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Tyrosine-protein kinase ABL Inhibitors (IC50, Ki)
Structure
Compound Name
Standard Type
Standard Values (in nM)
ImatinibIC50234.0 [1]
ImatinibKi13.0 [1], 37.0 [2], 7000.0 [3]
PonatinibIC501.08 [1]
DasatinibIC501.0 [1]
NilotinibIC5028.0 [1]

References
This online resource may be cited as follows
MLA
"Quest DatabaseTyrosine-protein kinase ABL Inhibitors (IC50, Ki)." AAT Bioquest, Inc.5 Dec2025https://www.aatbio.com/data-sets/tyrosine-protein-kinase-abl-inhibitors-ic50-ki.
APA
AAT Bioquest, Inc. (2025December 5). Quest DatabaseTyrosine-protein kinase ABL Inhibitors (IC50, Ki). AAT Bioquest. https://www.aatbio.com/data-sets/tyrosine-protein-kinase-abl-inhibitors-ic50-ki.
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