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Tyrosine-protein kinase BRK Inhibitors (IC50, Ki)
Structure
Compound Name
Standard Type
Standard Values (in nM)
StaurosporineIC50247.0 [1], 1250.0 [2]
IbrutinibIC503.3 [1]
Tyrphostin AG 808IC502320.0 [1], 53240.0 [2]
[3-Fluoro-4-[[6-methyl-3-(1H-pyrazol-4-yl)imidazo[1,2-a]pyrazin-8-yl]amino]phenyl]-piperazin-1-ylmethanoneIC5010.0 [1], 54.0 [2]
5-{[(5-Bromo-2-methoxyphenyl)methylidene]amino}-2,3-dihydro-1H-1,3-benzodiazol-2-oneIC5017110.0 [1], 100000.0 [2]

References
This online resource may be cited as follows
MLA
"Quest DatabaseTyrosine-protein kinase BRK Inhibitors (IC50, Ki)." AAT Bioquest, Inc.15 Dec2025https://www.aatbio.com/data-sets/tyrosine-protein-kinase-brk-inhibitors-ic50-ki.
APA
AAT Bioquest, Inc. (2025December 15). Quest DatabaseTyrosine-protein kinase BRK Inhibitors (IC50, Ki). AAT Bioquest. https://www.aatbio.com/data-sets/tyrosine-protein-kinase-brk-inhibitors-ic50-ki.
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