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Type-1 angiotensin II receptor Inhibitors (IC50, Ki)
Structure
Compound Name
Standard Type
Standard Values (in nM)
LosartanIC500.33 [1], 8.0 [2], 28.0 [3], 88.0 [4]
LosartanKi12.0 [1], 17.0 [2]
TelmisartanIC503.0 [1], 150.0 [2]
SaralasinIC500.57 [1], 1.0 [2]
SaralasinKi0.22 [1], 0.33 [2]

References
This online resource may be cited as follows
MLA
"Quest DatabaseType-1 angiotensin II receptor Inhibitors (IC50, Ki)." AAT Bioquest, Inc.4 Dec2025https://www.aatbio.com/data-sets/type-1-angiotensin-ii-receptor-inhibitors-ic50-ki.
APA
AAT Bioquest, Inc. (2025December 4). Quest DatabaseType-1 angiotensin II receptor Inhibitors (IC50, Ki). AAT Bioquest. https://www.aatbio.com/data-sets/type-1-angiotensin-ii-receptor-inhibitors-ic50-ki.
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