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Tyrosine-protein kinase JAK1 Inhibitors (IC50, Ki)
Structure
Compound Name
Standard Type
Standard Values (in nM)
TofacitinibIC503.2 [1]
TofacitinibKi0.68 [1], 0.7 [2]
RuxolitinibIC503.3 [1]
RuxolitinibKi0.09 [1], 0.2 [2]
FilgotinibIC5010.0 [1]

References
This online resource may be cited as follows
MLA
"Quest DatabaseTyrosine-protein kinase JAK1 Inhibitors (IC50, Ki)." AAT Bioquest, Inc.14 Dec2025https://www.aatbio.com/data-sets/tyrosine-protein-kinase-jak1-inhibitors-ic50-ki.
APA
AAT Bioquest, Inc. (2025December 14). Quest DatabaseTyrosine-protein kinase JAK1 Inhibitors (IC50, Ki). AAT Bioquest. https://www.aatbio.com/data-sets/tyrosine-protein-kinase-jak1-inhibitors-ic50-ki.
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