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Vasopressin V2 receptor Inhibitors (IC50, Ki)
StructureCompound NameStandard TypeStandard Values (in nM)
LixivaptanIC501.0 [1], 1.2 [2], 5.0 [3], 91.0 [4]
LixivaptanKi2.3 [1], 23.0 [2], 90.0 [3]
ArgipressinIC50242.0 [1]
ArgipressinKi1.2 [1], 1.36 [2], 1.48 [3], 32.0 [4]
Way-vna-932IC5080.0 [1], 80.3 [2]

References
This online resource may be cited as follows
MLA
"Quest DatabaseVasopressin V2 receptor Inhibitors (IC50, Ki)." AAT Bioquest, Inc.11 Oct2025https://www.aatbio.com/data-sets/vasopressin-v2-receptor-inhibitors-ic50-ki.
APA
AAT Bioquest, Inc. (2025October 11). Quest DatabaseVasopressin V2 receptor Inhibitors (IC50, Ki). AAT Bioquest. https://www.aatbio.com/data-sets/vasopressin-v2-receptor-inhibitors-ic50-ki.
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