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Tyrosine-protein kinase LCK Inhibitors (IC50, Ki)

Structure
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Compound Name
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Standard Type
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Standard Values (in nM)
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StaurosporineIC501.8 [1]
4-Amino-5-(4-Phenoxyphenyl)-7h-Pyrrolo[2,3-D]pyrimidin-7-Yl-CyclopentaneIC502.0 [1]
DasatinibIC500.4 [1], 1.0 [2], 3.0 [3], 4.0 [4]
N-(2-Chloro-6-methylphenyl)-2-[(cyclopropylcarbonyl)amino]-1,3-thiazole-5-carboxamideIC5035.0 [1], 880.0 [2]
5-(4-Phenoxyphenyl)-7-isopropyl-7H-pyrrolo[2,3-d]pyrimidine-4-amineIC501.0 [1], 10.0 [2], 11.0 [3]
5-(4-Phenoxyphenyl)-7-tert-butyl-7H-pyrrolo[2,3-d]pyrimidine-4-amineIC502.0 [1], 13.8 [2], 14.0 [3], 75.0 [4]
PiceatannolIC505000.0 [1], 66000.0 [2], 82000.0 [3]
DoramapimodIC501000.0 [1], 2100.0 [2], 20000.0 [3], 35000.0 [4]
1-(Tert-Butyl)-3-(p-tolyl)-1H-pyrazolo[3,4-d]pyrimidin-4-amineIC505.0 [1], 151.0 [2], 250.0 [3]
1-(Tert-Butyl)-3-(p-tolyl)-1H-pyrazolo[3,4-d]pyrimidin-4-amineKi63.1 [1]
7-[cis-4-(4-Methylpiperazin-1-Yl)cyclohexyl]-5-(4-Phenoxyphenyl)-7h-Pyrrolo[2,3-D]pyrimidin-4-AmineIC5015.0 [1], 240.0 [2]
N-(2-Bromophenyl)imidazo[1,5-a]quinoxalin-4-amineIC50170.0 [1]
Unii-mbe6kwv0QIIC504.0 [1]
Unii-mbe6kwv0QIKi4.0 [1], 5.5 [2]
3-(2-Aminoquinazolin-6-Yl)-4-Methyl-N-[3-(Trifluoromethyl)phenyl]benzamideIC500.2 [1], 1.0 [2]
5-(3-Phenoxyphenyl)-7-cyclopentyl-7H-pyrrolo[2,3-d]pyrimidine-4-amineIC50140.0 [1], 1180.0 [2], 1200.0 [3], 10000.0 [4]
2-[4-Amino-5-(4-phenoxy-phenyl)-pyrrolo[2,3-d]pyrimidin-7-yl]-cyclopentanolIC501.0 [1], 8.0 [2], 240.0 [3], 1320.0 [4]
3-[4-Amino-5-(4-phenoxy-phenyl)-pyrrolo[2,3-d]pyrimidin-7-yl]-cyclopentanolIC501.0 [1], 5.0 [2], 544.0 [3]
4-[4-Amino-5-(4-phenoxyphenyl)pyrrolo[2,3-d]pyrimidin-7-yl]cyclopentane-1,2-diolIC502.0 [1], 5.0 [2], 23.0 [3], 317.0 [4]
2-PropenaMide, N-[cis-4-[4-aMino-3-(4-phenoxyphenyl)-1H-pyrazolo[3,4-d]pyriMidin-1-yl]cyclohexyl]-IC500.88 [1], 1.0 [2]
ImatinibIC50160.0 [1], 320.0 [2]
CrizotinibIC501.0 [1], 2741.0 [2]
1-Tert-butyl-3-(4-chlorophenyl)-1H-pyrazolo[3,4-d]pyrimidin-4-amineIC504.0 [1]
1-Tert-butyl-3-(4-chlorophenyl)-1H-pyrazolo[3,4-d]pyrimidin-4-amineKi0.79 [1]
SaracatinibIC504.0 [1]
DamnacanthalIC5017.0 [1], 620.0 [2]
Tyrphostin A46IC507000.0 [1], 22000.0 [2]
N-(2-Chloro-6-methylphenyl)-7,8-dimethoxyimidazo[1,5-a]quinoxalin-4-amineIC502.0 [1]
N-(2-Chloro-6-methylphenyl)-7-methoxyimidazo[1,5-a]quinoxalin-4-amineIC508.7 [1]
N-(2-Chloro-6-methylphenyl)-8-methoxyimidazo[1,5-a]quinoxalin-4-amineIC503.0 [1], 280.0 [2]
N-(2-Chloro-6-methylphenyl)imidazo[1,5-a]quinoxalin-4-amineIC509.0 [1]
N4-(2-Chloro-6-methylphenyl)imidazo[1,5-a]quinoxaline-4,7-diamineIC5021.0 [1]
N-(2,6-Dimethylphenyl)-6,7-dimethoxyimidazo[1,5-a]quinoxalin-4-amineIC502.4 [1]
7,8-Dihydroxyisoquinoline-3-carboxamideIC50500.0 [1]
5-Thiazolecarboxamide, 2-amino-4-methyl-N-(2,4,6-trimethylphenyl)-IC503200.0 [1], 5000.0 [2]
N-(2-Chloro-6-methylphenyl)-2-[(phenylcarbonyl)amino]-1,3-thiazole-5-carboxamideIC50890.0 [1]
N-(2,6-Dimethylphenyl)-7,8-dimethoxyimidazo[1,5-a]quinoxalin-4-amineIC502.4 [1]
N-(2-Bromophenyl)-1-methylimidazo[1,5-a]quinoxalin-4-amineIC50180.0 [1]
N-(2-Chloro-6-methylphenyl)-7-morpholinoimidazo[1,5-a]quinoxalin-4-amineIC506.0 [1]
N-(2,6-Diethylphenyl)imidazo[1,5-a]quinoxalin-4-amineIC501690.0 [1]
N-Phenylimidazo[1,5-a]quinoxalin-4-amineIC50890.0 [1]
N-(2,6-Dimethylphenyl)imidazo[1,5-a]quinoxalin-4-amineIC5016.0 [1]
N-(2-Fluorophenyl)imidazo[1,5-a]quinoxalin-4-amineIC50390.0 [1]
N-(2-Chloro-4-methylphenyl)imidazo[1,5-a]quinoxalin-4-amineIC50240.0 [1]
N-(2-Chloro-6-methylphenyl)-6-methoxyimidazo[1,5-a]quinoxalin-4-amineIC503.0 [1], 280.0 [2]
7-Bromo-N-(2-chloro-6-methylphenyl)imidazo[1,5-a]quinoxalin-4-amineIC5014.0 [1]
N-(2-Methoxyphenyl)imidazo[1,5-a]quinoxalin-4-amineIC505520.0 [1]
4-(2-Chloro-6-methylanilino)imidazo[1,5-a]quinoxaline-7-carboxamideIC5030.0 [1]
N-(2-Chlorophenyl)imidazo[1,5-a]quinoxalin-4-amineIC5060.0 [1]
N-(4-(2-Chloro-6-methylphenylamino)imidazo[1,5-a]quinoxalin-7-yl)acetamideIC5011.0 [1]
N-(2-Chlorophenyl)-3-methylimidazo[1,5-a]quinoxalin-4-amineIC5030.0 [1]
N-(2,6-Difluorophenyl)imidazo[1,5-a]quinoxalin-4-amineIC50360.0 [1]
N-(2,6-Dichlorophenyl)imidazo[1,5-a]quinoxalin-4-amineIC509.0 [1]
N-(2,6-Dimethylphenyl)-9-nitroimidazo[1,5-a]quinoxalin-4-amineIC50100.0 [1]
N-(3-Fluorophenyl)imidazo[1,5-a]quinoxalin-4-amineIC501330.0 [1]
N-Mesitylimidazo[1,5-a]quinoxalin-4-amineIC5040.0 [1]
N-(2,6-Dibromophenyl)imidazo[1,5-a]quinoxalin-4-amineIC5050.0 [1]
N-(2-Chloro-4,6-dimethylphenyl)imidazo[1,5-a]quinoxalin-4-amineIC5030.0 [1]
N4-(2-Chloro-6-methylphenyl)-N7,N7-diethylimidazo[1,5-a]quinoxaline-4,7-diamineIC509.0 [1]
2-[[(Tert-butyloxy)carbonyl]-amino]-4-methyl-N-(2,4,6-trimethylphenyl)-1,3-thiazole-5-carboxamideIC501500.0 [1], 3000.0 [2]
N-(2-Chloro-6-methylphenyl)-6,7-dimethoxyimidazo[1,5-a]quinoxalin-4-amineIC502.0 [1]
7-Hydroxy-6-oxo-2,6-dihydroisoquinoline-3-carboxamideIC501900000.0 [1]
QuercetinIC5013000.0 [1]
IbrutinibIC502.0 [1]
Rosmarinic acidIC5024000.0 [1], 55000.0 [2]
TofacitinibIC503870.0 [1]
NintedanibIC5016.0 [1]
CeritinibIC50560.0 [1], 672.0 [2]
Nvp-aew541IC505600.0 [1]
Bms-536924IC50341.0 [1]
PDGF Receptor Tyrosine Kinase Inhibitor IVIC50100.0 [1]
Amg-458IC50730.0 [1], 1000.0 [2]
JNJ-28312141 free baseIC5088.0 [1], 3900.0 [2]
A-770041IC5080.0 [1], 147.0 [2]
Lavendustin cIC5010000.0 [1]
(4S,6Z,9S,10S)-9,10,18-Trihydroxy-16-methoxy-4-methyl-3-oxabicyclo[12.4.0]octadeca-1(14),6,15,17-tetraene-2,8-dioneIC50750.0 [1], 6200.0 [2]
7-(2,6-Dichlorophenyl)-5-methyl-N-[4-(2-pyrrolidin-1-ylethoxy)phenyl]-1,2,4-benzotriazin-3-amineKi29.4 [1]
Aim-100IC50122.0 [1]
AminogenisteinIC501000.0 [1], 1200.0 [2]
N-(4-Chlorophenyl)-6-[(6,7-dimethoxyquinolin-4-yl)oxy]naphthalene-1-carboxamideIC5038.0 [1]
Bms-986142IC5071.0 [1], 3800.0 [2]
N-Acetyl-O-phosphono-Tyr-Glu-Glu-Ile-GluIC501300.0 [1], 1500.0 [2]
N-[1-[(3-Fluorophenyl)methyl]indazol-5-yl]-5-[[(2S)-morpholin-2-yl]methoxymethyl]pyrrolo[2,1-f][1,2,4]triazin-4-amineIC505000.0 [1]
9H-Imidazo(4,5-H)isoquinolin-9-one, 2-((2,6-dichlorophenyl)amino)-1,8-dihydro-6,7-dimethyl-IC5026.0 [1], 110.0 [2]
4-N-(2-Chloro-6-methylphenyl)-7-N-[2-(dimethylamino)ethyl]-8-methoxyimidazo[1,5-a]quinoxaline-4,7-diamineIC501.7 [1]
Lck InhibitorIC507.0 [1], 1600.0 [2]
4'-Amino-7-hydroxyflavoneIC50100000.0 [1], 138000.0 [2]
N-(2-Chloro-6-methylphenyl)-8-fluoroimidazo[1,5-a]quinoxalin-4-amineIC5026.0 [1]
2-Methyl-N-pyrimidin-5-yl-5-[[3-(trifluoromethyl)benzoyl]amino]benzamideIC50239.0 [1], 240.0 [2]
N4-(2-Chloro-6-methylphenyl)imidazo[1,5-a]quinoxaline-4,8-diamineIC507.0 [1]
6-[4-[2-(Dimethylamino)ethoxy]phenyl]-N-[[(2S)-oxolan-2-yl]methyl]-5-phenylfuro[2,3-d]pyrimidin-4-amineIC506.0 [1]
Pyrazolo[3,4-d]pyrimidine 5IC5093.0 [1]
cis-3-[4-Amino-7-(3-azetidin-1-ylmethyl-cyclobutyl)-7H-pyrrolo[2,3-d]pyrimidin-5-yl]-phenolIC50690.0 [1]
7-[3-(Azetidin-1-ylmethyl)cyclobutyl]-5-[3-[[(2S)-oxolan-2-yl]methoxy]phenyl]pyrrolo[2,3-d]pyrimidin-4-amineIC508900.0 [1]
2-[[(Tert-butyloxy)carbonyl]-amino]-4-methyl-N-(2-chloro-6-methylphenyl)-1,3-thiazole-5-carboxamideIC5028000.0 [1]
4-Methyl-3-(3-(pyrimidin-4-yl)pyridin-2-ylamino)-N-(3-(trifluoromethyl)phenyl)benzamideIC503.5 [1], 25.0 [2]
(NE)-N-[[4-(2-chloro-6-methylanilino)-6,7-dimethoxyimidazo[1,5-a]quinoxalin-1-yl]methylidene]hydroxylamineIC504.3 [1]
N-(2-Amino-5-pyrimidinyl)-2-methyl-5-(((3-(trifluoromethyl)phenyl)carbonyl)amino)benzamideIC5014.0 [1], 149.0 [2]
4-Methyl-3-[2-(methylamino)quinazolin-6-yl]-N-[3-(trifluoromethyl)phenyl]benzamideIC500.27 [1], 0.3 [2]
4'-AminoflavoneIC50200000.0 [1], 210000.0 [2]
Items per page: 1 - 10 of 100
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References

This online tool may be cited as follows

MLA

"Quest Database™ Tyrosine-protein kinase LCK Inhibitors (IC50, Ki)." AAT Bioquest, Inc., 9 May. 2024, https://www.aatbio.com/data-sets/tyrosine-protein-kinase-lck-inhibitors-ic50-ki.

APA

AAT Bioquest, Inc. (2024, May 9). Quest Database™ Tyrosine-protein kinase LCK Inhibitors (IC50, Ki). AAT Bioquest. https://www.aatbio.com/data-sets/tyrosine-protein-kinase-lck-inhibitors-ic50-ki.
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