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WD repeat-containing protein 5 Inhibitors (IC50, Ki)

Structure
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Compound Name
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Standard Type
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Standard Values (in nM)
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▼
HMTase Inhibitor IXIC501.7 [1], 2.4 [2], 3000.0 [3]
N-[(1R)-7-(6,7-Dihydro-5H-pyrrolo[1,2-a]imidazol-2-yl)-1,2,3,4-tetrahydronaphthalen-1-yl]-3-methoxy-4-methylbenzamideIC5020000.0 [1]
N-[(1R)-7-(6,7-Dihydro-5H-pyrrolo[1,2-a]imidazol-2-yl)-1,2,3,4-tetrahydronaphthalen-1-yl]-3-methoxy-4-methylbenzamideKi9.36 [1], 26.8 [2]
N-[(1R)-6-(6,7-Dihydro-5H-pyrrolo[1,2-a]imidazol-2-yl)-2,3-dihydro-1H-inden-1-yl]-2-methylpyridine-4-carboxamideIC5020000.0 [1]
N-[(1R)-6-(6,7-Dihydro-5H-pyrrolo[1,2-a]imidazol-2-yl)-2,3-dihydro-1H-inden-1-yl]-2-methylpyridine-4-carboxamideKi65.1 [1], 182.0 [2]
2-(3,4-Dichlorophenyl)-N-[(1R)-6-(6,7-dihydro-5H-pyrrolo[1,2-a]imidazol-2-yl)-2,3-dihydro-1H-inden-1-yl]acetamideIC509270.0 [1]
2-(3,4-Dichlorophenyl)-N-[(1R)-6-(6,7-dihydro-5H-pyrrolo[1,2-a]imidazol-2-yl)-2,3-dihydro-1H-inden-1-yl]acetamideKi2.51 [1], 2.66 [2]
N-[(1R)-6-(6,7-Dihydro-5H-pyrrolo[1,2-a]imidazol-2-yl)-2,3-dihydro-1H-inden-1-yl]-3,5-dimethoxy-4-methylbenzamideIC503200.0 [1]
N-[(1R)-6-(6,7-Dihydro-5H-pyrrolo[1,2-a]imidazol-2-yl)-2,3-dihydro-1H-inden-1-yl]-3,5-dimethoxy-4-methylbenzamideKi0.9 [1], 1.0 [2]
N-[(1R)-6-(6,7-Dihydro-5H-pyrrolo[1,2-a]imidazol-2-yl)-2,3-dihydro-1H-inden-1-yl]-2-(3-methoxy-4-methylphenyl)acetamideIC5012000.0 [1]
N-[(1R)-6-(6,7-Dihydro-5H-pyrrolo[1,2-a]imidazol-2-yl)-2,3-dihydro-1H-inden-1-yl]-2-(3-methoxy-4-methylphenyl)acetamideKi4.94 [1], 8.37 [2]
2-Chloro-4-Fluoro-3-Methyl-N-[2-(4-Methylpiperazin-1-Yl)-5-Nitrophenyl]benzamideIC50338.2 [1], 338.6 [2]
N-[(3R,6S,9S,12R)-9-[3-(Diaminomethylideneamino)propyl]-6-ethyl-12-methyl-2,5,8,11-tetraoxo-3-phenyl-1,4,7,10-tetrazacyclohexadec-12-yl]-2-methylpropanamideIC500.9 [1]
N-Benzhydryl-1-[[(2S)-5-(diaminomethylideneamino)-2-[[2-ethyl-2-(2-methylpropanoylamino)butanoyl]amino]pentanoyl]amino]cyclopentane-1-carboxamideIC502.9 [1], 1000.0 [2]
N-[5-(4-Aminophenyl)-2-(4-methylpiperazin-1-yl)phenyl]-2-chloro-4-fluoro-3-methylbenzamideIC50206.1 [1]
2-Chloro-4-fluoro-3-methyl-N-[2-(4-methylpiperazin-1-yl)-5-phenylphenyl]-5-nitrobenzamideIC50207.2 [1]
2-Chloro-4-fluoro-3-methyl-N-[2-(4-methylpiperazin-1-yl)-5-phenylphenyl]benzamideIC50465.7 [1]
2-Chloro-4-fluoro-3-methyl-N-[2-(4-methylpiperazin-1-yl)-5-pyridin-4-ylphenyl]benzamideIC50103.9 [1]
(2S)-2-[[(2S)-2-Acetamidopropanoyl]amino]-N-[(2S,3R)-1-amino-3-hydroxy-1-oxobutan-2-yl]-5-(diaminomethylideneamino)pentanamideIC501000.0 [1]
(2S)-2-[[(2S)-2-Acetamidopropanoyl]amino]-N-[(2S,3R)-1-amino-3-hydroxy-1-oxobutan-2-yl]-5-(diaminomethylideneamino)pentanamideKi20.0 [1]
1,1'-Binaphthalene-2,2'-dicarboxylic acidIC506000.0 [1]
4-(2,3-Dihydro-imidazo[2,1-b]thiazol-6-yl)-phenolKi1000000.0 [1]
N-(3-Methoxyphenyl)-2-(4-methyl-1-piperazinyl)-5-nitrobenzamideIC5020000.0 [1]
2-(4-Ethoxyphenyl)imidazo[1,2-a]pyridineKi1000000.0 [1]
2-Phenyl-6,7-dihydro-5H-pyrrolo[1,2-a]imidazoleKi323000.0 [1]
2-(4-Methoxyphenyl)-6,7-dihydro-5H-pyrrolo[1,2-a]imidazoleKi61000.0 [1]
4-[3-[(2-Chloro-4-fluoro-3-methylbenzoyl)amino]-4-(4-methylpiperazin-1-yl)phenyl]benzoic acidIC50660.9 [1]
2-Chloro-4-fluoro-3-methyl-N-[2-(4-methylpiperazin-1-yl)-5-pyrimidin-5-ylphenyl]benzamideIC50733.3 [1]
2-Chloro-4-fluoro-3-methyl-N-[2-(4-methylpiperazin-1-yl)-5-(4-nitrophenyl)phenyl]benzamideIC50127.4 [1]
2,4,6-Trimethoxy-N-[2-(4-methylpiperazin-1-yl)-5-nitrophenyl]benzenesulfonamideIC5020000.0 [1]
N-(2-Chloro-4-fluoro-3-methylphenyl)-2-(4-methylpiperazin-1-yl)-5-nitrobenzamideIC5011400.0 [1]
N-(2-Chlorophenyl)-2-(4-methylpiperazin-1-yl)-5-nitrobenzamideIC5020000.0 [1]
2-Chloro-4-fluoro-3-methyl-N-[2-(4-methylpiperazin-1-yl)-5-nitrophenyl]-5-nitrobenzamideIC50130.0 [1]
4-[4-[(2-Chloro-4-fluoro-3-methylbenzoyl)amino]-3-(4-methylpiperazin-1-yl)phenyl]benzoic acidIC5020000.0 [1]
N-[5-Amino-2-(4-methylpiperazin-1-yl)phenyl]-2-chloro-4-fluoro-3-methylbenzamideIC5020000.0 [1]
3-[3-[(2-Chloro-4-fluoro-3-methylbenzoyl)amino]-4-(4-methylpiperazin-1-yl)phenyl]benzoic acidIC501604.0 [1]
2-Chloro-N-[5-(4-cyanophenyl)-2-(4-methylpiperazin-1-yl)phenyl]-4-fluoro-3-methylbenzamideIC50198.5 [1]
2-Chloro-4-fluoro-N-[5-(4-fluorophenyl)-2-(4-methylpiperazin-1-yl)phenyl]-3-methylbenzamideIC50392.6 [1]
2-Chloro-4-fluoro-3-methyl-N-[2-(4-methylpiperazin-1-yl)-4-pyridin-4-ylphenyl]benzamideIC5020000.0 [1]
2-Chloro-4-fluoro-3-methyl-N-[2-(4-methylpiperazin-1-yl)-4-(4-nitrophenyl)phenyl]benzamideIC5020000.0 [1]
N-[4-(4-Aminophenyl)-2-(4-methylpiperazin-1-yl)phenyl]-2-chloro-4-fluoro-3-methylbenzamideIC5020000.0 [1]
4-Fluoro-N-[2-(4-methylpiperazin-1-yl)-5-nitrophenyl]benzenesulfonamideIC5020000.0 [1]
4-Methoxy-N-[2-(4-methylpiperazin-1-yl)-5-nitrophenyl]benzenesulfonamideIC5020000.0 [1]
3,4-Dimethoxy-N-[2-(4-methylpiperazin-1-yl)-5-nitrophenyl]benzenesulfonamideIC5020000.0 [1]
Methyl 3-[(5-amino-2-chloro-4-fluoro-3-methylbenzoyl)amino]-4-(4-methylpiperazin-1-yl)benzoateIC5046.5 [1]
Phenyl 3-[(5-amino-2-chloro-4-fluoro-3-methylbenzoyl)amino]-4-(4-methylpiperazin-1-yl)benzoateIC5026.4 [1]
2-Chloro-4-fluoro-3-methyl-N-[5-nitro-2-(4-pyridin-2-ylpiperazin-1-yl)phenyl]benzamideIC5020000.0 [1]
5-Amino-2-chloro-4-fluoro-3-methyl-N-[2-(4-methylpiperazin-1-yl)-5-[4-(propanoylamino)phenyl]phenyl]benzamideIC5081.5 [1]
5-Amino-2-chloro-N-[5-[4-(cyclohexanecarbonylamino)phenyl]-2-(4-methylpiperazin-1-yl)phenyl]-4-fluoro-3-methylbenzamideIC50340.8 [1]
3-Amino-N-[5-(4-aminophenyl)-2-(4-methylpiperazin-1-yl)phenyl]-4-fluorobenzamideIC5013600.0 [1]
N-[5-(4-Acetamidophenyl)-2-(4-methylpiperazin-1-yl)phenyl]-5-amino-2-chloro-4-fluoro-3-methylbenzamideIC5070.1 [1]
2-Chloro-4-fluoro-N-[2-[4-(4-methoxyphenyl)piperazin-1-yl]-5-nitrophenyl]-3-methylbenzamideIC5020000.0 [1]
Tert-butyl N-[3-[4-[3-[(5-amino-2-chloro-4-fluoro-3-methylbenzoyl)amino]-4-(4-methylpiperazin-1-yl)phenyl]anilino]-3-oxopropyl]carbamateIC50102.1 [1]
3-Amino-4-fluoro-N-[2-(4-methylpiperazin-1-yl)-5-pyridin-4-ylphenyl]benzamideIC505800.0 [1]
4-Fluoro-N-[2-(4-methylpiperazin-1-yl)-5-pyridin-4-ylphenyl]-3-nitrobenzamideIC50197.6 [1]
3-Amino-N-[5-(4-aminophenyl)-2-(4-methylpiperazin-1-yl)phenyl]benzamideIC5020000.0 [1]
5-Amino-2-chloro-4-fluoro-3-methyl-N-[2-(4-methylpiperazin-1-yl)-5-phenylphenyl]benzamideIC5047.9 [1]
N-[2-(4-Methylpiperazin-1-yl)-5-(4-nitrophenyl)phenyl]-3-nitrobenzamideIC50285.1 [1]
5-Amino-2-chloro-4-fluoro-3-methyl-N-[5-[4-(3-methylbutanoylamino)phenyl]-2-(4-methylpiperazin-1-yl)phenyl]benzamideIC50104.6 [1]
5-Acetamido-2-chloro-4-fluoro-3-methyl-N-[2-(4-methylpiperazin-1-yl)-5-pyridin-4-ylphenyl]benzamideIC501363.0 [1]
2-Chloro-4-fluoro-3-methyl-N-[2-(4-methylpiperazin-1-yl)-5-pyridin-4-ylphenyl]-5-nitrobenzamideIC5077.1 [1]
2-Chloro-4-fluoro-N-[2-[4-(4-fluorophenyl)piperazin-1-yl]-5-nitrophenyl]-3-methylbenzamideIC5020000.0 [1]
5-Amino-N-[5-[4-[(2-amino-2-methylpropanoyl)amino]phenyl]-2-(4-methylpiperazin-1-yl)phenyl]-2-chloro-4-fluoro-3-methylbenzamideIC5030.1 [1]
Tert-butyl N-[2-[4-[3-[(5-amino-2-chloro-4-fluoro-3-methylbenzoyl)amino]-4-(4-methylpiperazin-1-yl)phenyl]anilino]-2-oxoethyl]carbamateIC501553.0 [1]
Methyl 4-[3-[(2-chloro-4-fluoro-3-methyl-5-nitrobenzoyl)amino]-4-(4-methylpiperazin-1-yl)phenyl]benzoateIC5092.5 [1]
5-Amino-N-[5-[4-[(2-aminoacetyl)amino]phenyl]-2-(4-methylpiperazin-1-yl)phenyl]-2-chloro-4-fluoro-3-methylbenzamideIC5062.5 [1]
Tert-butyl N-[1-[4-[3-[(5-amino-2-chloro-4-fluoro-3-methylbenzoyl)amino]-4-(4-methylpiperazin-1-yl)phenyl]anilino]-2-methyl-1-oxopropan-2-yl]carbamateIC50113.4 [1]
5-Amino-2-chloro-4-fluoro-3-methyl-N-[2-(4-methylpiperazin-1-yl)-5-pyridin-4-ylphenyl]benzamideIC5018.2 [1]
2-Chloro-4-fluoro-3-methyl-N-[5-nitro-2-(2-pyrrolidin-1-ylethylamino)phenyl]benzamideIC5020000.0 [1]
N-[4-[3-[(5-Amino-2-chloro-4-fluoro-3-methylbenzoyl)amino]-4-(4-methylpiperazin-1-yl)phenyl]phenyl]piperidine-4-carboxamideIC508.5 [1]
2-Chloro-4-fluoro-3-methyl-N-[2-(4-methylpiperazin-1-yl)-5-(4-nitrophenyl)phenyl]-5-nitrobenzamideIC50285.3 [1]
5-Amino-N-[5-[4-(4-aminobutanoylamino)phenyl]-2-(4-methylpiperazin-1-yl)phenyl]-2-chloro-4-fluoro-3-methylbenzamideIC507.6 [1]
5-Acetamido-2-chloro-4-fluoro-3-methyl-N-[2-(4-methylpiperazin-1-yl)-5-(4-nitrophenyl)phenyl]benzamideIC5020000.0 [1]
5-Amino-2-chloro-N-[5-[4-(cyclopropanecarbonylamino)phenyl]-2-(4-methylpiperazin-1-yl)phenyl]-4-fluoro-3-methylbenzamideIC5075.8 [1]
5-Amino-2-chloro-4-fluoro-3-methyl-N-[2-(4-methylpiperazin-1-yl)-5-[4-(2-methylpropanoylamino)phenyl]phenyl]benzamideIC5095.6 [1]
5-Amino-N-[5-(4-benzamidophenyl)-2-(4-methylpiperazin-1-yl)phenyl]-2-chloro-4-fluoro-3-methylbenzamideIC50421.9 [1]
5-Amino-N-[5-(4-aminophenyl)-2-(4-methylpiperazin-1-yl)phenyl]-2-chloro-4-fluoro-3-methylbenzamideIC5088.7 [1]
5-Amino-N-[5-[4-(3-aminopropanoylamino)phenyl]-2-(4-methylpiperazin-1-yl)phenyl]-2-chloro-4-fluoro-3-methylbenzamideIC5050.2 [1]
5-Amino-N-[5-[4-(2-aminopropanoylamino)phenyl]-2-(4-methylpiperazin-1-yl)phenyl]-2-chloro-4-fluoro-3-methylbenzamideIC5015.0 [1]
Tert-butyl N-[1-[4-[3-[(5-amino-2-chloro-4-fluoro-3-methylbenzoyl)amino]-4-(4-methylpiperazin-1-yl)phenyl]anilino]-1-oxopropan-2-yl]carbamateIC5077.9 [1]
5-Acetamido-N-[5-(4-aminophenyl)-2-(4-methylpiperazin-1-yl)phenyl]-2-chloro-4-fluoro-3-methylbenzamideIC503186.0 [1]
4-Fluoro-N-[2-(4-methylpiperazin-1-yl)-5-(4-nitrophenyl)phenyl]-3-nitrobenzamideIC501093.0 [1]
N-[2-(2-Aminoethylamino)-5-nitrophenyl]-2-chloro-4-fluoro-3-methylbenzamideIC5020000.0 [1]
N-[2-(4-Benzylpiperazin-1-yl)-5-nitrophenyl]-2-chloro-4-fluoro-3-methylbenzamideIC5020000.0 [1]
5-Amino-N-[5-[4-(butanoylamino)phenyl]-2-(4-methylpiperazin-1-yl)phenyl]-2-chloro-4-fluoro-3-methylbenzamideIC5076.0 [1]
2-Chloro-4-fluoro-N-[2-(3-imidazol-1-ylpropylamino)-5-nitrophenyl]-3-methylbenzamideIC5020000.0 [1]
Methyl 4-[3-[(5-amino-2-chloro-4-fluoro-3-methylbenzoyl)amino]-4-(4-methylpiperazin-1-yl)phenyl]benzoateIC5070.0 [1]
Tert-butyl N-[4-[4-[3-[(5-amino-2-chloro-4-fluoro-3-methylbenzoyl)amino]-4-(4-methylpiperazin-1-yl)phenyl]anilino]-4-oxobutyl]carbamateIC5080.4 [1]
Phenyl 3-[(4-fluoro-3-nitrobenzoyl)amino]-4-(4-methylpiperazin-1-yl)benzoateIC50483.5 [1]
Phenyl 3-[(3-amino-4-fluorobenzoyl)amino]-4-(4-methylpiperazin-1-yl)benzoateIC5020.0 [1]
Propan-2-yl 3-[(2-chloro-4-fluoro-3-methylbenzoyl)amino]-4-(4-methylpiperazin-1-yl)benzoateIC50263.5 [1]
Propan-2-yl 3-[(4-fluoro-3-nitrobenzoyl)amino]-4-(4-methylpiperazin-1-yl)benzoateIC501171.0 [1]
Cyclohexyl 3-[(2-chloro-4-fluoro-3-methyl-5-nitrobenzoyl)amino]-4-(4-methylpiperazin-1-yl)benzoateIC5020.0 [1]
Cyclohexyl 3-[(4-fluoro-3-nitrobenzoyl)amino]-4-(4-methylpiperazin-1-yl)benzoateIC5020.0 [1]
Ethyl 3-[(2-chloro-4-fluoro-3-methylbenzoyl)amino]-4-(4-methylpiperazin-1-yl)benzoateIC50283.9 [1]
Phenyl 3-[(2-chloro-4-fluoro-3-methylbenzoyl)amino]-4-(4-methylpiperazin-1-yl)benzoateIC50162.4 [1]
Cyclohexyl 3-[(2-chloro-4-fluoro-3-methylbenzoyl)amino]-4-(4-methylpiperazin-1-yl)benzoateIC5020.0 [1]
Cyclohexyl 3-[(3-amino-4-fluorobenzoyl)amino]-4-(4-methylpiperazin-1-yl)benzoateIC5020.0 [1]
Methyl 3-[(2-chloro-4-fluoro-3-methylbenzoyl)amino]-4-(4-methylpiperazin-1-yl)benzoateIC50433.2 [1]
Propan-2-yl 3-[(3-amino-4-fluorobenzoyl)amino]-4-(4-methylpiperazin-1-yl)benzoateIC5020.0 [1]
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References

This online tool may be cited as follows

MLA

"Quest Database™ WD repeat-containing protein 5 Inhibitors (IC50, Ki)." AAT Bioquest, Inc., 8 May. 2024, https://www.aatbio.com/data-sets/wd-repeat-containing-protein-5-inhibitors-ic50-ki.

APA

AAT Bioquest, Inc. (2024, May 8). Quest Database™ WD repeat-containing protein 5 Inhibitors (IC50, Ki). AAT Bioquest. https://www.aatbio.com/data-sets/wd-repeat-containing-protein-5-inhibitors-ic50-ki.
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