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Voltage-gated potassium channel subfamily A member 1/beta-1 Inhibitors (IC50, Ki)

Structure
Compound Name
Standard Type
Standard Values (in nM)
N-Benzyl-7-[(4-methylphenyl)sulfonylcarbamoylamino]-1,2,4,5-tetrahydro-3-benzazepine-3-carboxamideIC5050000.0 [1]
N-(4-Methylphenyl)sulfonyl-5-[(4-methylphenyl)sulfonylcarbamoylamino]-1,3-dihydroisoindole-2-carboxamideIC5016000.0 [1]
N-(4-Methylphenyl)sulfonyl-6-[(4-methylphenyl)sulfonylcarbamoylamino]-3,4-dihydro-1H-isoquinoline-2-carboxamideIC5030000.0 [1]
N-(3-Methylphenyl)sulfonyl-7-[(3-methylphenyl)sulfonylcarbamoylamino]-1,2,4,5-tetrahydro-3-benzazepine-3-carboxamideIC5047000.0 [1]
N-(2-Chlorophenyl)sulfonyl-7-[(2-chlorophenyl)sulfonylcarbamoylamino]-1,2,4,5-tetrahydro-3-benzazepine-3-carboxamideIC50181000.0 [1]
N-(4-Chlorophenyl)sulfonyl-7-[(4-chlorophenyl)sulfonylcarbamoylamino]-1,2,4,5-tetrahydro-3-benzazepine-3-carboxamideIC5051000.0 [1]
N-(4-Fluorophenyl)sulfonyl-7-[(4-fluorophenyl)sulfonylcarbamoylamino]-1,2,4,5-tetrahydro-3-benzazepine-3-carboxamideIC50191000.0 [1]
N-(4-Methoxyphenyl)sulfonyl-7-[(4-methoxyphenyl)sulfonylcarbamoylamino]-1,2,4,5-tetrahydro-3-benzazepine-3-carboxamideIC5038000.0 [1]
N-(4-Methylphenyl)sulfonyl-7-[(4-methylphenyl)sulfonylcarbamoylamino]-1,2,4,5-tetrahydro-3-benzazepine-3-carboxamideIC5059000.0 [1]
N-(4-Methylphenyl)sulfonyl-7-[(4-methylphenyl)sulfonylamino]-1,2,4,5-tetrahydro-3-benzazepine-3-carboxamideIC5081000.0 [1]
N-(4-Methylphenyl)sulfonyl-7-[(4-phenylphenyl)sulfonylamino]-1,2,4,5-tetrahydro-3-benzazepine-3-carboxamideIC5088000.0 [1]
N-(4-Tert-butylphenyl)sulfonyl-7-[(4-tert-butylphenyl)sulfonylcarbamoylamino]-1,2,4,5-tetrahydro-3-benzazepine-3-carboxamideIC5041000.0 [1]
1-(4-Methylphenyl)sulfonyl-3-[3-(4-methylphenyl)sulfonyl-1,2,4,5-tetrahydro-3-benzazepin-7-yl]ureaIC50102000.0 [1]



References

This online tool may be cited as follows

MLA

"Quest Database™ Voltage-gated potassium channel subfamily A member 1/beta-1 Inhibitors (IC50, Ki)." AAT Bioquest, Inc.9 May2024https://www.aatbio.com/data-sets/voltage-gated-potassium-channel-subfamily-a-member-1-beta-1-inhibitors-ic50-ki.

APA

AAT Bioquest, Inc. (2024May 9). Quest Database™ Voltage-gated potassium channel subfamily A member 1/beta-1 Inhibitors (IC50, Ki). AAT Bioquest. https://www.aatbio.com/data-sets/voltage-gated-potassium-channel-subfamily-a-member-1-beta-1-inhibitors-ic50-ki.
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