyl]carbamoylamino]-3-(4-hydroxyphenyl)propanoyl]amino]-N-[(2S)-5-(diaminomethylideneamino)-1-oxo-1-(1,3-thiazol-2-yl)pentan-2-yl]-3-methylbutanamideIC5012.0 [1]
3-(3-Carbamimidoylphenyl)-N-[4-(2-sulfamoylphenyl)phenyl]-1,2-oxazole-4-carboxamide;2,2,2-trifluoroacetic acidKi21.0 [1]
1-(3-Carbamimidoylphenyl)-N-[4-(2-sulfamoylphenyl)phenyl]pyrrole-2-carboxamide;2,2,2-trifluoroacetic acidKi56.0 [1]
2-(3-Carbamimidoylphenyl)-5-methyl-N-[4-(2-sulfamoylphenyl)phenyl]pyrazole-3-carboxamide;2,2,2-trifluoroacetic acidKi16.0 [1]
2-(3-Carbamimidoylphenyl)-N-[4-(2-sulfamoylphenyl)phenyl]pyrazole-3-carboxamide;2,2,2-trifluoroacetic acidKi15.0 [1]
Benzyl N-[(2S)-6-amino-1-oxo-1-[5-[[4-(2-phenylethoxy)phenyl]methyl]-1,2,4-oxadiazol-3-yl]hexan-2-yl]carbamateKi35.0 [1]
2-[3-[(2,2-Difluoro-2-pyridin-2-ylethyl)amino]-6-methyl-2-oxopyrazin-1-yl]-N-[(3-fluoropyridin-2-yl)methyl]acetamideIC50252.0 [1]
2-[3-[(2,2-Difluoro-2-pyridin-2-ylethyl)amino]-6-methyl-2-oxopyrazin-1-yl]-N-[(3-fluoropyridin-2-yl)methyl]acetamideKi252000.0 [1]
N-[(1S)-1-[4-(3-Amino-1H-indazol-6-yl)pyridin-2-yl]-2-phenylethyl]-4-(aminomethyl)cyclohexane-1-carboxamideKi64.0 [1]
3-Nitrobenzamidine hydrochlorideKi6309.57 [1], 79432.82 [2]
3-AminobenzenecarboximidamideKi6309.57 [1], 7943.28 [2]
CID 309369Ki10000.0 [1], 79432.82 [2]
SilymarinIC503700.0 [1]
ApixabanKi4200.0 [1]
BaicalinIC501000000.0 [1]
ArgatrobanKi1990.0 [1]
WogoninIC50105000.0 [1]
SivelestatIC502000.0 [1]
CamostatIC501.6 [1]
SulfaguanidineKi1350.0 [1]
Oroxylin AIC5061000.0 [1]
5-(N,N-Hexamethylene)amilorideIC5010000.0 [1]
ThromstopIC50169.0 [1]
VaborbactamIC501000000.0 [1]
DarexabanKi100000.0 [1]
Isoquinoline-1,3,4(2H)-trioneIC505000.0 [1]
GanhuangeninIC5088000.0 [1]
Skullcapflavone IIIC50110000.0 [1]
1-[n-(Naphthalen-2-Ylsulfonyl)glycyl-4-Carbamimidoyl-D-Phenylalanyl]piperidineKi690.0 [1]
Bms-262084IC5050.0 [1]
Unii-IF979jqu3SKi3290.0 [1]
4-[4-(4-Amidinophenyl)piperazinyl]benzenecarboxamidineKi513.0 [1]
N-[(6-Amino-2-methylpyridin-3-yl)methyl]-2-[3-(benzylsulfonylamino)-6-methyl-2-oxopyridin-1-yl]acetamideKi3200.0 [1]
(2S,3S,4S,5R,6S)-3,4,5-Trihydroxy-6-[3-[(4-methoxybenzoyl)amino]-2-[[4-(4-methyl-1,4-diazepan-1-yl)benzoyl]amino]phenoxy]oxane-2-carboxylic acidKi100000.0 [1]
LetaxabanIC5060000.0 [1]
2-[(1R,4S,7S,13S,19S,22S,25S,28S,31R,34S,40S,43S,49S)-25-(4-Aminobutyl)-49-benzyl-4,19-bis[(2S)-butan-2-yl]-34-[3-(diaminomethylideneamino)propyl]-28-[(1R)-1-hydroxyethyl]-22-(hydroxymethyl)-3,6,12,18,21,24,27,30,33,36,39,42,48,51-tetradecaoxo-53,54-dithia-2,5,11,17,20,23,26,29,32,35,38,41,47,50-tetradecazapentacyclo[29.20.4.07,11.013,17.043,47]pentapentacontan-40-yl]acetic acidKi0.1 [1]
4-[4-(4-Carbamimidoylphenyl)-1,4-diazepan-1-yl]benzamidineKi1900.0 [1]
2-{5-[Amino(iminio)methyl]-1H-benzimidazol-2-YL}benzenolateKi23000.0 [1]
alpha,alpha'-Di(amidinophenoxy)-p-xyleneKi316.0 [1]
Unii-1Y3JD5pemsIC50158000.0 [1]
4-[[2-[(4-Carbamimidoylphenoxy)methyl]phenyl]methoxy]benzamidineKi221.0 [1]
6-Chloro-2-(2-Hydroxybiphenyl-3-yl)-1H-Indole-5-CarboxamidineKi230.0 [1]
3-{5-[Amino(iminio)methyl]-1H-indol-2-YL}-1,1'-biphenyl-2-olateKi130.0 [1]
2-(2-Hydroxyphenyl)-1H-indole-5-carboxamidineKi8000.0 [1]
[2-[(3,5-Dimethyl-1-phenylpyrazol-4-yl)amino]-2-oxoethyl] 2-phenylacetateIC50200000.0 [1]
4-MethoxybenzenecarboximidamideKi100000.0 [1]
OroxindinIC501000000.0 [1]
N-[(1R,2S,5S)-2-[(5-Chloro-1H-indole-2-carbonyl)amino]-5-(dimethylcarbamoyl)cyclohexyl]-5-methyl-6,7-dihydro-4H-[1,3]thiazolo[5,4-c]pyridine-2-carboxamideKi100000.0 [1]
Unii-FS64O4K98AKi0.3 [1]
Thrombin Inhibitor 2Ki202000.0 [1]
3-Chloro-N-[2-[(4-fluorophenyl)carbamoyl]-4-methylphenyl]-1-benzothiophene-2-carboxamideKi5000.0 [1]
3-Chloro-N-[4-chloro-2-[(5-chloropyridin-2-yl)carbamoyl]-6-methoxyphenyl]-4-[[4,5-dihydro-1,3-oxazol-2-yl(methyl)amino]methyl]thiophene-2-carboxamideKi10000.0 [1]
(2R)-2-[(4-Chlorophenyl)carbamoylamino]-N-[4-(3-oxomorpholin-4-yl)phenyl]pentanamideIC5010000.0 [1]
Bms-344577Ki10000.0 [1]
1-(2-Naphthylmethyl)-2,3-dioxo-indoline-5-carboxamideIC50352000.0 [1]
1-[[5-(5-Chlorothiophen-2-yl)-1,2-oxazol-3-yl]methyl]-N-(1-propan-2-ylpiperidin-4-yl)indole-2-carboxamideKi100000.0 [1]
Benzo[b]thiophene-2-carboxamide,3-chloro-N-[2-[[(4-chlorophenyl)amino]carbonyl]-4-methylphenyl]-Ki5000.0 [1]
2-BenzylsulfonylguanidineKi1350.0 [1]
({3-[3-(5-Carbamimidoyl-1H-1,3-benzodiazol-2-yl)-2-hydroxyphenyl]-4-hydroxyphenyl}methyl)ureaKi3600.0 [1]
3-[[2-[(6R)-6-[(5-Chloro-2-methoxyphenyl)methyl]-3-(2,2-dimethylhydrazinyl)-7-oxo-5,6-dihydro-2H-1,4-diazepin-1-yl]acetyl]amino]benzoic acid;hydrochlorideIC5030000.0 [1]
Amido phenyl pyruvic acidKi10000.0 [1]
6-[4-[2-[[(3R)-3-Hydroxypyrrolidin-1-yl]methyl]phenyl]phenyl]-1-(4-methoxyphenyl)-3-(trifluoromethyl)-4,5-dihydropyrazolo[3,4-c]pyridin-7-oneKi3000.0 [1]
(3S)-2-[(2S)-2-[[(2S)-2-Cyclohexyl-2-(pyrazine-2-carbonylamino)acetyl]amino]-3,3-dimethylbutanoyl]-N-[1-(cyclopropylamino)-5,5-difluoro-1,2-dioxopentan-3-yl]-3,3a,4,5,6,6a-hexahydro-1H-cyclopenta[c]pyrrole-3-carboxamideKi50000.0 [1]
N-(3-Chloro-benzyl)-2-(6-methyl-2-oxo-3-phenylmethanesulfonylamino-2H-pyridin-1-yl)-acetamideKi20000.0 [1]
3-[2-(5-Chlorothiophen-2-yl)-3H-benzimidazol-5-yl]-N-[2-fluoro-4-(3-oxomorpholin-4-yl)phenyl]propanamideIC5010000.0 [1]
4-(Hydroxymethyl)benzamidineKi79432.82 [1]
6-[1-[(2S)-3-(6-Chloronaphthalen-2-yl)sulfonyl-2-hydroxypropanoyl]piperidin-4-yl]-3-methyl-7H-imidazo[1,5-c]imidazol-5-oneKi60000.0 [1]
Unii-XD269G3O31Ki8000.0 [1]
3-[6-[4-[2-[(Dimethylamino)methyl]phenyl]phenyl]-7-oxo-3-(trifluoromethyl)-4,5-dihydropyrazolo[3,4-c]pyridin-1-yl]benzamideKi1800.0 [1]
N-[2-(Diaminomethylideneamino)oxyethyl]-2-[3-[(2,2-difluoro-2-phenylethyl)amino]-6-methyl-2-oxopyrazin-1-yl]acetamideKi128.0 [1]
2-(1-Aminoisoquinolin-7-yl)-5-methyl-N-[4-(2-sulfamoylphenyl)phenyl]pyrazole-3-carboxamideKi2600.0 [1]
Items per page: 1 - 10 of 100
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References

This online tool may be cited as follows

MLA

"Quest Database™ Trypsin Inhibitors (IC50, Ki)." AAT Bioquest, Inc., 10 May. 2024, https://www.aatbio.com/data-sets/trypsin-inhibitors-ic50-ki.

APA

AAT Bioquest, Inc. (2024, May 10). Quest Database™ Trypsin Inhibitors (IC50, Ki). AAT Bioquest. https://www.aatbio.com/data-sets/trypsin-inhibitors-ic50-ki.
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