What are the examples of covalent inhibitors?
Posted April 4, 2024
Answer
The most well-known examples of covalent inhibitors include β-lactams, a group of antibacterial agents that includes penicillin and cephalosporin. Other examples include dimethyl fumarate, zanubrutinib, dacomitinib, and ibrutinib.
Additional resources
Covalent Inhibition in Drug Discovery
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