logo
Products
Technologies
Applications
Services
Resources
Selection Guides
About
Tyrosine-protein kinase BTK Inhibitors (IC50, Ki)
Structure
Compound Name
Standard Type
Standard Values (in nM)
IbrutinibIC500.5 [1]
IbrutinibKi4.8 [1]
FenebrutinibIC501.4 [1]
FenebrutinibKi0.91 [1], 1.3 [2], 1.6 [3], 3.4 [4], 12.6 [5]
7-(2-Hydroxypropan-2-yl)-4-[2-methyl-3-(4-oxoquinazolin-3-yl)phenyl]-9H-carbazole-1-carboxamideIC5026.0 [1]

References
This online resource may be cited as follows
MLA
"Quest DatabaseTyrosine-protein kinase BTK Inhibitors (IC50, Ki)." AAT Bioquest, Inc.7 Dec2025https://www.aatbio.com/data-sets/tyrosine-protein-kinase-btk-inhibitors-ic50-ki.
APA
AAT Bioquest, Inc. (2025December 7). Quest DatabaseTyrosine-protein kinase BTK Inhibitors (IC50, Ki). AAT Bioquest. https://www.aatbio.com/data-sets/tyrosine-protein-kinase-btk-inhibitors-ic50-ki.
BibTeXEndNoteRefMan