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Vitamin D receptor Inhibitors (IC50, Ki)

Structure
▲
▼
Compound Name
▲
▼
Standard Type
▲
▼
Standard Values (in nM)
▲
▼
CalcitriolIC501.24 [1], 6430.0 [2]
4-Chloro-N-[(2-chlorophenyl)-(2-methyl-1H-indol-3-yl)methyl]anilineIC5036800.0 [1]
(2S)-8-Amino-4-(3-methylbutyl)-7-(2-methylprop-1-enyl)-2-(2-methylpropyl)-2,5-dihydro-1H-1,4-benzodiazepin-3-oneIC5017000.0 [1], 20000.0 [2], 23000.0 [3], 26000.0 [4]
N-[(4-Methoxyphenyl)-(2-methyl-1H-indol-3-yl)methyl]-4-(trifluoromethyl)anilineIC50590.0 [1], 8100.0 [2], 12400.0 [3]
Deoxycholic acidIC5050000.0 [1], 150000.0 [2]
Ursodeoxycholic acidIC5050000.0 [1], 150000.0 [2]
Chenodeoxycholic acidIC5050000.0 [1], 150000.0 [2]
Cholic acidIC50150000.0 [1]
Lithocholic acidIC5013600.0 [1], 46700.0 [2]
Taurolithocholic acidIC5014500.0 [1], 50000.0 [2]
Hyodeoxycholic acidIC5050000.0 [1], 150000.0 [2]
Glycolithocholic acidIC5040100.0 [1], 50000.0 [2]
Sulfolithocholic acidIC5023300.0 [1], 50000.0 [2]
Calcitroic acidIC502290.0 [1], 100000.0 [2]
Lithocholic acid glucuronideIC5031500.0 [1], 150000.0 [2]
(3beta,5beta,9beta)-3-(Acetyloxy)cholan-24-Oic AcidIC5011000.0 [1], 50000.0 [2]
Methyl lithocholateIC5015100.0 [1], 150000.0 [2]
(1,3-Dioxoisoindol-2-yl) 4-ethylbenzenesulfonateIC5010500.0 [1], 10600.0 [2]
(5S)-5-[(2R)-2-[(1R,3As,4E,7aR)-4-[2-[(3R,5R)-3,5-dihydroxy-4-methylidenecyclohexylidene]ethylidene]-7a-methyl-2,3,3a,5,6,7-hexahydro-1H-inden-1-yl]propyl]-3-methylideneoxolan-2-oneIC50300.0 [1]
1-Ethyl-5-[3-[4-(2-hydroxy-3,3-dimethylbutoxy)-3-methylphenyl]pentan-3-yl]-N-[(2S)-1-hydroxypropan-2-yl]pyrrole-2-carboxamideIC50115.3 [1], 4300.0 [2]
(5R)-5-[(2R)-2-[(1R,3As,4E,7aR)-4-[2-[(3R,5R)-3,5-dihydroxy-4-methylidenecyclohexylidene]ethylidene]-7a-methyl-2,3,3a,5,6,7-hexahydro-1H-inden-1-yl]propyl]-3-methylideneoxolan-2-oneIC50300.0 [1], 1000.0 [2]
(6R)-6-[(1R,3As,4E,7aR)-4-[2-[(3R,5R)-3,5-dihydroxycyclohexylidene]ethylidene]-7a-methyl-2,3,3a,5,6,7-hexahydro-1H-inden-1-yl]-N-(2-aminophenyl)heptanamideIC50185.0 [1], 248.0 [2]
Lithocholic acid 24-glucuronideIC502860.0 [1], 150000.0 [2]
(1R,3R)-5-[(2E)-2-[(1S,3As,7aS)-1-[(5S)-5-(1-adamantyl)-5-hydroxypenta-1,3-diynyl]-7a-methyl-2,3,3a,5,6,7-hexahydro-1H-inden-4-ylidene]ethylidene]-2-methylidenecyclohexane-1,3-diolIC500.09 [1], 5.0 [2]
(3R,5S)-5-[(2R)-2-[(1R,3As,4E,7aR)-4-[(2Z)-2-[(3S,5R)-3,5-dihydroxy-2-methylidenecyclohexylidene]ethylidene]-7a-methyl-2,3,3a,5,6,7-hexahydro-1H-inden-1-yl]propyl]-3-hydroxy-3-methyl-1-(2-phenylethyl)pyrrolidin-2-oneIC50220.0 [1], 3300.0 [2]
(1R,3R)-5-[(2E)-2-[(1R,3As,7aR)-1-[(E,2R,6S)-6-(1-adamantyl)-6-hydroxyhex-3-en-2-yl]-7a-methyl-2,3,3a,5,6,7-hexahydro-1H-inden-4-ylidene]ethylidene]cyclohexane-1,3-diolIC5050.0 [1], 400.0 [2]
2-[(E)-2-(4-Hydroxyphenyl)vinyl]-5-(methoxycarbonyl)-1,3,3-trimethyl-3H-indoliumIC506800.0 [1], 13800.0 [2]
(1R,3S,5Z)-5-[(2E)-2-[(1R,3As,7aR)-1-[(2R,6S)-6-(1-adamantyl)-6-hydroxyhex-4-yn-2-yl]-7a-methyl-2,3,3a,5,6,7-hexahydro-1H-inden-4-ylidene]ethylidene]-4-methylidenecyclohexane-1,3-diolIC500.09 [1], 0.24 [2]
(1R,3S,5Z)-5-[(2E)-2-[(1R,3As,7aR)-1-[(2R,6R)-6-(1-adamantyl)-6-hydroxyhex-4-yn-2-yl]-7a-methyl-2,3,3a,5,6,7-hexahydro-1H-inden-4-ylidene]ethylidene]-4-methylidenecyclohexane-1,3-diolIC501.75 [1], 3.13 [2]
(1R,3R)-5-[(2E)-2-[(1R,3As,7aR)-1-[(2R)-6-hydroxy-6,6-bis(4-hydroxyphenyl)hexan-2-yl]-7a-methyl-2,3,3a,5,6,7-hexahydro-1H-inden-4-ylidene]ethylidene]-2-methylidenecyclohexane-1,3-diolIC50520.0 [1], 800.0 [2]
(1R,3R)-5-[(2E)-2-[(1R,3As,7aR)-1-[(2R,3S)-3-[3-hydroxy-3,3-bis(4-hydroxyphenyl)propyl]heptan-2-yl]-7a-methyl-2,3,3a,5,6,7-hexahydro-1H-inden-4-ylidene]ethylidene]-2-methylidenecyclohexane-1,3-diolIC50130.0 [1], 400.0 [2]
4-[3-[4-(Benzenesulfonylmethoxy)-3-methylphenyl]pentan-3-yl]-N-[2-(diethylamino)ethyl]-1-ethylpyrrole-2-carboxamideIC50125.4 [1], 650.0 [2]
N-[2-(Diethylamino)ethyl]-1-ethyl-5-[3-[3-methyl-4-(methylsulfanylmethoxy)phenyl]pentan-3-yl]pyrrole-2-carboxamideIC5089.1 [1], 970.0 [2]
N-[(2-Methyl-1H-indol-3-yl)-phenylmethyl]anilineIC5010900.0 [1], 30200.0 [2]
4-(Benzenesulfonyl)-5-ethylsulfonyl-2-thiophen-2-yl-1,3-oxazoleIC505300.0 [1], 8100.0 [2]
4-(Benzenesulfonyl)-5-propan-2-ylsulfonyl-2-thiophen-2-yl-1,3-oxazoleIC502600.0 [1], 22300.0 [2]
4-[(4-Fluorophenyl)sulfonyl]-5-(propylsulfonyl)-2-thien-2-yl-1,3-oxazoleIC501600.0 [1], 7100.0 [2]
4-[(4-Fluorophenyl)sulfonyl]-5-(isobutylsulfonyl)-2-thien-2-yl-1,3-oxazoleIC506200.0 [1], 6900.0 [2]
N-[(2-Methyl-1H-indol-3-yl)[4-(propan-2-yl)phenyl]methyl]pyridin-2-amineIC509100.0 [1], 15300.0 [2]
4-Chloro-N-[(2-methyl-1H-indol-3-yl)(pyridin-3-yl)methyl]anilineIC503200.0 [1], 75000.0 [2]
4-Chloro-N-[(2-methyl-1H-indol-3-yl)-pyridin-4-ylmethyl]anilineIC503700.0 [1], 51500.0 [2]
5-(Methoxycarbonyl)-2-[(E)-2-(4-methoxyphenyl)vinyl]-1,3,3-trimethyl-3H-indoliumIC503300.0 [1], 6000.0 [2]
2-[(E)-2-(4-Ethoxyphenyl)vinyl]-5-(methoxycarbonyl)-1,3,3-trimethyl-3H-indoliumIC505700.0 [1], 5900.0 [2]
5-Methoxy-2-{(E)-2-[4-(methoxycarbonyl)phenyl]vinyl}-1,3,3-trimethyl-3H-indoliumIC508600.0 [1], 11500.0 [2]
5-Methoxy-2-[(E)-2-(4-methoxyphenyl)vinyl]-1,3,3-trimethyl-3H-indoliumIC503900.0 [1], 5500.0 [2]
8-Amino-2,7-diisobutyl-4-isopentyl-4,5-dihydro-1H-benzo[e][1,4]diazepin-3(2H)-oneIC5030000.0 [1]
N-[(2-Methyl-1H-indol-3-yl)-(4-methylphenyl)methyl]anilineIC5014600.0 [1], 43600.0 [2]
3-[4-[Anilino-(2-methyl-1H-indol-3-yl)methyl]phenyl]propan-1-olIC5013100.0 [1], 58600.0 [2]
N-[(2-Chlorophenyl)-(2-methyl-1H-indol-3-yl)methyl]-4-methoxyanilineIC505800.0 [1], 26500.0 [2]
N-[(2-Chlorophenyl)-(2-methyl-1H-indol-3-yl)methyl]-2-methoxyanilineIC508600.0 [1], 24300.0 [2]
N-[(2-Methyl-1H-indol-3-yl)-(4-nitrophenyl)methyl]anilineIC5012200.0 [1], 28500.0 [2]
N-[(2-Chlorophenyl)-(2-methyl-1H-indol-3-yl)methyl]anilineIC508500.0 [1], 29800.0 [2]
N-[(4-Chlorophenyl)-(2-methyl-1H-indol-3-yl)methyl]anilineIC508100.0 [1], 31700.0 [2]
N-[1-(2-Methyl-1H-indol-3-yl)ethyl]anilineIC5020100.0 [1], 104800.0 [2]
N-[(2-Methyl-1H-indol-3-yl)-naphthalen-2-ylmethyl]anilineIC5015000.0 [1], 29600.0 [2]
N-[(2-Chlorophenyl)-(2-methyl-1H-indol-3-yl)methyl]-4-methylanilineIC508200.0 [1], 17700.0 [2]
N-[(2-Chlorophenyl)-(1H-indol-3-yl)methyl]anilineIC5020300.0 [1], 21600.0 [2]
N-[(4-Methoxyphenyl)-(2-methyl-1H-indol-3-yl)methyl]anilineIC5012100.0 [1], 31200.0 [2]
N-Benzyl-1-(2-chlorophenyl)-1-(2,6-dimethyl-1H-indol-3-yl)methanamineIC505800.0 [1], 59900.0 [2]
N-[(2-Chlorophenyl)-(2-methyl-1H-indol-3-yl)methyl]-2-methyl-1,3-benzothiazol-5-amineIC5015800.0 [1], 25000.0 [2]
3,4-Dimethoxy-N-[(2-methyl-1H-indol-3-yl)-(1,3-thiazol-2-yl)methyl]anilineIC508500.0 [1], 17300.0 [2]
N-[(2-Chlorophenyl)-(2-methyl-1H-indol-3-yl)methyl]-3,4-dimethylanilineIC50590.0 [1], 12800.0 [2]
3,4-Dimethoxy-N-[(4-methoxyphenyl)-(2-methyl-1H-indol-3-yl)methyl]anilineIC503200.0 [1], 11300.0 [2]
4-Chloro-N-[(2-methyl-1H-indol-3-yl)-(1,3-thiazol-2-yl)methyl]anilineIC503800.0 [1], 11900.0 [2]
3,4-Dimethoxy-N-[(2-methyl-1H-indol-3-yl)-[4-(trifluoromethyl)phenyl]methyl]anilineIC504400.0 [1], 21800.0 [2]
N-Benzyl-1-(2-chlorophenyl)-1-(2-methyl-1H-indol-3-yl)methanamineIC505400.0 [1], 7200.0 [2]
1-(2-Chlorophenyl)-1-(2,6-dimethyl-1H-indol-3-yl)-N-[[4-(trifluoromethyl)phenyl]methyl]methanamineIC509100.0 [1], 35200.0 [2]
N-[(2,6-Dimethyl-1H-indol-3-yl)-pyridin-3-ylmethyl]-2-methoxypyridin-3-amineIC505400.0 [1], 32300.0 [2]
N-[(2-Chlorophenyl)-(2,6-dimethyl-1H-indol-3-yl)methyl]-4-(trifluoromethoxy)anilineIC505000.0 [1], 17200.0 [2]
1-(2-Chlorophenyl)-1-(2,6-dimethyl-1H-indol-3-yl)-N-[(4-methylphenyl)methyl]methanamineIC503400.0 [1], 9500.0 [2]
4-Chloro-N-[(2-methoxypyridin-3-yl)-(2-methyl-1H-indol-3-yl)methyl]anilineIC5014100.0 [1], 14200.0 [2]
N-[(2-Chlorophenyl)-(2,6-dimethyl-1H-indol-3-yl)methyl]pyridin-3-amineIC506700.0 [1], 29300.0 [2]
4-Chloro-N-[1H-imidazol-2-yl-(2-methyl-1H-indol-3-yl)methyl]anilineIC506100.0 [1], 16700.0 [2]
N-[(2-Chlorophenyl)-(2-methyl-1H-indol-3-yl)methyl]-3,4-dimethoxyanilineIC503000.0 [1], 7200.0 [2]
3,4-Dimethoxy-N-[(2-methyl-1H-indol-3-yl)-[4-(trifluoromethoxy)phenyl]methyl]anilineIC502200.0 [1], 22800.0 [2]
4-Chloro-N-[(2-chlorophenyl)-(2,6-dimethyl-1H-indol-3-yl)methyl]anilineIC505200.0 [1], 15600.0 [2]
4-Chloro-N-[(2-chlorophenyl)-(6-methoxy-2-methyl-1H-indol-3-yl)methyl]anilineIC507300.0 [1], 63100.0 [2]
N-[(2-Chlorophenyl)-(2,6-dimethyl-1H-indol-3-yl)methyl]-2-methoxypyridin-3-amineIC5012200.0 [1], 101400.0 [2]
Methyl 3-[[2-(3-methoxyphenyl)-4-methyl-1,3-oxazol-5-yl]methoxy]benzoateIC505560.0 [1], 17100.0 [2]
Methyl 2-[4-[[2-(2-methoxyphenyl)-4-methyl-1,3-oxazol-5-yl]methoxy]phenyl]acetateIC503820.0 [1], 11130.0 [2]
Methyl 4-[[2-(3-methoxyphenyl)-4-methyl-1,3-oxazol-5-yl]methoxy]benzoateIC505670.0 [1], 8890.0 [2]
Methyl 3-[4-[[2-(2-methoxyphenyl)-4-methyl-1,3-oxazol-5-yl]methoxy]phenyl]propanoateIC5010100.0 [1], 13600.0 [2]
Methyl 2-[[2-(3-methoxyphenyl)-4-methyl-1,3-oxazol-5-yl]methoxy]benzoateIC506750.0 [1], 15400.0 [2]
Methyl 2-[4-[[2-(3-methoxyphenyl)-4-methyl-1,3-oxazol-5-yl]methoxy]phenyl]acetateIC50660.0 [1], 13900.0 [2]
3-[4-[[2-(3-Methoxyphenyl)-4-methyl-1,3-oxazol-5-yl]methoxy]phenyl]propanoic acidIC503350.0 [1], 26700.0 [2]
Methyl 3-[4-[[2-(3-methoxyphenyl)-4-methyl-1,3-oxazol-5-yl]methoxy]phenyl]propanoateIC502880.0 [1], 6700.0 [2]
Methyl 2-[[2-(2-methoxyphenyl)-4-methyl-1,3-oxazol-5-yl]methoxy]benzoateIC503250.0 [1], 20200.0 [2]
2-[4-[[2-(3-Methoxyphenyl)-4-methyl-1,3-oxazol-5-yl]methoxy]phenyl]acetic acidIC503600.0 [1], 27700.0 [2]
3-[[2-(3-Methoxyphenyl)-4-methyl-1,3-oxazol-5-yl]methoxy]benzoic acidIC5033140.0 [1], 33200.0 [2]
4-[[2-(3-Methoxyphenyl)-4-methyl-1,3-oxazol-5-yl]methoxy]benzoic acidIC5080000.0 [1], 100000.0 [2]
2-[[2-(3-Methoxyphenyl)-4-methyl-1,3-oxazol-5-yl]methoxy]benzoic acidIC5033000.0 [1], 40400.0 [2]
Methyl 4-[[2-(2-methoxyphenyl)-4-methyl-1,3-oxazol-5-yl]methoxy]benzoateIC504850.0 [1], 17900.0 [2]
3-[4-[[2-(2-Methoxyphenyl)-4-methyl-1,3-oxazol-5-yl]methoxy]phenyl]propanoic acidIC5080000.0 [1], 100000.0 [2]
Methyl 3-[[2-(2-methoxyphenyl)-4-methyl-1,3-oxazol-5-yl]methoxy]benzoateIC502500.0 [1], 7330.0 [2]
(23S)-1alpha-Hydroxy-25,27-didehydrovitamin D3 26,23-lactoneIC506.3 [1]
(23R)-1alpha-Hydroxy-25,27-didehydrovitamin D3 26,23-lactoneIC506.0 [1]
Unii-W3DX0X37FVIC5038.0 [1]
2,5-Dimethoxybenzenesulfonic acid (1,3-dioxo-2-isoindolyl) esterIC5037600.0 [1]
(2S)-3-[4-[3-[4-[(2R)-2-Hydroxy-3,3-dimethylbutoxy]-3-methylphenyl]pentan-3-yl]-2-methylphenoxy]propane-1,2-diolKi12.0 [1]
6-(Piperidine-1-sulfonyl)-benzothiazol-2-ylamineIC502000.0 [1]
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References

This online tool may be cited as follows

MLA

"Quest Database™ Vitamin D receptor Inhibitors (IC50, Ki)." AAT Bioquest, Inc., 9 May. 2024, https://www.aatbio.com/data-sets/vitamin-d-receptor-inhibitors-ic50-ki.

APA

AAT Bioquest, Inc. (2024, May 9). Quest Database™ Vitamin D receptor Inhibitors (IC50, Ki). AAT Bioquest. https://www.aatbio.com/data-sets/vitamin-d-receptor-inhibitors-ic50-ki.
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