 | N-Tert-butyl-8-[[[(1S,2S)-2-(3-methyl-1,2,4-oxadiazol-5-yl)cyclopropanecarbonyl]amino]methyl]-5-[3-(trifluoromethoxy)phenyl]-3,4-dihydro-1H-isoquinoline-2-carboxamide | IC50 | 800.0 [1] |
 | 1-Benzyl-5-methyl-3-(piperidin-1-ylmethyl)indole | IC50 | 3400.0 [1] |
 | 1-[(3-Chlorophenyl)methyl]-5-methyl-3-(piperidin-1-ylmethyl)indole | IC50 | 2200.0 [1] |
 | 5-Methyl-1-[(3-nitrophenyl)methyl]-3-(piperidin-1-ylmethyl)indole | IC50 | 3000.0 [1] |
 | 1-[(4-Fluorophenyl)methyl]-5-methyl-3-(piperidin-1-ylmethyl)indole | IC50 | 4800.0 [1] |
 | 5-Methyl-1-[(4-methylphenyl)methyl]-3-(piperidin-1-ylmethyl)indole | IC50 | 3600.0 [1] |
 | 1-[(4-Chlorophenyl)methyl]-5-methyl-3-(piperidin-1-ylmethyl)indole | IC50 | 3000.0 [1] |
 | 5-Methyl-1-[(2-nitrophenyl)methyl]-3-(piperidin-1-ylmethyl)indole | IC50 | 1800.0 [1] |
 | 1-(2-Methoxyphenyl)-5-(4-methoxyphenyl)-3-(2,2,6,6-tetramethyloxan-4-yl)oxypyrazole | IC50 | 9.4 [1] |
 | 1-(2-Methoxyphenyl)-5-(4-methoxyphenyl)-3-(2,2,6,6-tetramethylthian-4-yl)oxypyrazole | IC50 | 6.0 [1] |
 | 4-[1-(2-Methoxyphenyl)-5-(4-methoxyphenyl)pyrazol-3-yl]oxy-2,2,6,6-tetramethylthiane 1,1-dioxide | IC50 | 3.0 [1] |
 | 4-[1-(2-Methoxyphenyl)-5-(4-methoxyphenyl)pyrazol-3-yl]oxy-2,2,6,6-tetramethylthiane 1-oxide | IC50 | 7.6 [1] |
 | 5-(4-Chlorophenyl)-1-(2-methoxyphenyl)-3-(2,2,6,6-tetramethylthian-4-yl)oxypyrazole | IC50 | 5.9 [1] |
 | 4-[5-(4-Chlorophenyl)-1-(2-methoxyphenyl)pyrazol-3-yl]oxy-2,2,6,6-tetramethylthiane 1,1-dioxide | IC50 | 1.9 [1] |
 | 5-(4-Chlorophenyl)-1-(2-methoxyphenyl)-3-[(2,2,4,4-tetramethyloxetan-3-yl)methoxy]-1H-pyrazole | IC50 | 3.1 [1] |
 | 4-[5-(4-Chlorophenyl)-1-(2-methoxyphenyl)pyrazol-3-yl]oxy-2,2,6,6-tetramethylcyclohexan-1-one | IC50 | 9.7 [1] |
 | 4-[5-(4-Chlorophenyl)-1-(2-methoxyphenyl)pyrazol-3-yl]oxy-2,2,6,6-tetramethylcyclohexan-1-ol | IC50 | 39.0 [1] |
 | 4-[2-(2-Methoxyphenyl)-5-(2,2,6,6-tetramethyloxan-4-yl)oxypyrazol-3-yl]benzonitrile | IC50 | 7.2 [1] |
 | 4-[2-(2-Methoxyphenyl)-5-(2,2,6,6-tetramethylthian-4-yl)oxypyrazol-3-yl]benzonitrile | IC50 | 12.0 [1] |
 | 4-[2-(2-Methoxyphenyl)-5-(2,2,6,6-tetramethyl-1,1-dioxothian-4-yl)oxypyrazol-3-yl]benzonitrile | IC50 | 2.4 [1] |
 | 4-[2-(2-Methoxyphenyl)-5-(2,2,6,6-tetramethyl-1-oxothian-4-yl)oxypyrazol-3-yl]benzonitrile | IC50 | 14.0 [1] |
 | Tert-butyl 4-[5-(4-chlorophenyl)-1-(2-methoxyphenyl)pyrazol-3-yl]oxypiperidine-1-carboxylate | IC50 | 30.0 [1] |
 | 4-{[5-(4-Chlorophenyl)-1-(2-methoxyphenyl)-1H-pyrazol-3-yl]oxy}cyclohexanone | IC50 | 28.0 [1] |
 | 1-Acetyl-4-{[5-(4-chlorophenyl)-1-(2-methoxyphenyl)-1H-pyrazol-3-yl]oxy}piperidine | IC50 | 26.0 [1] |
 | 4-[5-(4-Chlorophenyl)-1-(2-methoxyphenyl)pyrazol-3-yl]oxy-N,N-dimethylpiperidine-1-carboxamide | IC50 | 14.0 [1] |
 | 4-[5-(4-Chlorophenyl)-1-(2-methoxyphenyl)pyrazol-3-yl]oxy-1-methylsulfonylpiperidine | IC50 | 15.0 [1] |
 | 5-(4-Chlorophenyl)-1-(2-methoxyphenyl)-3-(oxan-4-yloxy)pyrazole | IC50 | 15.0 [1] |
 | 5-(4-Chlorophenyl)-1-(2-methoxyphenyl)-3-(thian-4-yloxy)pyrazole | IC50 | 28.0 [1] |
 | 4-[5-(4-Chlorophenyl)-1-(2-methoxyphenyl)pyrazol-3-yl]oxy-1-(2,2,2-trifluoroethyl)piperidine | IC50 | 31.0 [1] |
 | 1-[4-[5-(4-Chlorophenyl)-1-(2-methoxyphenyl)pyrazol-3-yl]oxypiperidin-1-yl]-2,2,2-trifluoroethanone | IC50 | 31.4 [1] |
 | 4-[5-(4-Chlorophenyl)-1-(2-methoxyphenyl)pyrazol-3-yl]oxythiane 1,1-dioxide | IC50 | 30.0 [1] |
 | Tert-butyl N-[4-[5-(4-chlorophenyl)-1-(2-methoxyphenyl)pyrazol-3-yl]oxycyclohexyl]carbamate | IC50 | 62.0 [1] |
 | N-[4-[5-(4-Chlorophenyl)-1-(2-methoxyphenyl)pyrazol-3-yl]oxycyclohexyl]-2,2,2-trifluoroacetamide | IC50 | 11.0 [1] |
 | 4-[5-(4-Chlorophenyl)-1-(2-methoxyphenyl)pyrazol-3-yl]oxy-1-(trifluoromethylsulfonyl)piperidine | IC50 | 24.0 [1] |
 | 4-[5-(4-Chlorophenyl)-1-(2-methoxyphenyl)pyrazol-3-yl]oxy-1-cyclopropylsulfonylpiperidine | IC50 | 9.0 [1] |
 | 5-(4-Chlorophenyl)-3-(4,4-difluorocyclohexyl)oxy-1-(2-methoxyphenyl)pyrazole | IC50 | 41.0 [1] |
 | 5-(4-Chlorophenyl)-3-(1,4-dioxaspiro[4.5]decan-8-yloxy)-1-(2-ethylphenyl)pyrazole | IC50 | 81.0 [1] |
 | Tert-Butyl 4-{[5-(4-chlorophenyl)-1-(2-ethylphenyl)-1H-pyrazol-3-yl]oxy}piperidine-1-carboxylate | IC50 | 50.0 [1] |
 | 4-{[5-(4-Chlorophenyl)-1-(2-ethylphenyl)-1H-pyrazol-3-yl]oxy}-1-(methylsulfonyl)piperidine | IC50 | 98.5 [1] |
 | 4-[5-(4-Chlorophenyl)-1-(2-propan-2-yloxyphenyl)pyrazol-3-yl]oxy-1-methylsulfonylpiperidine | IC50 | 21.5 [1] |
 | 4-[5-(4-Chlorophenyl)-1-(2-methoxyphenyl)pyrazol-3-yl]oxy-1-propan-2-ylsulfonylpiperidine | IC50 | 36.0 [1] |
 | Tert-butyl-3-((5-(4-chlorophenyl)-1-(2-methoxyphenyl)-1H-pyrazol-3-yl)oxy)azetidine-1-carboxylate | IC50 | 67.0 [1] |
 | 5-(4-Chlorophenyl)-1-(2-methoxyphenyl)-3-(2,2,6,6-tetramethyloxan-4-yl)oxypyrazole | IC50 | 7.6 [1] |
 | 5-(4-Chlorophenyl)-1-(2-methoxyphenyl)-3-(1-propan-2-ylsulfonylazetidin-3-yl)oxypyrazole | IC50 | 36.0 [1] |
 | 5-(4-Chlorophenyl)-1-(2-methoxyphenyl)-3-(1-methylsulfonylazetidin-3-yl)oxypyrazole | IC50 | 31.0 [1] |
 | [3-[5-(4-Chlorophenyl)-1-(2-methoxyphenyl)pyrazol-3-yl]oxyazetidin-1-yl]-phenylmethanone | IC50 | 85.0 [1] |
 | 4-[5-(4-Chlorophenyl)-1-(2-propan-2-yloxyphenyl)pyrazol-3-yl]oxy-1-propan-2-ylsulfonylpiperidine | IC50 | 7.0 [1] |
 | 3-[5-(4-Chlorophenyl)-1-(2-methoxyphenyl)pyrazol-3-yl]oxy-N-methoxy-N-methylazetidine-1-carboxamide | IC50 | 14.0 [1] |
 | 4-[3-[5-(4-Chlorophenyl)-1-(2-methoxyphenyl)pyrazol-3-yl]oxyazetidin-1-yl]sulfonyl-3,5-dimethyl-1,2-oxazole | IC50 | 8.0 [1] |
 | 4-[5-(4-Chlorophenyl)-1-(2-methoxyphenyl)pyrazol-3-yl]oxycyclohexan-1-amine | IC50 | 400.0 [1] |
 | 4-[5-(4-Chlorophenyl)-1-(2-methoxyphenyl)pyrazol-3-yl]oxy-2,2,6,6-tetramethylthiane 1-oxide | IC50 | 1.5 [1] |
Calculator
