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Vasopressin V1 receptor Inhibitors (IC50, Ki)

Structure
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Compound Name
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Standard Type
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Standard Values (in nM)
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MozavaptanIC502000.0 [1]
1-(1-(4-(3-Acetylaminopropoxy)benzoyl)-4-piperidyl)-3,4-dihydro-2(1H)-quinolinoneIC50440.0 [1]
2-[4-[4-(7-(111C)Methoxynaphthalen-1-yl)piperazin-1-yl]butyl]-4-methyl-1,2,4-triazine-3,5-dioneKi10000.0 [1]
N-[2-[4-[4-(Dimethylamino)piperidin-1-yl]-4-oxobutoxy]-4-(5,6,7,8-tetrahydrothieno[3,2-b]azepine-4-carbonyl)phenyl]-2-phenylbenzamideIC503.0 [1]
N-[4-[8-[2-(Dimethylamino)ethyl]-6,7-dihydro-5H-thieno[2,3-b][1,4]diazepine-4-carbonyl]phenyl]-2-phenylbenzamideIC50400.0 [1]
2-Phenyl-N-[4-[8-(pyridin-3-ylmethyl)-6,7-dihydro-5H-thieno[2,3-b][1,4]diazepine-4-carbonyl]phenyl]benzamideIC50700.0 [1]
N-[4-[8-[2-(4-Methyl-1,4-diazepan-1-yl)acetyl]-6,7-dihydro-5H-thieno[2,3-b][1,4]diazepine-4-carbonyl]phenyl]-2-phenylbenzamideIC5010000.0 [1]
N-[4-(8-Benzyl-6,7-dihydro-5H-thieno[2,3-b][1,4]diazepine-4-carbonyl)phenyl]-2-phenylbenzamideIC50400.0 [1]
N-[4-[8-[2-(4-Methylpiperazin-1-yl)ethyl]-6,7-dihydro-5H-thieno[2,3-b][1,4]diazepine-4-carbonyl]phenyl]-2-phenylbenzamideIC501000.0 [1]
N-[2-[4-[4-(Diethylamino)piperidin-1-yl]-4-oxobutoxy]-4-(5,6,7,8-tetrahydrothieno[3,2-b]azepine-4-carbonyl)phenyl]-2-phenylbenzamideIC504.0 [1]
N-[4-[8-(Dimethylamino)-5,6,7,8-tetrahydrothieno[3,2-b]azepine-4-carbonyl]phenyl]-2-phenylbenzamideIC502000.0 [1]
N-[3-Methoxy-4-(5,6,7,8-tetrahydrothieno[3,2-b]azepine-4-carbonyl)phenyl]-2-phenylbenzamideIC50490.0 [1]
N-[2-[4-Oxo-4-(4-piperidin-1-ylpiperidin-1-yl)butoxy]-4-(5,6,7,8-tetrahydrothieno[3,2-b]azepine-4-carbonyl)phenyl]-2-phenylbenzamideIC5010.0 [1]
N-[2-[4-[2-(Dimethylamino)ethyl-methylamino]butoxy]-4-(5,6,7,8-tetrahydrothieno[3,2-b]azepine-4-carbonyl)phenyl]-2-phenylbenzamideIC505.0 [1]
2-Methyl-N-[4-(5,6,7,8-tetrahydrothieno[3,2-b]azepine-4-carbonyl)phenyl]benzamideIC504000.0 [1]
2-Phenyl-N-[4-(5,6,7,8-tetrahydro-1H-pyrrolo[3,2-b]azepine-4-carbonyl)phenyl]benzamideIC502100.0 [1]
2-Phenyl-N-[4-[8-(2-pyrrolidin-1-ylethyl)-6,7-dihydro-5H-thieno[2,3-b][1,4]diazepine-4-carbonyl]phenyl]benzamideIC50800.0 [1]
N-[2-Methoxy-4-(5,6,7,8-tetrahydrothieno[3,2-b]azepine-4-carbonyl)phenyl]-2-phenylbenzamideIC5050.0 [1]
N-[4-(1-Methyl-5,6,7,8-tetrahydropyrrolo[3,2-b]azepine-4-carbonyl)phenyl]-2-phenylbenzamideIC50210.0 [1]
N-[4-[8-[Methyl(2-pyridin-3-ylethyl)amino]-5,6,7,8-tetrahydrothieno[3,2-b]azepine-4-carbonyl]phenyl]-2-phenylbenzamideIC502200.0 [1]
N-[4-[8-(Dimethylamino)-5,6,7,8-tetrahydrothieno[3,2-b]azepine-4-carbonyl]-2-methoxyphenyl]-2-phenylbenzamideIC503000.0 [1]
N-[2-Hydroxy-4-(5,6,7,8-tetrahydrothieno[3,2-b]azepine-4-carbonyl)phenyl]-2-phenylbenzamideIC5060.0 [1]
2-Chloro-N-[4-(5,6,7,8-tetrahydrothieno[3,2-b]azepine-4-carbonyl)phenyl]benzamideIC50290.0 [1]
N-[2-[2-[4-(Dimethylamino)piperidin-1-yl]-2-oxoethoxy]-4-(5,6,7,8-tetrahydrothieno[3,2-b]azepine-4-carbonyl)phenyl]-2-phenylbenzamideIC5050.0 [1]
2-Phenyl-N-[4-(5,6,7,8-tetrahydrofuro[3,2-b]azepine-4-carbonyl)phenyl]benzamideIC502900.0 [1]
N-[2-[4-(4-Methylpiperazin-1-yl)butoxy]-4-(5,6,7,8-tetrahydrothieno[3,2-b]azepine-4-carbonyl)phenyl]-2-phenylbenzamideIC505.0 [1]
N-[2-[4-(4-Methylpiperazin-1-yl)-4-oxobutoxy]-4-(5,6,7,8-tetrahydrothieno[3,2-b]azepine-4-carbonyl)phenyl]-2-phenylbenzamideIC5010.0 [1]
N-[2-[4-(4-Methyl-1,4-diazepan-1-yl)-4-oxobutoxy]-4-(5,6,7,8-tetrahydrothieno[3,2-b]azepine-4-carbonyl)phenyl]-2-phenylbenzamideIC5050.0 [1]
2-Phenyl-N-[4-(5,6,7,8-tetrahydrothieno[3,2-b]azepine-4-carbonyl)phenyl]benzamideIC50300.0 [1]
N-[4-[8-(Dimethylamino)-5,6,7,8-tetrahydrothieno[3,2-b]azepine-4-carbonyl]phenyl]-2-methylbenzamideIC50780.0 [1]
N-[2-[3-(4-Methyl-1,4-diazepan-1-yl)propoxy]-4-(5,6,7,8-tetrahydrothieno[3,2-b]azepine-4-carbonyl)phenyl]-2-phenylbenzamideIC501.0 [1]
N-[1-Hydroxy-3-[4-[4-(2-oxo-3,4-dihydroquinolin-1-yl)piperidine-1-carbonyl]phenoxy]propyl]acetamideIC50600.0 [1]
N-[1-Hydroxy-3-[4-[4-(2-oxoquinolin-1-yl)piperidine-1-carbonyl]phenoxy]propyl]acetamideIC503300.0 [1]
Items per page: 1 - 10 of 33
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References

This online tool may be cited as follows

MLA

"Quest Database™ Vasopressin V1 receptor Inhibitors (IC50, Ki)." AAT Bioquest, Inc., 9 May. 2024, https://www.aatbio.com/data-sets/vasopressin-v1-receptor-inhibitors-ic50-ki.

APA

AAT Bioquest, Inc. (2024, May 9). Quest Database™ Vasopressin V1 receptor Inhibitors (IC50, Ki). AAT Bioquest. https://www.aatbio.com/data-sets/vasopressin-v1-receptor-inhibitors-ic50-ki.
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