Fentanyl succinimidyl ester

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Fax	1-800-609-2943
Email	sales@aatbio.com
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Physical properties

Molecular weight	477.56
Solvent	DMSO

Storage, safety and handling

H-phrase	H303, H313, H333
Hazard symbol	XN
Intended use	Research Use Only (RUO)
R-phrase	R20, R21, R22
Storage	Freeze (< -15 °C); Minimize light exposure
UNSPSC	12171501

Alternative formats

Fentanyl maleimide

Overview SDS Protocol

Molecular weight

477.56

Fentanyl succinmidyl ester can be conveniently used to make biological conjugates of fentanyl that are used to develop fentanyl assays and tests. It specifically reacts with aliphatic amines such as lysine residue of proteins under slightly basic conditions (pH 7.5-9.5).

Calculators

Common stock solution preparation

Table 1. Volume of DMSO needed to reconstitute specific mass of Fentanyl succinimidyl ester to given concentration. Note that volume is only for preparing stock solution. Refer to sample experimental protocol for appropriate experimental/physiological buffers.

	0.1 mg	0.5 mg	1 mg	5 mg	10 mg
1 mM	209.398 µL	1.047 mL	2.094 mL	10.47 mL	20.94 mL
5 mM	41.88 µL	209.398 µL	418.796 µL	2.094 mL	4.188 mL
10 mM	20.94 µL	104.699 µL	209.398 µL	1.047 mL	2.094 mL

Molarity calculator

Enter any two values (mass, volume, concentration) to calculate the third.

Mass (Calculate)		Molecular weight		Volume (Calculate)		Concentration (Calculate)		Moles
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Images

Figure 1. Chemical structure for Fentanyl succinmidyl ester.

References

View all 9 references: Citation Explorer

A fentanyl vaccine constructed upon opsonizing antibodies specific for the Galα1-3Gal epitope.
Authors: Wang, Jiaxing and Ellis, Beverly and Zhou, Bin and Eubanks, Lisa M and Blake, Steven and Janda, Kim D
Journal: Chemical communications (Cambridge, England) (2020): 6551-6554

[Study of the Metabolism of New Drugs of Abuse].
Authors: Kanamori, Tatsuyuki
Journal: Yakugaku zasshi : Journal of the Pharmaceutical Society of Japan (2019): 699-704

A chemically contiguous hapten approach for a heroin-fentanyl vaccine.
Authors: Natori, Yoshihiro and Hwang, Candy S and Lin, Lucy and Smith, Lauren C and Zhou, Bin and Janda, Kim D
Journal: Beilstein journal of organic chemistry (2019): 1020-1031

Use of hepatocytes isolated from a liver-humanized mouse for studies on the metabolism of drugs: application to the metabolism of fentanyl and acetylfentanyl.
Authors: Kanamori, Tatsuyuki and Togawa-Iwata, Yuko and Segawa, Hiroki and Yamamuro, Tadashi and Kuwayama, Kenji and Tsujikawa, Kenji and Inoue, Hiroyuki
Journal: Forensic toxicology (2018): 467-475

In Vitro and In Vivo Metabolite Identification Studies for the New Synthetic Opioids Acetylfentanyl, Acrylfentanyl, Furanylfentanyl, and 4-Fluoro-Isobutyrylfentanyl.
Authors: Watanabe, Shimpei and Vikingsson, Svante and Roman, Markus and Green, Henrik and Kronstrand, Robert and Wohlfarth, Ariane
Journal: The AAPS journal (2017): 1102-1122

Fentanyl-related 4-heteroanilido piperidine OHM3295 augments splenic natural killer activity and induces analgesia through opioid receptor pathways.
Authors: Baker, M L and Brockunier, L L and Bagley, J R and France, C P and Carr, D J
Journal: The Journal of pharmacology and experimental therapeutics (1995): 1285-92

Gamma-scintigraphy and early hepatocellular dysfunction during posttraumatic sepsis.
Authors: McGinty, M P and Stewart, R M and Fabian, M J and Fabian, T C and Proctor, K G
Journal: Surgery (1994): 535-43

Alfentanil pharmacokinetics and metabolism in humans.
Authors: Meuldermans, W and Van Peer, A and Hendrickx, J and Woestenborghs, R and Lauwers, W and Heykants, J and Vanden Bussche, G and Van Craeyvelt, H and Van der Aa, P
Journal: Anesthesiology (1988): 527-34

Association between UGT2B7 gene polymorphisms and fentanyl sensitivity in patients undergoing painful orthognathic surgery.
Authors: Muraoka, Wataru and Nishizawa, Daisuke and Fukuda, Kenichi and Kasai, Shinya and Hasegawa, Junko and Wajima, Koichi and Nakagawa, Taneaki and Ikeda, Kazutaka
Journal: Molecular pain : 1744806916683182