Structure | Compound Name | Standard Type | Standard Values (in nM) |
|---|---|---|---|
| Tofacitinib | IC50 | 34.0 [1] | |
| Tofacitinib | Ki | 4.39 [1], 7.3 [2], 7.8 [3] | |
| Ruxolitinib | IC50 | 19.0 [1] | |
| Ruxolitinib | Ki | 0.5 [1], 0.55 [2] | |
| Pyridone 6 | IC50 | 1.0 [1], 5.0 [2], 1700.0 [3] | |
MLA | "Quest Database™ Tyrosine-protein kinase TYK2 Inhibitors (IC50, Ki)." AAT Bioquest, Inc., 28 Dec. 2025, https://www.aatbio.com/data-sets/tyrosine-protein-kinase-tyk2-inhibitors-ic50-ki. | |
APA | AAT Bioquest, Inc. (2025, December 28). Quest Database™ Tyrosine-protein kinase TYK2 Inhibitors (IC50, Ki). AAT Bioquest. https://www.aatbio.com/data-sets/tyrosine-protein-kinase-tyk2-inhibitors-ic50-ki. | |
| BibTeX | EndNote | RefMan |