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Tyrosine-protein kinase BLK Inhibitors (IC50, Ki)
Structure
Compound Name
Standard Type
Standard Values (in nM)
IbrutinibIC500.5 [1]
CanertinibIC5029.0 [1], 50.0 [2]
4-[(3-Bromophenyl)amino]-6-acrylamidoquinazolineIC505470.0 [1], 10000.0 [2]
7-[cis-4-(4-Methylpiperazin-1-Yl)cyclohexyl]-5-(4-Phenoxyphenyl)-7h-Pyrrolo[2,3-D]pyrimidin-4-AmineIC5046.0 [1], 370.0 [2]
1-((2S,5R)-5-((7H-Pyrrolo[2,3-d]pyrimidin-4-yl)amino)-2-methylpiperidin-1-yl)prop-2-en-1-oneIC5019000.0 [1]

References
This online resource may be cited as follows
MLA
"Quest DatabaseTyrosine-protein kinase BLK Inhibitors (IC50, Ki)." AAT Bioquest, Inc.21 Jan2026https://www.aatbio.com/data-sets/tyrosine-protein-kinase-blk-inhibitors-ic50-ki.
APA
AAT Bioquest, Inc. (2026January 21). Quest DatabaseTyrosine-protein kinase BLK Inhibitors (IC50, Ki). AAT Bioquest. https://www.aatbio.com/data-sets/tyrosine-protein-kinase-blk-inhibitors-ic50-ki.
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