Structure | Compound Name | Standard Type | Standard Values (in nM) |
|---|---|---|---|
| Cabozantinib | IC50 | 10.1 [1] | |
| 3-(2-Phenylethynyl)-1-propan-2-ylpyrazolo[3,4-d]pyrimidin-4-amine | IC50 | 56.5 [1] | |
| 3-(5-Cyclopropyl-1,2-oxazol-3-yl)-1-propan-2-ylpyrazolo[3,4-d]pyrimidin-4-amine | IC50 | 4.0 [1] | |
| N-(5-Tert-butyl-1,2-oxazol-3-yl)-2-(4-imidazo[1,2-a]pyridin-6-ylphenyl)acetamide | IC50 | 250.0 [1] | |
| Vandetanib | IC50 | 49.0 [1], 97.0 [2], 100.0 [3], 102.0 [4], 950.0 [5] | |
MLA | "Quest Database™ Tyrosine-protein kinase receptor RET Inhibitors (IC50, Ki)." AAT Bioquest, Inc., 15 Dec. 2025, https://www.aatbio.com/data-sets/tyrosine-protein-kinase-receptor-ret-inhibitors-ic50-ki. | |
APA | AAT Bioquest, Inc. (2025, December 15). Quest Database™ Tyrosine-protein kinase receptor RET Inhibitors (IC50, Ki). AAT Bioquest. https://www.aatbio.com/data-sets/tyrosine-protein-kinase-receptor-ret-inhibitors-ic50-ki. | |
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