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Vasopressin V1a receptor Inhibitors (IC50, Ki)
Structure
Compound Name
Standard Type
Standard Values (in nM)
ArgipressinKi1.13 [1]
LixivaptanIC50150.0 [1], 180.0 [2], 230.0 [3], 5000.0 [4]
LixivaptanKi44.0 [1], 6000.0 [2]
RelcovaptanIC5013.0 [1]
RelcovaptanKi0.19 [1], 0.52 [2], 0.7 [3], 0.85 [4], 1.48 [5]

References
This online resource may be cited as follows
MLA
"Quest DatabaseVasopressin V1a receptor Inhibitors (IC50, Ki)." AAT Bioquest, Inc.4 Dec2025https://www.aatbio.com/data-sets/vasopressin-v1a-receptor-inhibitors-ic50-ki.
APA
AAT Bioquest, Inc. (2025December 4). Quest DatabaseVasopressin V1a receptor Inhibitors (IC50, Ki). AAT Bioquest. https://www.aatbio.com/data-sets/vasopressin-v1a-receptor-inhibitors-ic50-ki.
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