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Tyrosine-protein kinase receptor RET Inhibitors (IC50, Ki)
Structure
Compound Name
Standard Type
Standard Values (in nM)
CabozantinibIC5010.1 [1]
3-(2-Phenylethynyl)-1-propan-2-ylpyrazolo[3,4-d]pyrimidin-4-amineIC5056.5 [1]
3-(5-Cyclopropyl-1,2-oxazol-3-yl)-1-propan-2-ylpyrazolo[3,4-d]pyrimidin-4-amineIC504.0 [1]
N-(5-Tert-butyl-1,2-oxazol-3-yl)-2-(4-imidazo[1,2-a]pyridin-6-ylphenyl)acetamideIC50250.0 [1]
VandetanibIC5049.0 [1], 97.0 [2], 100.0 [3], 102.0 [4], 950.0 [5]

References
This online resource may be cited as follows
MLA
"Quest DatabaseTyrosine-protein kinase receptor RET Inhibitors (IC50, Ki)." AAT Bioquest, Inc.15 Dec2025https://www.aatbio.com/data-sets/tyrosine-protein-kinase-receptor-ret-inhibitors-ic50-ki.
APA
AAT Bioquest, Inc. (2025December 15). Quest DatabaseTyrosine-protein kinase receptor RET Inhibitors (IC50, Ki). AAT Bioquest. https://www.aatbio.com/data-sets/tyrosine-protein-kinase-receptor-ret-inhibitors-ic50-ki.
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