Structure | Compound Name | Standard Type | Standard Values (in nM) |
|---|---|---|---|
| Tofacitinib | IC50 | 3.2 [1] | |
| Tofacitinib | Ki | 0.68 [1], 0.7 [2] | |
| Ruxolitinib | IC50 | 3.3 [1] | |
| Ruxolitinib | Ki | 0.09 [1], 0.2 [2] | |
| Filgotinib | IC50 | 10.0 [1] | |
MLA | "Quest Database™ Tyrosine-protein kinase JAK1 Inhibitors (IC50, Ki)." AAT Bioquest, Inc., 14 Dec. 2025, https://www.aatbio.com/data-sets/tyrosine-protein-kinase-jak1-inhibitors-ic50-ki. | |
APA | AAT Bioquest, Inc. (2025, December 14). Quest Database™ Tyrosine-protein kinase JAK1 Inhibitors (IC50, Ki). AAT Bioquest. https://www.aatbio.com/data-sets/tyrosine-protein-kinase-jak1-inhibitors-ic50-ki. | |
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