Structure | Compound Name | Standard Type | Standard Values (in nM) |
|---|---|---|---|
| Argipressin | Ki | 1.13 [1] | |
| Lixivaptan | IC50 | 150.0 [1], 180.0 [2], 230.0 [3], 5000.0 [4] | |
| Lixivaptan | Ki | 44.0 [1], 6000.0 [2] | |
| Relcovaptan | IC50 | 13.0 [1] | |
| Relcovaptan | Ki | 0.19 [1], 0.52 [2], 0.7 [3], 0.85 [4], 1.48 [5] | |
MLA | "Quest Database™ Vasopressin V1a receptor Inhibitors (IC50, Ki)." AAT Bioquest, Inc., 4 Dec. 2025, https://www.aatbio.com/data-sets/vasopressin-v1a-receptor-inhibitors-ic50-ki. | |
APA | AAT Bioquest, Inc. (2025, December 4). Quest Database™ Vasopressin V1a receptor Inhibitors (IC50, Ki). AAT Bioquest. https://www.aatbio.com/data-sets/vasopressin-v1a-receptor-inhibitors-ic50-ki. | |
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