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Tyrosine-protein kinase TYK2 Inhibitors (IC50, Ki)
Structure
Compound Name
Standard Type
Standard Values (in nM)
TofacitinibIC5034.0 [1]
TofacitinibKi4.39 [1], 7.3 [2], 7.8 [3]
RuxolitinibIC5019.0 [1]
RuxolitinibKi0.5 [1], 0.55 [2]
Pyridone 6IC501.0 [1], 5.0 [2], 1700.0 [3]

References
This online resource may be cited as follows
MLA
"Quest DatabaseTyrosine-protein kinase TYK2 Inhibitors (IC50, Ki)." AAT Bioquest, Inc.28 Dec2025https://www.aatbio.com/data-sets/tyrosine-protein-kinase-tyk2-inhibitors-ic50-ki.
APA
AAT Bioquest, Inc. (2025December 28). Quest DatabaseTyrosine-protein kinase TYK2 Inhibitors (IC50, Ki). AAT Bioquest. https://www.aatbio.com/data-sets/tyrosine-protein-kinase-tyk2-inhibitors-ic50-ki.
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